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公开(公告)号:WO2005074603A2
公开(公告)日:2005-08-18
申请号:PCT/US2005003196
申请日:2005-02-03
Applicant: ABBOTT LAB , WISHART NEIL , FRIEDMAN MICHAEL , ARNOLD LEE D , YANG BRYANT , FIX-STENZEL SHANNON R , ERICSSON ANNA , MICHAELIDES MICHAEL R , QIAN XIAO-DONG , HOLMES JAMES H , STEINMAN DOUGLAS H , TIAN ZHENGPING , WITTENBERGER STEVEN J
Inventor: WISHART NEIL , FRIEDMAN MICHAEL , ARNOLD LEE D , YANG BRYANT , FIX-STENZEL SHANNON R , ERICSSON ANNA , MICHAELIDES MICHAEL R , QIAN XIAO-DONG , HOLMES JAMES H , STEINMAN DOUGLAS H , TIAN ZHENGPING , WITTENBERGER STEVEN J
IPC: C07D487/04
CPC classification number: C07D487/04
Abstract: A compound of Formula (I), wherein the substituents are as defined herein, which are useful as kinase inhibitors.
Abstract translation: 式(I)的化合物,其中取代基如本文所定义,其可用作激酶抑制剂。
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公开(公告)号:EP1730148A4
公开(公告)日:2009-08-19
申请号:EP05722668
申请日:2005-02-03
Applicant: ABBOTT LAB
Inventor: WISHART NEIL , FRIEDMAN MICHAEL , ARNOLD LEE D , YANG BRYANT , FIX-STENZEL SHANNON R , ERICSSON ANNA , MICHAELIDES MICHAEL R , QIAN XIAO-DONG , HOLMES JAMES H , STEINMAN DOUGLAS H , TIAN ZHENGPING , WITTENBERGER STEVEN J
IPC: C07D487/04 , A61K31/381 , A61K31/519 , A61K31/5377 , C07D239/70 , C07D263/54 , C07D295/03 , C07D513/06
CPC classification number: C07D487/04
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公开(公告)号:AT228122T
公开(公告)日:2002-12-15
申请号:AT00905758
申请日:2000-01-27
Applicant: ABBOTT LAB
Inventor: CURTIN MICHAEL L , DAI YUJIA , DAVIDSEN STEVEN K , HEYMAN HOWARD R , HOLMES JAMES H , MICHAELIDES MICHAEL R , STEINMAN DOUGLAS H
IPC: A61K31/341 , A61K31/357 , A61K31/40 , A61K31/421 , A61P1/02 , A61P1/04 , A61P17/02 , A61P19/02 , A61P19/10 , A61P27/02 , A61P29/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07D207/09 , C07D207/14 , C07D207/48 , C07D263/04 , C07D307/14 , C07D317/28 , A61K31/335
Abstract: Compounds having the formula are matrix metalloproteinase inhibitors. Also disclosed are matrix metalloproteinase-inhibiting compositions and methods of inhibiting matrix metalloproteinase in a mammal.
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公开(公告)号:BR0007278A
公开(公告)日:2001-11-27
申请号:BR0007278
申请日:2000-01-27
Applicant: ABBOTT LAB
Inventor: CURTIN MICHAEL L , DAI YUJIA , DAVIDSEN STEVEN K , HEYMAN HOWARD R , HOLMES JAMES H , MICHAELIDES MICHAEL R , STEINMAN DOUGLAS H
IPC: A61K31/341 , A61K31/357 , A61K31/40 , A61K31/421 , A61P1/02 , A61P1/04 , A61P17/02 , A61P19/02 , A61P19/10 , A61P27/02 , A61P29/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07D207/09 , C07D207/14 , C07D207/48 , C07D263/04 , C07D307/14 , C07D317/28 , A61K31/335
Abstract: Compounds having the formula are matrix metalloproteinase inhibitors. Also disclosed are matrix metalloproteinase-inhibiting compositions and methods of inhibiting matrix metalloproteinase in a mammal.
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公开(公告)号:PT1147101E
公开(公告)日:2003-04-30
申请号:PT00905758
申请日:2000-01-27
Applicant: ABBOTT LAB
Inventor: STEINMAN DOUGLAS H , DAVIDSEN STEVEN K , CURTIN MICHAEL L , DAI YUJIA , HEYMAN HOWARD R , HOLMES JAMES H , MICHAELIDES MICHAEL R
IPC: A61K31/341 , A61K31/357 , A61K31/40 , A61K31/421 , A61P1/02 , A61P1/04 , A61P17/02 , A61P19/02 , A61P19/10 , A61P27/02 , A61P29/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07D207/09 , C07D207/14 , C07D207/48 , C07D263/04 , C07D307/14 , C07D317/28 , A61K31/335
Abstract: Compounds having the formula are matrix metalloproteinase inhibitors. Also disclosed are matrix metalloproteinase-inhibiting compositions and methods of inhibiting matrix metalloproteinase in a mammal.
