公开(公告)号：DE19547882A1

公开(公告)日：1997-06-26

申请号：DE19547882

申请日：1995-12-21

Applicant: BASF AG

Inventor： KLINTZ RALF DR ,  KIRSTGEN REINHARD DR ,  KOENIG HARTMANN DR ,  RACK MICHAEL DR ,  HAMPRECHT GERHARD DR ,  SCHAEFER PETER DR ,  HEISTRACHER ELISABETH DR ,  ZAGAR CYRILL DR ,  HARRIES VOLKER DR ,  KRAMER JACOBUS JAN DE DR

IPC: A01N43/82 ,  A01N43/836 ,  C07D285/08

Abstract: Thiadiazols have the formula (I), in which the index and the substituents have the following meaning: n equals 1, 2, 3, 4 or 5, whereas the R substituents may differ from each other when n is higher than 1; R stands for alkyl, alkenyl or alkinyl, nitro, cyano, halogen, C1-C4-alkyl halide, C1-C4-alkoxy, C1-C4-alkoxy halide, C1-C4-alkylthio, C1-C4-alkyl sulfonyl, C1-C4-alkylcarbonyl, C1-C4-alkoxycarbonyl and when n > 1 a 1,3-butadien-1,4-yl or oxy-(C1-C2-alkylidene)-oxy group bonded to two adjacent C atoms of the phenyl radical, whereas said group may be partially or completely halogenated. Also disclosed is a process for preparing these compounds, mixtures containing the same and their use for controlling nematodes.

公开(公告)号：AP2344A

公开(公告)日：2011-12-28

申请号：AP2008004353

申请日：2006-06-30

Applicant: BASF AG

Inventor： CULBERTSON DEBORAH L ,  ANSPAUGH DOUGLAS D DR ,  RACK MICHAEL DR

IPC: A01N43/56 ,  C07D401/04

Abstract: wherein the variables and the indices are as defined per the description, processes for preparing the compounds I, pesticidal compositions comprising compounds I, use of compounds I for the control of insects, acarids or nematodes, and methods for treating, controlling, preventing or protecting animals against infestation or infection by parasites by use of compounds of formula I.

公开(公告)号：DE19738084A1

公开(公告)日：1999-03-04

申请号：DE19738084

申请日：1997-09-01

Applicant: BASF AG

Inventor： MENKE OLAF DR ,  GOETZ ROLAND DR ,  RACK MICHAEL DR ,  HAMPRECHT GERHARD DR ,  MENGES MARKUS DR ,  REINHARD ROBERT DR ,  SCHAEFER PETER DR ,  ZAGAR CYRILL DR ,  WESTPHALEN KARL-OTTO DR ,  WALTER HELMUT DR ,  MISLITZ ULF DR

IPC: A01N43/80 ,  C07D405/06 ,  C07D413/06 ,  C07D417/06 ,  C07F9/6584 ,  C07D239/54 ,  A01N43/54 ,  A01N43/84 ,  A01N57/02 ,  C07D403/06 ,  C07F9/6564 ,  C07F9/6571

