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61.发明公开항암제로 유용한5-(3-아릴-1-피리딜-1Ｈ-피라졸-4-일메틸렌)-티아졸리딘-2,4-디온 유도체 失效用作抗肿瘤剂的5-（3-亚甲基-1-吡咯烷-1-基） - 吡咯-4-基]甲基] - 噻唑烷-2,4-二酮衍生物
公开(公告)号：KR1020060102768A
公开(公告)日：2006-09-28
申请号：KR1020050024691
申请日：2005-03-24
Applicant: 씨제이제일제당 (주) , 한국화학연구원
IPC: C07D417/14
Abstract: 본 발명은 5-(3-아릴-1-피리딜-
1H -피라졸-4-일메틸렌)-티아졸리딘-2,4-디온 유도체 또는 이의 약제학적으로 허용가능한 염과 이의 제조방법 및 이를 유효활성 성분으로 함유하는 항암제 조성물에 관한 것이다.
5-(3-아릴-1-피리딜-1H-피라졸-4-일메틸렌)-티아졸리딘-2,4-디온, 세포분열저해제, CDC25B, 탈인산화효소, 항암제-
公开(公告)号：KR100392073B1
公开(公告)日：2003-07-22
申请号：KR1020000052918
申请日：2000-09-07
Applicant: 한국화학연구원
IPC: A01N43/80
Abstract: PURPOSE: Provided are 5-benzyloxymethyl-1,2-isoxazoline derivatives having an excellent herbicidal activity, its manufacturing method and herbicides containing the derivative as an active ingredient. CONSTITUTION: 5-benzyloxymethyl-1,2-isoxazoline derivative is represented by the formula(I), in which each X1, X2 and X3 represents hydrogen, methyl group, ethyl group, halogen group, methoxy group or nitro group (provided that it is an exception that X1, X2 and X3 are decimals all together); and Y1, Y2 and Y3 are respectively hydrogen or fluorine.
Abstract translation: 目的：提供具有优异除草活性的5-苄氧基甲基-1,2-异恶唑啉衍生物，其制备方法和含有该衍生物作为活性成分的除草剂。 构成：5-苄氧甲基-1,2-异恶唑啉衍生物由式（Ⅰ）表示，其中X1，X2和X3代表氢，甲基，乙基，卤素基，甲氧基或硝基（条件是它 是X1，X2和X3都是小数的例外）; Y1，Y2和Y3分别为氢或氟。
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63.发明公开
公开(公告)号：KR1020010028478A
公开(公告)日：2001-04-06
申请号：KR1019990040742
申请日：1999-09-21
Applicant: 한국화학연구원
IPC: A01N43/00
CPC classification number: A01N43/80 , C07D413/10
Abstract: PURPOSE: Provided is N-(5-isoxazoline methyloxyphenyl)-3,4,5,6-tetrahydrophthalimide derivative which shows a great herbicidal effect only on weed without damaging crops like rice and is useful as a plant growth control agent. CONSTITUTION: A method for manufacturing N-(5-isoxazolinemethyloxyphenyl)-3,4,5,6-tetrahydrophthalimide derivative is characterized by the step of reacting a compound of the formula (2) with nitrileoxide or precursor in the presence of solvents like dichloromethane, tetrahydrofuran, benzene, ethyl ether, and C1-C4 alcohol. In the formula (1), R is an alkyl group of C1-C3, phenyl group, substituted phenyl group, cyano group, carboxylic acid group, or carboxylic acid ester group. The substituted phenyl group is a phenyl group having the same or different 1-3 substituents among an alkyl group of C1-C3, haloalkyl group of C1-C3, methylsulfonyl group, alkoxy group of C1-C3, halogen atom, cyano group, nitro group, carboxylic acid group, and carboxylic acid ester group.
