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公开(公告)号:ZA969402B
公开(公告)日:1998-05-08
申请号:ZA969402
申请日:1996-11-08
Applicant: BASF AG
Inventor: KLING ANDREAS , JANSSEN BERND , AMBERG WILHELM , HAUPT ANDREAS , RITTER KURT , BUSCHMANN ERNST , BERNARD HARALD , MUELLER STEFAN , ZIERKE THOMAS , BARLOZZARI TERESA , ARRUDA MONIKA DE , ROBINSON SIMON
Abstract: Novel peptides of the formulaA-B-D-E-F-L,wherein A, B, D, E, F, and L have the meanings stated in the specification, and their preparation are disclosed. The novel compounds are suitable for controlling diseases.
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公开(公告)号:NO982100A
公开(公告)日:1998-05-08
申请号:NO982100
申请日:1998-05-08
Applicant: BASF AG
Inventor: KLING ANDREAS , JANSSEN BERND , AMBERG WILHELM , HAUPT ANDREAS , RITTER KURT , BUSCHMANN ERNST , BERNARD HARALD , MUELLER STEFAN , ZIERKE THOMAS , BARLOZZARI TERESA , ARRUDA MONIKA DE , ROBINSON SIMON
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公开(公告)号:BG61610B2
公开(公告)日:1998-01-30
申请号:BG10096196
申请日:1996-11-06
Applicant: BASF AG
Inventor: AMBERG WILHELM , BERNARD HARALD , BUSCHMANN ERNST , HAUPT ANDREAS , JANITSCHKE LOTHAR , JANSSEN BERND , KARL ULRICH , KLING ANDREAS , MUELLER STEFAN , DE POTZOLLI BERND , RITTER KURT , THYES MARCO , ZIERKE THOMAS
Abstract: The invention relates to compound Me2Val - Val - MeVal - Pro- Pro - NHBzl.HCl showing antineoplastic activity. It is producedform a compound with the formulaZ - Val - Val - MeVal - Pro - OR1where Z and R1 have the meanings listed in the description.
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公开(公告)号:ZA966372B
公开(公告)日:1998-01-26
申请号:ZA966372
申请日:1996-07-26
Applicant: BASF AG
Inventor: BUSCHMANN ERNST , ZIERKE THOMAS
IPC: C07C231/02 , C07C237/02 , C07K1/06 , C07K1/08 , C07K7/06 , C07K , C07C
Abstract: PCT No. PCT/EP96/03075 Sec. 371 Date Jan. 20, 1998 Sec. 102(e) Date Jan. 20, 1998 PCT Filed Jul. 12, 1996 PCT Pub. No. WO97/05096 PCT Pub. Date Feb. 13, 1997A process for preparing alpha -(N,N-dialkylamino) carboxamides of the formula I where the substituents have the stated meanings, comprises reacting the corresponding free acids with primary or secondary amines in the presence of anhydrides of an alkanephosphonic acid.
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公开(公告)号:NZ285092A
公开(公告)日:1998-01-26
申请号:NZ28509295
申请日:1995-04-26
Applicant: BASF AG
Inventor: AMBERG WILHELM , BERNARD HARALD , BUSCHMANN ERNST , HAUPT ANDREAS , JANITSCHKTE LOTHAR , JANSSEN BERND , KARL ULRICH , KLING ANDREAS , MULLER STEFAN , DE POTZOLLI BERND , RITTER KURT , THYES MARCO , ZIERKE THOMAS
IPC: A61K38/08 , A61P35/00 , C07K1/08 , A61K38/00 , C07K5/10 , C07K5/103 , C07K7/06 , C07K14/52 , C07K5/02
Abstract: PCT No. PCT/EP95/01577 Sec. 371 Date Nov. 4, 1996 Sec. 102(e) Date Nov. 4, 1996 PCT Filed Apr. 26, 1995 PCT Pub. No. WO95/30691 PCT Pub. Date Nov. 16, 1995The compound Me2Val-Val-MeVal-Pro-Pro-NHBzlxHCl is described. It is prepared from Z-Val-Val-MeVal-Pro-OR1 where Z and R1 have the meanings stated in the description. The compound shows antineoplastic activity.