Abstract: 3-Arylmethyluracil derivatives (I.1)-(I.4) are new, where A = H, 1-4C alkyl, NH2, 1-4C alkylamino or di-(1-4C alkyl)amino; X = O or S; n = not defined; R1 = 1-4C haloalkyl; R2 = H, halo or 1-3C alkyl; R3-R5 = H, CN, thiocyanato, halo, 1-4C haloalkyl, 1-4C haloalkoxy, 1-4C haloalkylthio, 1-4C alkyl or 1-4C alkoxy; R6, R7 = 1-4C alkyl, NH2, 1-4C alkylamino or di(1-4C alkyl)amino, or R6 and R7 together form =O; R8 may be in position alpha or beta and R3 is in the other position; R8 = (1) H, halo, amino, 1-4C alkylsulphonylamino or di(1-4C alkyl)amino; (2) 1-6C alkoxy, 1-6C alkylthio, 3-6C cycloalkoxy, 3-6C cycloalkylthio, 2-6C alkenyloxy, 5-7C cycloalkenyloxy, 2-6C alkenylthio, 2-6C alkynyloxy, 2-6C alkynylthio, (1-6C alkyl)carbonyloxy, (1-6C alkyl)carbonylthio, (1-6C alkoxy)carbonyloxy, (2-6C alkenyl)carbonyloxy, (2-6C alkenyl)carbonylthio, (2-6C alkynyl)carbonyloxy, (2-6C alkynyl)carbonylthio, 1-6C alkylsulphonyloxy or 1-6C alkylsulphonyl, where the last 18 groups may contain 1-4 substituents; (3) CT-R11, C(R11)(Y1R12)(Y2R13), C(R11)=C(R14)CN, C(R11)=C(R14)CO-R15, CH(R11)-CH(R14)CO-R15, C(R11)=C(R14)-CH2-CO-R15, C(R11)=C(R14)-C(R16)=C(R17)-CO-R15, C(R11)=C(R14)-CH2-CH(R18)CO-R15, CO-OR19, CO-SR19, CO-N(R19)-OR20, C?=C-CO-NH-OR20, C?=C-CO-N(R19)-OR20, , C?=C-CS-NH-OR20, C?=C-CS-N(R19)-OR20, C(R11)=C(R14)-CO-NH-OR20, C(R11)=C(R14)-CO-N(R19)-OR20, C(R11)=C(R14)-CS-NH-OR20, C(R11)=C(R14)-CS-N(R19)-OR20, C(R11)=C(R14)-C(R21)=N-OR20, C(R21)=N-OR20, C?=C-C(R21)=N-OR20, C(Y1R12)(Y2R13)-OR19, C(Y1R12)(Y2R13)-SR19, C(Y1R12)(Y2R13)-N(R23)(R24), N(R23)(R24), CO-N(R23)(R24), or groups of formula (i), (ii), -C?=C-(i), -C?=C-(ii), -C(R11)=C(R14)-(i) or -C(R11)=C(R14 )-(ii); Y1, Y2 = S or O; theta = 1-3C alkylene optionally substituted by 1-6C alkyl; R11 = H, CN, 1-6C alkyl, 1-6C haloalkyl, 2-6C alkenyl, 2-6C alkynyl, 3-6C cycloalkyl, 1-6C alkoxy-(1-6C alkyl) or (1-6C alkoxy)carbonyl; R12, R13 = 1-6C alkyl, 1-6C haloalkyl, 3-6C alkenyl, 3-6C alkynyl or 1-6C alkoxy-(1-6C alkyl) or R12 and R13 together form a 2-4 membered carbon chain which is optionally substituted and can contain non-adjacent O, S or N atoms instead of C atoms or be condensed or form a spiro attachment with a 3-7 membered ring; R14 = H, CN, halo, 1-6C alkyl, 1-6C haloalkyl, 1-6C alkoxy, (1-6C alkyl)carbonyl or (1-6C alkoxy)carbonyl; R15 = H, OR22, SR22, 1-6C alkyl (optionally substituted by one or two 1-6C alkoxy groups), 2-6C alkenyl, 2-6C alkynyl, 1-6C haloalkyl, 3-6C cycloalkyl, 1-6C alkylthio-(1-6C alkyl), 1-6C alkyliminooxy, N(R23)(R24) or optionally substituted phenyl; R22 has the same meanings as R19; R16 = H, CN, halo, 1-6C alkyl, 3-6C alkenyl, 3-6C alkynyl, 1-6C alkoxy-(1-6C alkyl), (1-6C alkyl)carbonyl, (1-6C alkoxy)carbonyl, N(R25)(R26) or optionally substituted phenyl; R25, R26 have the same meanings as R23 and R24; R17 = H, halo, CN, 1-6C alkyl, 1-6C alkoxy, 1-6C haloalkyl, (1-6C alkyl)carbonyl or (1-6C alkoxy)carbonyl; R18 = H, CN, 1-6C alkyl or (1-6C alkoxy)carbonyl; R19 = H, 1-6C alkyl, 1-6C haloalkyl, 2-6C alkenyl or 2-6C alkynyl (where the latter four groups are optionally substituted), (1-6C alkyl)carbonyl, (1-6C haloalkyl)carbonyl, (1-6C alkoxy)carbonyl, 1-6C alkylaminocarbonyl, di-(1-6C alkyl)aminocarbonyl, 1-6C alkoxyimino-(1-6C alkyl), 3-6C cycloalkyl, phenyl or phenyl-(1-6C alkyl), where the phenyl ring is optionally substituted; R20 = H, 1-6C alkyl, 1-6C haloalkyl, 3-6C cycloalkyl, 3-6C alkenyl, 3-6C alkynyl, hydroxy-(1-6C alkyl), 1-6C alkoxy-(1-6C alkyl), 1-6C alkylthio-(1-6C alkyl), cyano-(1-6C alkyl), (1-6C alkyl)carbonyl-(1-6C alkyl), (1-6C alkoxy)carbonyl-(1-6C alkyl), (1-6C alkoxy)carbonyl-(2-6C alkenyl), (1-6C alkyl)carbonyloxy-(1-6C alkyl) or phenyl-(1-6C alkyl), where the phenyl ring may contain 1-3 substituents; R

