公开(公告)号：CA2482414C

公开(公告)日：2010-11-16

申请号：CA2482414

申请日：2003-04-25

Applicant: BASF AG

Inventor： ENGEL STEFAN ,  KEIL MICHAEL ,  OTT CHRISTIAN ,  RACK MICHAEL

IPC: C07C253/30 ,  C07B61/00 ,  C07C255/56

Abstract: The invention relates to a method for producing 3-trifluoromethylphenyl-4-cyanobenzyl ketone by reacting a 3-trifluoromethyl benzoic acid-C1-C2-alkyl ester with 4-tolunitrile in an aprotic polar solvent or in an aprotic polar solvent mixture in the presence of at least one equimolar quantity of a base, whereby the base is selected among potassium alcoholates of primary C1-C4 alkanols.

公开(公告)号：CA2331816C

公开(公告)日：2010-11-16

申请号：CA2331816

申请日：1999-05-04

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  VON DEYN WOLFGANG ,  GEBHARDT JOACHIM ,  RACK MICHAEL ,  LOCHTMAN RENE ,  GOTZ NORBERT ,  KEIL MICHAEL ,  WITSCHEL MATTHIAS ,  HAGEN HELMUT ,  MISSLITZ ULF ,  BAUMANN ERNST

IPC: C07D261/04 ,  C07C20060101 ,  C07C201/12 ,  C07C205/44 ,  C07C249/06 ,  C07C251/40 ,  C07C251/48 ,  C07C251/52 ,  C07C253/00 ,  C07C255/50 ,  C07C317/32 ,  C07C319/14 ,  C07C323/09 ,  C07D20060101 ,  C07D261/02 ,  C07D261/08 ,  C07D413/02 ,  C07D413/10

Abstract: The invention relates to a method for producing isoxazolene of the formula (1), where the substituents have the following meanings: R1 is hydrogen, C1-C6 alkyl, R2 is C1-C6 alkyl, R3, R4, R5 are hydrogen, C1-C6 alkyl or R4 and R5 together form a linkage, R6 is a heterocyclic ring, and n is 0, 1 or 2. Said method comprises the production of an intermediate compound of the formula (VI) where R1, R3, R4 and R5 have the meanings given above. This step is followed by halogenation, thiomethylation, oxidation and acylation to yield compounds of formula (I). The invention also relates to new intermediate products for producing compounds of formula (I) and new methods for producing the intermediate products.

公开(公告)号：PL205226B1

公开(公告)日：2010-03-31

申请号：PL37105703

申请日：2003-02-06

Applicant: BASF AG

Inventor： MAYER GUIDO ,  CULLMANN OLIVER ,  WOLF BERND ,  KEIL MICHAEL

IPC: C07C249/12 ,  C07B61/00 ,  C07C251/38 ,  C07C251/48

公开(公告)号：CZ301413B6

公开(公告)日：2010-02-24

申请号：CZ20024177

申请日：2001-06-29

Applicant: BASF AG

Inventor： LOCHTMAN RENE ,  KEIL MICHAEL ,  GEBHARDT JOACHIM ,  RACK MICHAEL ,  VON DEYN WOLFGANG

IPC: C07D261/04 ,  C07C209/74 ,  C07C209/82 ,  C07C211/46 ,  C07C211/52 ,  C07D261/08

Abstract: Rešení se týká zpusobu prípravy 4-bromanilinových derivátu obecného vzorce I, ve kterém: R.sup.1.n. je C.sub.1.n.-C.sub.6.n.-alkyl, R.sup.2.n. je isoxazolový, isoxazolinový nebo isoxazolidinový kruh, s bromacním cinidlem v pyridinu nebo ve smesi rozpouštedel obsahující alespon 55 % hmotn. pyridinu.

公开(公告)号：PE20081460A1

公开(公告)日：2008-12-07

申请号：PE2007001378

申请日：2007-10-12

Applicant: BASF AG

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  ERK PETER ,  SAXELL HEIDI EMILIA ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  MAYER GUIDO ,  WOLF BERND ,  COX GERHARD ,  MICHEL ALFRED ,  ZAGAR CYRILL ,  REINHARD ROBERT ,  SIEVERNICH BERND

IPC: A01N43/48 ,  A01N43/54 ,  C07D239/54

Abstract: SE REFIERE A UNA FORMA CRISTALINA II DE 2-CLORO-5-[3,6-DIHIDRO-3-METIL-2,6-DIOXO-4-(TRIFLUOROMETIL)-1-(2H)-PIRIMIDINIL]-4-FLUORO-N-[[METIL(1-METILETIL)AMINO]SULFONIL]BENZAMIDA O FENILURACILO I, EXCENTA DE SOLVENTE, QUE PRESENTA UN DIAFRACTOGRAMA DE RAYOS X QUE MUESTRAN AL MENOS DOS DE LOS SIGUIENTES REFLEJOS EXPRESADOS EN 2 THETA: 6,3; 9,4; 10,9; 11,9; 12,6; 15,0; 15,8; 17,1 ± 0,3; ENTRE OTROS; Y UN PICO DE FUSION DENTRO DEL RANGO QUE VA DE 170 A 200 ºC. TAMBIEN SE REFIERE A UNA COMPOSICION FITOPROTECTORA PREFERENTEMENTE EN FORMA DE CONCENTRADO DE SUSPENSION ACUOSO O NO ACUOSO; Y UN PROCEDIMIENTO DE PREPARACION, SIENDO UTIL PARA CONTROLAR EL CRECIMIENTO DE VEGETACION NO DESEADA

