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公开(公告)号:CZ139198A3
公开(公告)日:1998-09-16
申请号:CZ139198
申请日:1996-10-30
Applicant: BASF AG
Inventor: KLING ANDREAS , JANSSEN BERND , AMBERG WILHELM , HAUPT ANDREAS , RITTER KURT , BUSCHMANN ERNST , BERNARD HARALD , MULLER STEFAN , ZIERKE THOMAS , BARLOZZARI TERESA , DE ARRUDA MONIKA , ROBINSON SIMON
Abstract: Novel peptides of the formulaA-B-D-E-F-L,wherein A, B, D, E, F, and L have the meanings stated in the specification, and their preparation are disclosed. The novel compounds are suitable for controlling diseases.
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公开(公告)号:CA2264723A1
公开(公告)日:1998-03-12
申请号:CA2264723
申请日:1997-08-21
Applicant: BASF AG
Inventor: ZIERKE THOMAS , SCHAEFER BERND
IPC: C07D213/81 , C07B43/00 , C07C257/10 , C07D213/73 , C07D213/78 , C07D271/06 , C07D401/12 , C07D413/12 , C07K1/06 , C07K5/062
Abstract: The invention concerns a process for preparing amidines and their salts with inorganic or organic acids. According to this process, the corresponding nitrile is reacted with ammonia, a C1-C6 alkylamine or hydrazine in the presence of a mercapto carboxylic acid and optionally in the presence of an inorganic or organic ammonium salt.
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公开(公告)号:AU688037B2
公开(公告)日:1998-03-05
申请号:AU2408395
申请日:1995-04-26
Applicant: BASF AG
Inventor: AMBERG WILHELM , BERNARD HARALD , BUSCHMANN ERNST , HAUPT ANDREAS , JANITSCHKE LOTHAR , JANSSEN BERND , KARL ULRICH , KLING ANDREAS , MULLER STEFAN , POTZOLLI BERND DE , RITTER KURT , THYES MARCO , ZIERKE THOMAS
Abstract: PCT No. PCT/EP95/01577 Sec. 371 Date Nov. 4, 1996 Sec. 102(e) Date Nov. 4, 1996 PCT Filed Apr. 26, 1995 PCT Pub. No. WO95/30691 PCT Pub. Date Nov. 16, 1995The compound Me2Val-Val-MeVal-Pro-Pro-NHBzlxHCl is described. It is prepared from Z-Val-Val-MeVal-Pro-OR1 where Z and R1 have the meanings stated in the description. The compound shows antineoplastic activity.
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公开(公告)号:TR9700803T1
公开(公告)日:1998-02-21
申请号:TR9700803
申请日:1996-02-12
Applicant: BASF AG
Inventor: BOEHM HANS JOACHIM , HOEFFKEN HANS WOLFGANG , HORNBERGER WILFRIED , KOSER STEFAN , MACK HELMUT , PFEIFFER THOMAS , ZIERKE THOMAS , SEITZ WERNER
IPC: A61K31/00 , A61K38/55 , A61P7/02 , C07D205/04 , C07D207/16 , C07D213/53 , C07D213/63 , C07D213/72 , C07D213/78 , C07D213/79 , C07D239/28 , C07D241/14 , C07D241/24 , C07D401/12 , C07K5/06 , C07K5/062 , C07K5/078
CPC classification number: C07D213/78 , C07D205/04 , C07D207/16 , C07D239/28 , C07D241/24 , C07D401/12 , C07K5/06165
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公开(公告)号:ID17873A
公开(公告)日:1998-02-05
申请号:ID972839
申请日:1997-08-14
Applicant: BASF AG
Inventor: BAUCKE DORIT , LANGE UDO , MACK HELMUT , SEITZ WERNER , ZIERKE THOMAS , HOFFKEN HANS WOLFGANG , HORNBERGER WILFRIED
IPC: A61K38/00 , A61K38/05 , A61P7/02 , A61P29/00 , A61P35/00 , A61P35/04 , C07K5/06 , C07K5/062 , C07K5/065 , C07D403/00 , C07D407/00 , C07D411/00 , A61K31/33
Abstract: PCT No. PCT/EP97/04104 Sec. 371 Date Feb. 10, 1999 Sec. 102(e) Date Feb. 10, 1999 PCT Filed Jul. 29, 1997 PCT Pub. No. WO98/06741 PCT Pub. Date Feb. 19, 1998Compounds of the formula where A, B, E and D have the meanings indicated in the description, and their preparation are described. The substances are suitable for controlling diseases.