公开(公告)号：DE19636995A1

公开(公告)日：1998-03-19

申请号：DE19636995

申请日：1996-09-12

Applicant: BASF AG

Inventor： HAMPRECHT GERHARD DR ,  GEBHARDT JOACHIM DR ,  ISAK HEINZ DR ,  RACK MICHAEL DR ,  RHEINHEIMER JOACHIM DR ,  SCHAEFER PETER DR

IPC: B01J31/24 ,  C07D213/24 ,  C07D213/61 ,  C07D213/62 ,  A01N43/40

Abstract: Process for the production of substituted phenylpyridines having formula (I), characterized by the fact that substituted pyridine having formula (II) is made to react with an aryl compound having formula (III).

公开(公告)号：DE19633751A1

公开(公告)日：1998-02-26

申请号：DE19633751

申请日：1996-08-22

Applicant: BASF AG

Inventor： SCHAEFER PETER DR ,  HAMPRECHT GERHARD DR ,  MENGES MARKUS DR ,  MENKE OLAF DR ,  RACK MICHAEL DR ,  ZAGAR CYRILL DR ,  WALTER HELMUT DR ,  WESTPHALEN KARL-OTTO DR ,  MISLITZ ULF DR

IPC: A01N43/76 ,  A01N43/84 ,  C07D213/61 ,  C07D213/70 ,  C07D413/04 ,  C07D417/04 ,  A01N43/48 ,  A01N43/72 ,  C07D213/89 ,  C07D401/04

Abstract: Substituted 2-arylpyridine of formula (I) and salts thereof. In said formula (I), R = SH, SO2OH, SO2C1, SO2NH2, C1-C6-Alkylthio, C1-C6-Alkyl sulfinyl, C1-C6-alkylsulfonyl, C1-C6-alkylamino-sulfonyl, Di(C1-C6-alkyl)aminosulfonyl; R , R = H, halogen; R = H, C1-C6-alkyl, C1-C6-halogenalkyl, cyano-C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, C1-C4-halogen-alkoxy-C1-C4-alkyl, C1-C6-alkylthio-C1-C6-alkyl, C1-C6 alkyl sulfinyl-C1-C6-alkyl, C1-C6-alkylsulfonyl-C1-C6-alkyl, C1-C4-alkoxy-C1-C4-alkoxy-C1-C4-alkyl, C1-C6-alkoxycarbonyl-C1-C6-alkyl, C1-C3-alkoxy-C1-C3-alkoxycarbonyl-C1-C6-alkyl, C2-C4-alkenyloxy-C1-C4-alkyl, C3-C4-alkinyloxy-C1-C4-alkyl, C3-C7-cycloalkyl, C3-C7-cycloalkyl-C1-C6-alkyl, C3-C7-cycloalkyloxy-C1-C6-alkyl, C3-C7-cycloalkylthio-C1-C6-alkyl, C3-C8-alkenyl, C3-C8-alkinyl, C3-C8-halogenalkenyl, C3-C8-halogenalkinyl, C1-C6-alkoxy-C3-C8-alkenyl, C1-C6-alkoxy-C3-C8-alkinyl, C1-C6-alkylcarbonyl, C1-C6-alkylsulfonyl, C3-C6-alkenyloxy, C3-C6-alkinyloxy or eventually substituted benzyl; X = -O-, -S-, -NH-, -N(CH3)-, -CH2-; Y = chemical bond, -CO-, C(R ,R ); R ,R = H, NO2, CN, OCH3, SCH3, halogen, C1-C4-alkyl, C1-C4-halogenalkyl, C1-C4-alkoxycarbonyl, C2-C6-alkenyl, C3-C6-alkinyl, C1-C4-alkoxycarbonyl-C1-C4-alkyl. Application as herbicide; for plant desiccation/defoliation.

