公开(公告)号：CA2482809A1

公开(公告)日：2003-11-13

申请号：CA2482809

申请日：2003-04-30

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  TORMO I BLASCO JORDI ,  STRATHMANN SIEGFRIED ,  MUELLER BERND ,  GEWEHR MARKUS ,  BLETTNER CARSTEN ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  SCHWOEGLER ANJA ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  LORENZ GISELA ,  SCHAEFER PETER ,  STIERL REINHARD

IPC: A01N43/90 ,  C07C69/65 ,  C07D487/04 ,  C07D239/00 ,  C07D249/00 ,  C07C69/612 ,  C07C69/738

Abstract: Disclosed are a method for producing fungicidal triazolopyrimidine compounds , agents containing said compounds, and the use thereof for controlling harmfu l fungi. Also disclosed are triazolopyrimidines of formula (I), in which the substituents have the following meaning: L1 represents alkyl; L2 represents halogen; L3 represents hydrogen or halogen; X represents halogen, cyano, alkyl, alkoxy, or haloalkoxy; R1, R2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, alkenyl, alkadienyl, alkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-unit to ten-unit saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group O, N, or S. R1 and R2 can also form a five-unit or six-unit ring along with the nitrogen at om to which they are linked. Said ring can be interrupted and/or substituted by an atom from the group O, N, and S while R1 and/or R2 can be substituted according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing said compounds, and the use thereof for controlling harmful fungi.

公开(公告)号：AU2005266555B2

公开(公告)日：2011-09-08

申请号：AU2005266555

申请日：2005-07-22

Applicant: BASF AG

Inventor： GROTE THOMAS ,  MULLER BERND ,  STIERL REINHARD ,  RHEINHEIMER JOACHIM ,  SCHWOGLER ANJA ,  GRAMMENOS WASSILIOS ,  SCHERER MARIA ,  SCHOFL ULRICH ,  GEWEHR MARKUS ,  SCHAFER PETER ,  STRATHMANN SIEGFRIED ,  RETHER JAN ,  BLETTNER CARSTEN ,  HUNGER UDO ,  SCHIEWECK FRANK ,  KOHLE HARALD

IPC: C07D401/04 ,  A01N43/54

Abstract: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type, whereby: k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R, independent of one another, represents halogen, OH, CN, NO C-C alkyl, C-C alkyl halide, C-C alkoxy, C-C alkoxy halide, C-C alkenyl, C-C alkynyl, C-C cycloalkyl, C-C alkoxy-C-C alkyl, amino, phenoxy, which is optionally substituted by halogen or C-C alkyl, NHR, NR, C(R)=N-OR, S(=O)A or C(=O)A, or two radicals R bound to adjacent carbon atoms can, together, also represent a group -O-Alk-O-, wherein Alk represents a linear or branched C-C alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R represents C-C alkyl halide, C-C alkoxy, C-C alkoxy halide, hydroxy, halogen, CN or NO; whereby R can also represent hydrogen or C-C alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R represents a radical that differs from halogen, C-C alkyl, C-C alkoxy and C-C alkyl halide, and; R represents C-C alkyl.

公开(公告)号：NZ556448A

公开(公告)日：2010-12-24

申请号：NZ55644806

申请日：2006-01-30

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MULLER BERND ,  NAVE BARBARA ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  JABS THORSTEN ,  BLETTNER CARSTEN

IPC: A61K31/506 ,  A61K31/505 ,  A61P35/00 ,  C07D239/42 ,  C07D239/48 ,  C07D401/04 ,  C07D403/04 ,  C07D417/04

Abstract: Disclosed is the use of substituted 5-phenyl pyrimidines of the formula I and their pharmaceutically acceptable salts for the manufacture of a medicament for therapy of cancer or cancerous diseases, wherein X is a group of the formula NR1R2; Y is a radical selected from the group consisting of halogen, cyano, alkyl, and alkoxy; and wherein the other substituents are as defined herein. Also disclosed is a pharmaceutical composition for therapy of cancer or cancerous diseases which comprises a 5-phenyl pyrimidine derivative as defined above or a pharmaceutically acceptable salt thereof and a pharmaceutically acceptable carrier.