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公开(公告)号:ZA9606372B
公开(公告)日:1998-01-26
申请号:ZA9606372
申请日:1996-07-26
Applicant: BASF AG
Inventor: BUSCHMANN ERNST , ZIERKE THOMAS
IPC: C07C231/02 , C07C237/02 , C07K1/06 , C07K1/08 , C07K7/06 , C07K , C07C
CPC classification number: C07K7/06 , C07C231/02 , C07K1/082 , Y02P20/55
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公开(公告)号:MX9705970A
公开(公告)日:1997-11-29
申请号:MX9705970
申请日:1996-02-06
Applicant: BASF AG
Inventor: SEITZ WERNER , MACK HELMUT , ZIERKE THOMAS , BOHM HANS-JOACHIM , HOFFKEN HANS WOLFGANG , KOSER STEFAN , PFEIFFER THOMAS , HORNBERGER WILFRIED
Abstract: Se describen inhibidores de la tromba de la formula I: donde R1, A, B y D tienen los significados indicados en la descripcion, y productos intermedios para la preparacion de los mismos. Los compuestos I son adecuados para controlar enfermedades.
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公开(公告)号:MX9706069A
公开(公告)日:1997-10-31
申请号:MX9706069
申请日:1996-02-12
Applicant: BASF AG
Inventor: BOHM HANS-JOACHIM , HOFFKEN HANS WOLFGANG , HORNBERGER WILFRIED , KOSER STEFAN , MACK HELMUT , PFEIFFER THOMAS , SEITZ WERNER , ZIERKE THOMAS
IPC: A61K31/00 , A61K38/55 , A61P7/02 , C07D205/04 , C07D207/16 , C07D213/53 , C07D213/63 , C07D213/72 , C07D213/78 , C07D213/79 , C07D239/28 , C07D241/14 , C07D241/24 , C07D401/12 , C07K5/06 , C07K5/062 , C07K5/078 , C07K05/06 , A61K31/40 , A61K31/445
Abstract: Se describen compuestos de la Formula (I): en los cuales A, B, D, R1 y R2 tienen los significados indicados en la memoria. Los compuestos son apropiados para combatir enfermedades. Los nuevos compuestos se preparan usando un compuesto intermedio de la formula donde G y M tienen los significados indicados en la cláusula 4.
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公开(公告)号:ZA961276B
公开(公告)日:1997-08-19
申请号:ZA961276
申请日:1996-02-19
Applicant: BASF AG
Inventor: BOEHM HANS-JOACHIM , HOEFFKEN HANS WOLFGANG , HORNBERGER WILFRIED , KOSER STEFAN , MACK HELMUT , PFEIFFER THOMAS , SEITZ WERNER , ZIERKE THOMAS
IPC: A61K20060101 , C07K20060101 , C12N20060101 , C07K , A61K , C12N
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公开(公告)号:FI973282A0
公开(公告)日:1997-08-08
申请号:FI973282
申请日:1997-08-08
Applicant: BASF AG
Inventor: SEITZ WERNER , MACK HELMUT , ZIERKE THOMAS , BOEHM HANS-JOACHIM , HOEFFKEN HANS WOLFGANG , KOSER STEFAN , PFEIFFER THOMAS , HORNBERGER WILFRIED
Abstract: PCT No. PCT/EP96/00472 Sec. 371 Date Jul. 30, 1997 Sec. 102(e) Date Jul. 30, 1997 PCT Filed Feb. 6, 1996 PCT Pub. No. WO96/24609 PCT Pub. Date Aug. 15, 1996Thrombin inhibitors of the formula where R1, A, B and D have the meaning indicated in the description, and intermediates for the preparation thereof are described. The compounds I are suitable for controlling diseases.
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