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公开(公告)号:CA2382751A1
公开(公告)日:2000-11-30
申请号:CA2382751
申请日:2000-05-24
Applicant: COR THERAPEUTICS INC
Inventor: CLIZBE LANE , SONG YONGHONG , MARLOWE CHARLES , ZHU BING-YAN , SU TING , SCARBOROUGH ROBERT M
IPC: C07D233/61 , A61K31/165 , A61K31/167 , A61K31/18 , A61K31/198 , A61K31/216 , A61K31/277 , A61K31/341 , A61K31/40 , A61K31/404 , A61K31/415 , A61K31/422 , A61K31/4402 , A61K31/472 , A61K33/22 , A61P7/02 , A61P7/04 , A61P9/00 , A61P9/04 , A61P9/08 , A61P9/10 , A61P43/00 , C07C311/46 , C07C317/32 , C07D209/08 , C07D213/56 , C07D217/22 , C07D231/12 , C07D295/16 , C07D307/54 , C07D307/68 , C07D413/04 , C07D521/00
Abstract: The present application relates to compounds of the general formula A-Y-D-E- G- J-K-L, wherein A, Y, D, E, G, J, K and L have the meanings given in the description, having activity against mammalian factor Xa. The compounds are useful in vitroor in vivofor preventing or treating coagulation disorders.
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公开(公告)号:CA2374788A1
公开(公告)日:2000-11-30
申请号:CA2374788
申请日:2000-05-24
Applicant: COR THERAPEUTICS INC
Inventor: ZHU BING-YAN , SCARBOROUGH ROBERT M
IPC: A61K31/155 , A61K31/18 , A61K31/275 , A61K31/401 , A61K31/402 , A61K31/451 , A61P7/02 , A61P9/00 , A61P9/04 , A61P9/10 , C07C311/46 , C07D207/16 , C07D211/60 , C07D241/04 , C07D243/08 , C07D401/04 , C07D403/04 , C07D413/04 , A61K31/40 , A61P7/00 , C07C311/39
Abstract: Compounds, e.g. described in Table (1), their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful in vitroor in vivofor preventing or treating coagulation disorders.
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公开(公告)号:AU4166400A
公开(公告)日:2000-08-29
申请号:AU4166400
申请日:2000-02-11
Applicant: COR THERAPEUTICS INC
Inventor: SONG YOUNGHONG , SCARBOROUGH ROBERT M JR , ZHU BING-YAN
IPC: C07D295/14 , A61K31/18 , A61K31/192 , A61K31/195 , A61K31/216 , A61K31/341 , A61K31/40 , A61K31/41 , A61K31/415 , A61K31/4174 , A61K31/44 , A61K31/4409 , A61K31/472 , A61K31/4725 , A61K31/495 , A61K31/505 , A61K31/517 , A61P7/00 , A61P7/02 , A61P7/04 , A61P9/00 , A61P9/10 , A61P11/00 , A61P31/04 , A61P43/00 , C07C257/18 , C07C311/29 , C07C311/46 , C07C311/51 , C07D213/56 , C07D213/58 , C07D213/70 , C07D213/74 , C07D213/75 , C07D217/22 , C07D231/12 , C07D233/61 , C07D239/42 , C07D239/94 , C07D257/04 , C07D295/16 , C07D307/54 , C07D401/12 , C07D521/00
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公开(公告)号:CA2299610A1
公开(公告)日:1999-02-18
申请号:CA2299610
申请日:1998-08-11
Applicant: COR THERAPEUTICS INC
Inventor: SCARBOROUGH ROBERT M , ZHU BING-YAN
Abstract: Novel compounds, their salts and compositions related thereto having activity against mammalian factory Xa are disclosed. The compounds are useful in vitro or vivo for preventing or treating coagulation disorders and have formula (I).
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公开(公告)号:AU6896298A
公开(公告)日:1998-11-11
申请号:AU6896298
申请日:1998-04-13
Applicant: COR THERAPEUTICS INC
Inventor: ZHU BING-YAN , SCARBOROUGH ROBERT M JR , SU TING
IPC: A61K38/00 , A61K8/63 , A61P7/02 , A61P9/02 , A61P9/10 , A61Q7/00 , A61Q7/02 , C07K5/02 , C07K5/06 , C07K5/062 , C07K5/072 , C07K5/078 , A61K38/05
Abstract: Novel compounds, their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful in vitro or in vivo for preventing or treating coagulation disorders.
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公开(公告)号:CA2268264A1
公开(公告)日:1998-04-23
申请号:CA2268264
申请日:1997-10-10
Applicant: COR THERAPEUTICS INC
Inventor: ZHU BING-YAN , SCARBOROUGH ROBERT M
IPC: A61K38/00 , A61P7/02 , A61P9/02 , A61P9/10 , C07D417/12 , C07F5/02 , C07K5/06 , C07D417/14 , A61K31/425
Abstract: Novel compounds, their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful in vitro or in vivo for preventing or treating coagulation disorders.
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公开(公告)号:AU6590296A
公开(公告)日:1996-12-30
申请号:AU6590296
申请日:1996-06-05
Applicant: COR THERAPEUTICS INC
Inventor: MARLOWE CHARLES K , SCARBOROUGH ROBERT M JR , LAIBELMAN ALAN M , SINHA UMA , ZHU BING-YAN
IPC: A61K38/00 , A61P7/02 , C07C279/24 , C07C281/06 , C07C309/30 , C07C335/38 , C07K5/06 , C07K5/068 , C07K5/072 , C07K5/08 , A61K38/55
Abstract: Novel compounds, their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful in vitro or in vivo for preventing or treating coagulation disorders.
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公开(公告)号:CA2224180A1
公开(公告)日:1996-12-19
申请号:CA2224180
申请日:1996-06-05
Applicant: COR THERAPEUTICS INC
Inventor: SCARBOROUGH ROBERT M , ZHU BING-YAN , SINHA UMA , LAIBELMAN ALAN M , MARLOWE CHARLES K
IPC: C07D277/24 , A61K31/42 , A61K31/421 , A61K31/423 , A61K31/425 , A61K31/426 , A61K31/428 , A61K38/00 , A61P7/02 , A61P9/00 , C07C311/64 , C07D263/14 , C07D263/56 , C07D277/68 , C07K5/06 , C07K5/065 , C07K5/072 , C07K5/078 , C07K5/08 , C07K5/09 , C07K5/027 , A61K38/06 , C07K5/097 , G01N1/28
Abstract: Novel compounds, their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful in vitro or in vivo for preventing or treating coagulation disorders.
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公开(公告)号:AU1454602A
公开(公告)日:2002-04-08
申请号:AU1454602
申请日:2001-10-01
Applicant: COR THERAPEUTICS INC
Inventor: ZHANG PENGLIE , LI WENHAO , HUANG WENRONG , WANG LINGYAN , JIA ZHAOZHONG JON , SCARBOROUGH ROBERT M JR , ZHU BING-YAN
IPC: A61P7/02 , C07D239/91 , C07D401/04 , C07D401/14 , C07D409/14 , C07D487/04 , A61K31/517 , A61K31/519
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公开(公告)号:AU1128102A
公开(公告)日:2002-04-08
申请号:AU1128102
申请日:2001-10-01
Applicant: COR THERAPEUTICS INC
Inventor: ZHU BING-YAN , HUANG WENRONG , ZHANG PENGLIE , JIA ZHAOZHONG JON , BAO LIANG , WU YANHONG , SCARBOROUGH ROBERT M JR
IPC: A61P7/02 , C07D213/75 , C07D401/12 , C07D401/14 , C07D401/00
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