公开(公告)号：UA84569C2

公开(公告)日：2008-11-10

申请号：UAA200601927

申请日：2004-07-15

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  TORMO I BLASCO JORDI ,  GUPSER ANDREAS ,  BLETTNER CARSTEN ,  WAGNER OLIVER ,  SCHOEFL ULRICH ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA

IPC: C07D239/42

公开(公告)号：EA010566B1

公开(公告)日：2008-10-30

申请号：EA200600212

申请日：2004-07-15

Applicant: BASF AG

Inventor： SCHWOGLER ANJA ,  GEWEHR MARCUS ,  MULLER BERND ,  GROTE THOMAS ,  GRAMMENOS WAASSILIOS ,  TORMO I BLASCO JORDI ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  BLETTNER CARSTEN ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  WAGNER OLIVER ,  STIERL REINHARD ,  SCHOFL ULRICH ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA

IPC: C07D239/42

Abstract: Изобретениеотноситсяк 2-замещеннымпиримидинамформулы Iвкоторойиндекс n изаместители Rдо R, атакже L имеютуказанныев описаниизначенияи Rсоответствуетформуламвкоторых R, X и Rимеютуказанныев описаниизначения; атакжек способуихполучения, ксодержащимихпестициднымсредствами ихприменениюв качествепестицидов.

公开(公告)号：NZ546218A

公开(公告)日：2008-07-31

申请号：NZ54621804

申请日：2004-09-10

Applicant: BASF AG

Inventor： GRAMMENOS WASSILIOS ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  WAGNER OLIVER ,  GOTZ NORBERT ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

IPC: C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12 ,  C07C311/18 ,  A01N41/06

Abstract: Disclosed are 4-piridinylmethylsulfonamide derivatives of the formula I wherein the substituents are defined within the specification. Also disclosed is a method of controlling phytopathogenic harmful fungi, which comprises treating the fungi or the materials, plants, the soil or seeds to be protected against fungal attack with an effective amount of the above compounds of formula I.

公开(公告)号：BRPI0514924A

公开(公告)日：2008-06-24

申请号：BRPI0514924

申请日：2005-09-05

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  MUELLER BERND ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  SCHWOEGLER ANJA ,  RHEINHEIMER JOACHIM ,  BLETTNER CARSTEN ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  WAGNER OLIVER ,  RETHER JAN ,  STRATHMANN SIEGFRIED ,  STIERL REINHARD ,  SCHERER MARIA

IPC: C07D213/82 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  C07D231/14 ,  C07D277/56

Abstract: The invention relates to (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I) and to salts of said anilides that can be used for agricultural purposes for controlling pathogenic fungi. In said formula, the variables are defined as follows: A represents a phenyl or at least a monounsaturated 5- or 6-membered heterocycle comprising 1, 2 or 3 heteroatoms, selected from N, O, S, S(-O) and S(-O) 2 as ring members, whereby phenyl and the monounsaturated 5- or 6-membered heterocycle can be unsubstituted or can be substituted according to the description; B represents a group of general formula (II), in which the variables R 3 , R 4 , R 5 and the index m are defined as cited in the claims and the description; Y represents oxygen or sulphur, R 1 represents H, OH, alkyl, cycloalkyl, alkoxy, haloalkyl, halocycloalkyl or haloalkoxy; R 2 represents halogen, nitro, CN, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, haloalkyl, halocycloalkyl, haloalkenyl, haloalkynyl or haloalkoxy; and n represents 0, 1, 2, 3 or 4; and salts that can be used for agricultural purposes. The invention also relates to the use of the (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I), to a method for controlling pathogenic fungi and to a crop protection agent containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound.