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公开(公告)号:NO20013669A
公开(公告)日:2001-09-27
申请号:NO20013669
申请日:2001-07-26
Applicant: ABBOTT LAB
Inventor: CURTIN MICHAEL L , DAI YUJIA , DAVIDSEN STEVEN K , HEYMAN HOWARD R , HOLMES JAMES H , MICHAELIDES MICHAEL R , STEINMAN DOUGLAS H
IPC: A61K31/341 , A61K31/357 , A61K31/40 , A61K31/421 , A61P1/02 , A61P1/04 , A61P17/02 , A61P19/02 , A61P19/10 , A61P27/02 , A61P29/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07D207/09 , C07D207/14 , C07D207/48 , C07D263/04 , C07D307/14 , C07D317/28 , A61K31/335
CPC classification number: C07D263/04 , C07D207/09 , C07D207/48 , C07D307/14 , C07D317/28
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公开(公告)号:ES2187443T3
公开(公告)日:2003-06-16
申请号:ES00905758
申请日:2000-01-27
Applicant: ABBOTT LAB
Inventor: CURTIN MICHAEL L , DAI YUJIA , DAVIDSEN STEVEN K , HEYMAN HOWARD R , HOLMES JAMES H , MICHAELIDES MICHAEL R
IPC: A61K31/341 , A61K31/357 , A61K31/40 , A61K31/421 , A61P1/02 , A61P1/04 , A61P17/02 , A61P19/02 , A61P19/10 , A61P27/02 , A61P29/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07D207/09 , C07D207/14 , C07D207/48 , C07D263/04 , C07D307/14 , C07D317/28 , A61K31/335
Abstract: Compounds having the formula are matrix metalloproteinase inhibitors. Also disclosed are matrix metalloproteinase-inhibiting compositions and methods of inhibiting matrix metalloproteinase in a mammal.
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公开(公告)号:HU0105477A2
公开(公告)日:2002-05-29
申请号:HU0105477
申请日:2000-01-27
Applicant: ABBOTT LAB
Inventor: CURTIN MICHAEL L , DAI YUJIA , DAVIDSEN STEVEN K , HEYMAN HOWARD R , HOLMES JAMES H , MICHAELIDES MICHAEL R , STEINMAN DOUGLAS H
IPC: A61K31/341 , A61K31/357 , A61K31/40 , A61K31/421 , A61P1/02 , A61P1/04 , A61P17/02 , A61P19/02 , A61P19/10 , A61P27/02 , A61P29/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07D207/09 , C07D207/14 , C07D207/48 , C07D263/04 , C07D307/14 , C07D317/28
Abstract: Compounds having the formula are matrix metalloproteinase inhibitors. Also disclosed are matrix metalloproteinase-inhibiting compositions and methods of inhibiting matrix metalloproteinase in a mammal.
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公开(公告)号:SK10582001A3
公开(公告)日:2001-12-03
申请号:SK10582001
申请日:2000-01-27
Applicant: ABBOTT LAB
Inventor: CURTIN MICHAEL L , DAI YUJIA , DAVIDSEN STEVEN K , HEYMAN HOWARD R , HOLMES JAMES H , MICHAELIDES MICHAEL R , STEINMAN DOUGLAS H
IPC: A61K31/341 , A61K31/357 , A61K31/40 , A61K31/421 , A61P1/02 , A61P1/04 , A61P17/02 , A61P19/02 , A61P19/10 , A61P27/02 , A61P29/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07D207/09 , C07D207/14 , C07D207/48 , C07D263/04 , C07D307/14 , C07D317/28 , A61K31/335
Abstract: Compounds having the formula are matrix metalloproteinase inhibitors. Also disclosed are matrix metalloproteinase-inhibiting compositions and methods of inhibiting matrix metalloproteinase in a mammal.
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公开(公告)号:AU764383B2
公开(公告)日:2003-08-14
申请号:AU2739100
申请日:2000-01-27
Applicant: ABBOTT LAB
Inventor: CURTIN MICHAEL L , DAI YUJIA , DAVIDSEN STEVEN K , HEYMAN HOWARD R , HOLMES JAMES H , MICHAELIDES MICHAEL R , STEINMAN DOUGLAS H
IPC: A61K31/341 , A61K31/357 , A61K31/40 , A61K31/421 , A61P1/02 , A61P1/04 , A61P17/02 , A61P19/02 , A61P19/10 , A61P27/02 , A61P29/00 , A61P35/00 , A61P35/04 , A61P43/00 , C07D207/09 , C07D207/14 , C07D207/48 , C07D263/04 , C07D307/14 , C07D317/28 , A61K31/335
Abstract: Compounds having the formula are matrix metalloproteinase inhibitors. Also disclosed are matrix metalloproteinase-inhibiting compositions and methods of inhibiting matrix metalloproteinase in a mammal.
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