公开(公告)号：DE19605903A1

公开(公告)日：1997-08-21

申请号：DE19605903

申请日：1996-02-17

Applicant: BASF AG

Inventor： OBERDORF KLAUS DR ,  GRAMMENOS WASSILIOS DR ,  SAUTER HUBERT DR ,  GROTE THOMAS DR ,  MUELLER BERND DR ,  KIRSTGEN REINHARD DR ,  MUELLER RUTH DR ,  BAYER HERBERT DR ,  PTOCK ARNE DR ,  RACK MICHAEL DR ,  HARREUS ALBRECHT DR ,  ROEHL FRANZ DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR ,  STRATHMANN SIEGFRIED DR ,  HARRIES VOLKER DR

IPC: A01N43/40 ,  C07D213/64 ,  C07D213/643 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12 ,  C07D213/61 ,  A01N43/54 ,  A01N43/66

Abstract: The invention concerns pyridyl-phenyl- and benzylethers of formula (I), and their salts and N-oxides, in which the substituents and indices have the following meanings: Q is C(CO2CH3)=CHCH3, C(CO2CH3)=CHOCH3, C(CONH2)=NOCH3, C(CO2CH3)=NOCH3, C(CONHCH3)=NOCH3 or N(OCH3)-CO2CH3; n is 0 or 1; R is hydrogen or an organic group bonded via a carbon atom; R is hydrogen, cyano, halogen or an organic group bonded via a carbon, oxygen, sulphur or nitrogen atom; R is hydrogen, halogen, C1-C4 alkyl or C1-C2 alkyl halide; x is 0, 1 or 2; R is cyano, nitro, halogen or an organic group bonded via a carbon, oxygen, sulphur or nitrogen atom; y is 0, 1, 2 or 3; and R is cyano, halogen, C1-C4 alkyl, C1-C4 alkyl halide or C1-C4 alkoxy. The invention further concerns a process and intermediate products for preparing these substances and their use.

公开(公告)号：DE19548781A1

公开(公告)日：1997-07-03

申请号：DE19548781

申请日：1995-12-27

Applicant: BASF AG

Inventor： WAGNER OLIVER DR ,  WETTERICH FRANK DR ,  EICKEN KARL DR ,  RACK MICHAEL DR ,  HAMPRECHT GERHARD DR ,  LAMM GUNTHER DR ,  SPEAKMAN JOHN-BRYAN DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR ,  STRATHMANN SIEGFRIED DR

IPC: A01N43/40 ,  A01N43/42 ,  A01N43/54 ,  A01N43/78 ,  A01N43/90 ,  C07D213/70 ,  C07D213/71 ,  C07D213/82 ,  C07D213/85 ,  C07D215/54 ,  C07D239/38 ,  C07D277/74 ,  C07D277/76 ,  C07D513/04 ,  A01N43/48 ,  C07D241/18 ,  C07D241/44 ,  C07D251/14

Abstract: Fungicide contains a substd, alkyl(thio-, sulphinyl- or sulphonyl-)-heterocyclic cpd. of formula A-S(O)m-A'-X-CO-Q (I) or its salt or N-oxide. A = a gp. of formula (a)-(d); U = CR2 or N; V = CR4 or N; R1-R4 = H, CN, NO2, halo, CONH2, SO2Me, 1-4C alkyl (opt. substd. by halo or 1-4C alkoxy), 1-4C alkoxy, 1-4C haloalkoxy, 1-4C alkylthio, 1-4C alkoxy-carbonyl, Ar, OAr or Het; Ar = aryl (opt. mono-, di- or trisubstd. by CN, NO2, halo, 1-4C alkyl (opt. substd. by halo or 1-4C alkoxy), 1-4C alkoxy, 1-4C haloalkoxy, 1-4C alkylthio, 1-4C alkoxy-carbonyl or 1-4C acyl); Het = heteroaryl (opt. substd. as for Ar); m, = 0-2; A' = 1,2-ethylidene or 1,3-propylidene opt. substd. by A1 or A2; A1 = 1-8C alkyl, 1-8C haloalkyl, 2-8C alkenyl, 2-8C haloalkenyl or 2-8C alkynyl (all opt. mono-, di- or trisubstd. by CN, 1-4C alkoxy, 1-4C haloalkyl, 1-4C alkylthio, 1-4C alkoxy-carbonyl, 3-7C cycloalkyl or 5-7C cycloalkenyl); A2 = 3-7C cycloalkyl or 5-7C cycloalkenyl (both opt. substd. by 1 or more halo or 1-3 CN, halo, 1-4C alkyl, 1-4C haloalkyl and 1-4C alkoxy); X = O, S or NR5; R5 = H, 1-8C alkyl or 3-7C cycloalkyl; Q = aryl or heteroaryl (opt. opt. mono-, di- or trisubstd. by CN, NO2, halo, 1-4C alkyl (opt. substd. by halo or 1-4C alkoxy), 1-4C alkoxy, 1-4C haloalkoxy, 1-4C alkylthio, 1-4C alkoxy-carbonyl, 1-4C acyl, 1-4C alkylsulphinyl, 1-4C alkylsulphonyl, Ar, OAr or Het), 3-7C cycloalkyl or 5-7C cycloalkenyl (both opt. substd. by 1 or more halo or 1-3 CN, halo, 1-4C alkyl, 1-4C haloalkyl, 1-4C alkoxy(1-4C) alkyl, 1-4C haloalkoxy, 1-4C alkoxy, 1-4C alkylthio, 1-4C alkoxy-carbonyl, 3-7C cycloalkyl, 5-7C cycloalkenyl, Ar, OAr or Het), or aryl-(1-4C)alkyl ((opt. opt. mono-, di- or trisubstd. by CN, NO2, halo, 1-4C alkyl (opt. substd. by halo or 1-4C alkoxy), 1-4C alkoxy, 1-4C haloalkoxy, 1-4C alkylthio, 1-4C alkoxy-carbonyl, 1-4C acyl, Ar, OAr or Het). Compounds (I) are new, with provisos.