公开(公告)号：EA010633B1

公开(公告)日：2008-10-30

申请号：EA200500510

申请日：1999-05-04

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  VON DEYN WOLFGANG ,  GEBHARDT JOACHIM ,  RACK MICHAEL ,  LOCHTMAN RENE ,  GOTZ RENE ,  KEIL MICHAEL ,  WITSCHEL MATTHIAS ,  HAGEN HELMUT ,  MISSLITZ ULF ,  BOUMANN ERNST

IPC: C07D261/04 ,  C07C20060101 ,  C07C201/12 ,  C07C205/44 ,  C07C249/06 ,  C07C251/48 ,  C07C251/52 ,  C07C253/00 ,  C07C255/50 ,  C07C317/32 ,  C07C319/14 ,  C07C323/09 ,  C07D20060101 ,  C07D251/40 ,  C07D261/02 ,  C07D261/08 ,  C07D319/14 ,  C07D413/02 ,  C07D413/10

Abstract: Изобретениеотноситсяк способуполучениясоединенийформулы XVгдеостаткиимеютследующеезначение: X - NO, S(O)Ry; Rx, Ry независимодруготдругаозначаютгалоген, карбоксил, карбоксамид, N-алкилкарбоксамид, N,N-диалкилкарбоксамид, фенил, C-Cалкил, C-Cалкокси, C-Cалкилтио; m равно 0, 1, 2, 3 или 4; n равно 0, 1 или 2. Изобретениеотноситсятакжек новомусоединениюформулы XV ик применениюспособаполучениясоединенияформулы XV.

公开(公告)号：CA2667559A1

公开(公告)日：2008-05-15

申请号：CA2667559

申请日：2007-11-05

Applicant: BASF AG

Inventor： GROENING CARSTEN ,  KEIL MICHAEL ,  KUHN OLIVER ,  LONGLET JON J ,  SUKOPP MARTIN

IPC: C07D231/44 ,  A01N43/00 ,  A01N43/56 ,  A61K31/415 ,  A61P33/00

Abstract: The present invention relates to a process for the sulfinylation of a pyr azole derivative, characterized in that 5-amino-1-[2,6-dichloro-4-(trifluoro methyl)phenyl]-1H-pyrazole-3- carbonitrile (II) is reacted with a sulfinylat ing agent selected from trifluoromethylsulfinic acid, trifluoromethylsulfini c acid anhydride, and a trifluoromethylsulfinate alkaline or alkaline earth metal salt and mixtures of the acid and/or the salt(s), in the presence of a t least one amine acid complex wherein the amine(s) are selected from tertia ry amines and the acid(s) are selected from hydrofluoric, hydrochloric, hydr obromic and hydroiodic acid and sulfonic acid derivatives, and with the addi tion of a halogenating agent.

公开(公告)号：UY30645A1

公开(公告)日：2008-05-02

申请号：UY30645

申请日：2007-10-12

Applicant: BASF AG

Inventor： ROBERT REINHARD ,  BERND WOLF ,  GUIDO MAYER ,  WERNER SEITZ ,  GERHARD HAMPRECHT ,  SAXELL HEIDI ,  PETER ERK ,  WEVER JAN ,  KEIL MICHAEL ,  LOHR SANDRA ,  GEBHARDT JOACHIM ,  SCHMIDT THOMAS ,  ZAGAR DR CYRILL ,  COX G

IPC: C07D239/54 ,  A01N43/54

Abstract: La presente invencion se refiere a una forma cristalina de 2-cloro-5-[3,6-dihidro-3-metil-2,6-dioxo-4-(trifluorometil)-1-(2H)piridiminil]-4-fluoro-N-[[metil(1-metiletil)amino]sulfonil]benzam ida. La invencion también se refiere a un proceso para la preparacion de esta forma cristalina y a formulaciones fitoprotectoras que comprenden esta forma cristalina del feniluracilo.

公开(公告)号：DE502004005772D1

公开(公告)日：2008-01-31

申请号：DE502004005772

申请日：2004-12-01

Applicant: BASF AG

Inventor： HAMPRECHT GERHARD ,  PUHL MICHAEL ,  WOLF BERND ,  KEIL MICHAEL ,  REINHARD ROBERT ,  SEITZ WERNER ,  MAYER GUIDO

IPC: C07D239/56 ,  C07D239/54

Abstract: A process is described for preparing 3-phenyl(thio)uracils or 3-phenyldithiouracils of the formula I, by reacting a phenyl iso(thio)cyanate of the formula II with an enamine of the formula III and, if appropriate, in a further step, the resulting 3-phenyl(thio)uracil or 3-phenyldithiouracil of the formula I where R1=R1a, when R1=hydrogen, is reacted with an aminating agent of the formula IV to give 3-phenyl(thio)uracils or 3-phenyldithiouracils of the formula I where R1=amino where the variables R1, R1a, R2, R3, R4, X1, X2, X3, Ar, A and L1 are each as defined in claim 1.

公开(公告)号：AT377002T

公开(公告)日：2007-11-15

申请号：AT99938237

申请日：1999-07-14

Applicant: BASF AG

Inventor： GOLSCH DIETER ,  KEIL MICHAEL ,  ISAK HEINZ ,  MAYER HORST

IPC: C07D213/80 ,  C07B43/00 ,  C07D213/78