Abstract translation: 目的：提供N-（5-异恶唑啉甲氧基苯基）-3,4,5,6-四氢邻苯二甲酰亚胺衍生物，其仅在杂草上显示出很好的除草效果，而不损害作物如水稻，并且可用作植物生长调节剂。 构成：制备N-（5-异恶唑啉甲氧基苯基）-3,4,5,6-四氢邻苯二甲酰亚胺衍生物的方法的特征在于使式（2）的化合物与硝酸氧化物或前体在溶剂如二氯甲烷 ，四氢呋喃，苯，乙醚和C 1 -C 4醇。 式（1）中，R为C1-C3，苯基，取代苯基，氰基，羧酸基或羧酸酯基的烷基。 取代的苯基是C1-C3的烷基，C1-C3的卤代烷基，甲基磺酰基，C1-C3的烷氧基，卤素原子，氰基，硝基中的1-3个取代基相同或不同的苯基 基团，羧酸基和羧酸酯基。
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公开(公告)号：KR1020000013379A
公开(公告)日：2000-03-06
申请号：KR1019980032207
申请日：1998-08-07
Applicant: 한국화학연구원
IPC: C07D261/20
Abstract: PURPOSE: A hexahydro-1,2-benzisoxazol derivative is excellent in weeding activity and innoxious to paddy rice. CONSTITUTION: A hexahydro-1,2-benzisoxazol derivative represented by the following formula, wherein Xn is a hydrogen, a C1-C3 alkyl group, a C2-C4 alkenyl group, a C2-C4 alkynyl group, a C1-C3 alkoxyl group, a C1-C3 haloalkyl group, a C1-C3 thioalkyl group, a C1-C3 alkylsulfenyl group, a C1-C3 alkylsulfonyl group, a halogen group, a nitro group, a nitrile group, or a composite substituent thereof; Yn is a hydrogen, a C1-C6 alkyl group, a halogen group, a nitro group, a nitrile group, or a composite substituent thereof; Yn is a hydrogen, a C1-C3 alkyl group, a halogen group, a nitro group, a nitrile group, or a composite substituent thereof; and R is a hydrogen or a methyl group.
Abstract translation: 目的：六氢-1,2-苯并异恶唑衍生物具有优良的除草活性和无害水稻。 构成：由下式表示的六氢-1,2-苯并异恶唑衍生物，其中Xn为氢，C1-C3烷基，C2-C4烯基，C2-C4炔基，C1-C3烷氧基 C1-C3卤代烷基，C1-C3硫代烷基，C1-C3烷基亚磺酰基，C1-C3烷基磺酰基，卤素基，硝基，腈基或其复合取代基; Yn为氢，C1-C6烷基，卤素基，硝基，腈基或其复合取代基; Yn为氢，C1-C3烷基，卤素基，硝基，腈基或其复合取代基; R为氢或甲基。
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公开(公告)号：KR1019960034181A
公开(公告)日：1996-10-22
申请号：KR1019950007218
申请日：1995-03-31
Applicant: 한국화학연구원
IPC: C07D239/28 , C07D213/89 , C07D239/30 , C07D239/42 , C07D241/52
Abstract: 본 발명은 방향족 헤테로고리 아민 N-옥사이드의 제조방법에 관한 것으로서, 더욱 상세하게는 다음 구조식(Ⅲ)로 표시되는 방향족 헤테로고리 아민을 불화수소(HF) 수용액 촉매, 디메틸포름아미드와 메탄을 혼합용매 하에서 m-클로로과벤조산 산화제로 반응시켜, 짧은시간에 높은 수율로 다음 구조식(Ⅰ)로 표시되는 방향족 헤테로고리 아민 N-옥사이드를 제조하는 신규 제조방법에 관한 것이다.
상기 식에서, X 및 Y는 각각 같거나 다른 것으로서 CH 또는 N이며, R은 클로로, 카르복실산, 아미노, 옥소, C
1 ~C
4 의 알킬 또는 리보스(ribose)이며, n은 치환기 R의 갯수로서 1 내지 3의정수이다.-
Patent Agency Ranking
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公开(公告)号：KR1019950006923B1
公开(公告)日：1995-06-26
申请号：KR1019920009493
申请日：1992-06-01
Applicant: 한국화학연구원
IPC: A01N43/10
Abstract: A 2,3-dihydrothiophenyl cyclohexane-1,3-dione derivative of formula (I) for using herbicide and plant growth regulating agent is prepd. by reacting the compound of formula (II) and H2NOR3˜HCl in an inert organic solvent. In the formula, R1 is H or C1˜C4 alkyl, R2 is C1˜C6 alkenyl, C2˜C6 alkynyl or C1˜C6 haloalkyl, R3 is H, C1˜C6 alkyl, C2˜C6 alkenyl, C2˜C6 alkynyl, C1˜C6 haloalkyl, C2˜C6 haloalkenyl, C2˜C6 haloalkynyl, C1˜C6 alkoxyalkyl, C1˜C6 alkylthioalkyl, benzyl or haloalkanoyl group.
Abstract translation: 使用除草剂和植物生长调节剂的式（I）的2,3-二氢噻吩环己烷-1,3-二酮衍生物是制备的。 通过使式（II）化合物和H 2 NOR 3〜HCl在惰性有机溶剂中反应。 在该式中，R 1为H或C 1〜C 4烷基，R 2为C 1〜C 6烯基，C 2〜C 6炔基或C 1 -C 6卤代烷基，R 3为H，C 1〜C 6烷基，C 2〜C 6烯基，C 2〜C 6炔基，C 1 C 6卤代烷基，C 2〜C 6卤代烯基，C 2〜C 6卤代炔基，C 1 -C 6烷氧基烷基，C 1〜C 6烷硫基烷基，苄基或卤代烷酰基。
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