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公开(公告)号:HU213384B
公开(公告)日:1997-05-28
申请号:HU9400743
申请日:1992-09-01
Applicant: BASF AG
Inventor: BUSCHMANN ERNST , REISSENWEBER GERNOT , SCHAEFER BERND
IPC: C07C253/10 , C07C253/30 , C07F9/535
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公开(公告)号:FI964446A
公开(公告)日:1997-01-03
申请号:FI964446
申请日:1996-11-05
Applicant: BASF AG
Inventor: AMBERG WILHELM , BERNARD HARALD , BUSCHMANN ERNST , HAUPT ANDREAS , JANITSCHKE LOTHAR , JANSSEN BERND , KARL ULRICH , KLING ANDREAS , MUELLER STEFAN , DE POTZOLLI BERND , RITTER KURT , THYES MARCO , ZIERKE THOMAS
Abstract: Compounds of the formulawhere R1, R2, R3 and R4 have the meaning stated in the description, and a process for preparing them are described. The compounds are suitable as starting material for synthesizing substances which are active against tumors.
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公开(公告)号:FI964448A0
公开(公告)日:1996-11-05
申请号:FI964448
申请日:1996-11-05
Applicant: BASF AG
Inventor: AMBERG WILHELM , BERNARD HARALD , BUSCHMANN ERNST , HAUPT ANDREAS , JANITSCHKE LOTHAR , JANSSEN BERND , KARL ULRICH , KLING ANDREAS , MUELLER STEFAN , DE POTZOLLI BERND , RITTER KURT , THYES MARCO , ZIERKE THOMAS
IPC: A61K38/08 , A61K38/00 , A61P35/00 , C07K1/08 , C07K5/10 , C07K5/103 , C07K7/06 , C07K14/52 , C07K
Abstract: PCT No. PCT/EP95/01577 Sec. 371 Date Nov. 4, 1996 Sec. 102(e) Date Nov. 4, 1996 PCT Filed Apr. 26, 1995 PCT Pub. No. WO95/30691 PCT Pub. Date Nov. 16, 1995The compound Me2Val-Val-MeVal-Pro-Pro-NHBzlxHCl is described. It is prepared from Z-Val-Val-MeVal-Pro-OR1 where Z and R1 have the meanings stated in the description. The compound shows antineoplastic activity.
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公开(公告)号:ZA953584B
公开(公告)日:1996-11-04
申请号:ZA953584
申请日:1995-05-04
Applicant: BASF AG
Inventor: BUSCHMANN ERNST , AMBERG WILHELM , BERNARD HARALD , HAUPT ANDREAS , JANSSEN BERND , KARL ULRICH , KLING ANDREAS , MUELLER STEFAN , JANITSCHKE LOTHAR , RITTER KURT , THYES MARCO , ZIERKE THOMAS , POTZOLLI BERND DE
IPC: A61K38/08 , A61P35/00 , A61K38/00 , C07K1/08 , C07K5/10 , C07K5/103 , C07K7/06 , C07K14/52 , C07K , A61K
Abstract: PCT No. PCT/EP95/01577 Sec. 371 Date Nov. 4, 1996 Sec. 102(e) Date Nov. 4, 1996 PCT Filed Apr. 26, 1995 PCT Pub. No. WO95/30691 PCT Pub. Date Nov. 16, 1995The compound Me2Val-Val-MeVal-Pro-Pro-NHBzlxHCl is described. It is prepared from Z-Val-Val-MeVal-Pro-OR1 where Z and R1 have the meanings stated in the description. The compound shows antineoplastic activity.
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公开(公告)号:ES2081132T3
公开(公告)日:1996-02-16
申请号:ES92920403
申请日:1992-09-24
Applicant: BASF AG
Inventor: KLEIN ULRICH , NEUMANN ULRICH , MACKENROTH WOLFGANG , RENZ GUENTER , KRIEG WOLFGANG , MACKENROTH CHRISTIANE , BUSCHMANN ERNST , DE KRAMER JACOBUS JAN , MILLI ROLAND
IPC: C07C29/10 , A01N31/04 , A01N49/00 , C07C29/60 , C07C29/62 , C07C33/02 , C07C41/48 , C07C41/54 , C07C43/178 , C07C43/313 , C07C43/315
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