公开(公告)号：BRPI0514067A

公开(公告)日：2008-05-27

申请号：BRPI0514067

申请日：2005-07-28

Applicant: BASF AG

Inventor： BLETTNER CARSTEN ,  DIETZ JOCHEN ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHAMANN SIEGFRIED ,  STIERL REINHARD ,  SCHWOEGLER ANJA ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  A01N20060101 ,  A01N43/50 ,  A01N43/54 ,  A01N43/653 ,  A01N43/84 ,  A01N47/04 ,  A01N47/14 ,  A01N47/24 ,  A01N47/38 ,  A01N57/12 ,  A01N59/20

Abstract: Fungicidal mixtures, comprising as active components 1) a 5-chloro-6-phenyl-7-heterocyclylaminotriazolopyrimidine of the formula I, in which D together with the nitrogen atom forms a pyrrolidine, piperidine or azepine ring, which rings are unsubstituted or substituted by one or two methyl groups or by an ethyl, propyl or butyl group; and L is methyl, fluorine or chlorine; and 2) at least one active compound II selected from the following groups: A) azoles; B) strobilurins; C) acylalanines; D) amine derivatives; E) anilinopyrimidines; F) dicarboximides; G) cinnamides and analogs; H) antibiotics; K) dithiocarbamates; L) heterocyclic compounds according to the description; M) sulfur and copper fungicides; N) nitrophenyl derivatives; O) phenylpyrroles; P) sulfenic acid derivatives; Q) other fungicides according to the description; or R) growth retardants; in a synergistically effective amount, novel triazolopyrimidines, methods for controlling harmful fungi using compounds or mixtures of a compound I with an active compound of groups A) to R) and the use of the compounds I with the active compounds of groups A) to R) for preparing such mixtures, and also compositions comprising these compounds or mixtures.

公开(公告)号：MA29431B1

公开(公告)日：2008-05-02

申请号：MA30200

申请日：2007-09-10

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  DIETZ JOCHEN ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GRAMMENOS WASSILIOS ,  HUENGER UDO ,  MUELLER BERND ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  LOHMANN JAN KLAAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  STRATHMANN SIEGFRIED ,  STIERL REINHARD

IPC: C07D231/14 ,  A01N43/56

Abstract: L'INVENTION CONCERNE DES ANILIDES D'ACIDE CARBOXYLIQUE PYRAZOLE DE FORMULE (I) DANS LAQUELLE LES VARIABLES ONT LES SIGNIFICATIONS SUIVANTES : N EST ZÉRO OU 2; M SIGNIFIE 2 OU 3; X1 DÉSIGNE FLUORE OU CHLORE; X2 REPRÉSENTE HALOGÈNE; Y SIGNIFIE CN, NO2, ALKYLE C1-C4, HALOGÉNURE D'ALKYLE C1-C4, MÉTHOXY OU MÉTHYLTHIO; P EST ZÉRO OU 1; R1 DÉSIGNE FLUORE, CHLORE, BROME, ALKYLE C1-C4, HALOGÉNURE D'ALKYLE C1-C4; R2 REPRÉSENTE HYDROGÈNE OU HALOGÈNE; R3 DÉSIGNE HYDROGÈNE, MÉTHYLE OU ÉTHYLE; W REPRÉSENTE O OU S; À CONDITION QUE, LORSQUE A) W = O, R1 = MÉTHYLE ET R3 REPRÉSENTE HYDROGÈNE, R2 NE SIGNIFIE PAS FLUOR, OU BIEN LORSQUE B) W = O, N = 0, M = 2, P = 0, R2 ET R3 REPRÉSENTENT HYDROGÈNE, R1 NE SIGNIFIE PAS TRIFLUOROMÉTHYLE OU DIFLUOROMÉTHYLE. LA PRÉSENTE INVENTION PORTE ÉGALEMENT SUR DES PROCÉDÉS POUR RÉALISER CES COMPOSÉS, SUR DES AGENTS LES CONTENANT ET SUR DES PROCÉDÉS POUR LES UTILISER DANS LA LUTTE ANTIFONGIQUE.

公开(公告)号：BRPI0513032A

公开(公告)日：2008-04-22

申请号：BRPI0513032

申请日：2005-07-06

Applicant: BASF AG

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

Abstract: Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R 1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R 2 is hydrogen or a group R 1 , R 1 and R 2 together with the nitrogen atom, to which they are attached, may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and which may comprise one to three further heteroatoms from the groups consisting of O, N and S as ring member and/or may be substituted according to the description; L is fluorine, chlorine or methyl; X is cyano, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy or C 1 -C 2 -haloalkoxy, where X is not methyl if R 1 and R 2 together are n-pentylene or 3-methyl-n-pentylene and L is fluorine, or R 1 and R 2 together are 3-methyl-n-pentylene and L is chlorine; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.