公开(公告)号：DE19546699A1

公开(公告)日：1997-06-19

申请号：DE19546699

申请日：1995-12-14

Applicant: BASF AG

Inventor： OBERDORF KLAUS DR ,  GRAMMENOS WASSILIOS DR ,  SAUTER HUBERT DR ,  GROTE THOMAS DR ,  KIRSTGEN REINHARD DR ,  MUELLER RUTH DR ,  MUELLER BERND DR ,  ROEHL FRANZ DR ,  RACK MICHAEL DR ,  BAYER HERBERT DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR ,  STRATHMANN SIEGFRIED DR ,  HARRIES VOLKER DR

IPC: A01N43/54 ,  C07D239/34 ,  A01N37/52

Abstract: 2-(pyrimidin-4-yloxy)methyl)phenylacetic acid derivatives of formula (I) and their salts and N-oxides are new. R1 = H or 1-4C alkyl; R2 = halo, CH3, CH2CH3, halomethyl or haloethyl; R3 = phenyl, phenoxy, phenoxymethyl, benzyloxy or heteroaryl, (all optionally ring-substituted), H, amino, OH, SH, halo, 1-8C alkyl (optionally substituted by Ar or halo), alkoxy-(1-4C alkyl), alkoxy, mono- or di- alkylamino, alkylthio, alkylsulphoxy, alkylsulphonyl, 3-8C cycloalkyl, trialkylsilyloxy; Ar = phenyl (optionally mono- or di-substituted by halo, CN, NO2, 1-4C alkyl, 1-4C haloalkyl or 1-4C alkoxy); R4 = H, CN, halo, 1-4C alkyl, 1-4C haloalkyl or 1-4C alkoxy; Q = C(=NOCH3)CONHCH3, C(=NOCH3)COOCH3 or N(OCH3)COOCH3; alkyl, alkoxy have 1-8 C unless specified otherwise.

公开(公告)号：DE19545878A1

公开(公告)日：1997-06-12

申请号：DE19545878

申请日：1995-12-08

Applicant: BASF AG

Inventor： MUELLER BERND DR ,  SAUTER HUBERT DR ,  BAYER HERBERT DR ,  GRAMMENOS WASSILIOS DR ,  GROTE THOMAS DR ,  KIRSTGEN REINHARD DR ,  OBERDORF KLAUS DR ,  ROEHL FRANZ DR ,  GOETZ NORBERT DR ,  RACK MICHAEL DR ,  MUELLER RUTH DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR ,  STRATHMANN SIEGFRIED DR ,  HARRIES VOLKER DR ,  PTOCK ARNE DR

IPC: C07D213/75 ,  A01N47/18 ,  C07D213/74 ,  C07D213/76 ,  C07D213/79 ,  C07D213/81 ,  C07D401/12 ,  C07D401/14 ,  C07D405/12 ,  C07D405/14 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D413/14 ,  C07D417/12 ,  C07D417/14 ,  C07D215/38 ,  C07D471/04 ,  C07D491/04 ,  C07D495/04 ,  A01N43/40

Abstract: The invention relates to pyridyl carbamates of formula (I), in which the index and the substituents have the follwing meaning: R' is hydrogen, optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, alkyl carbonyl and alkoxy carbonyl; R" is optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, or where V is an amino group, also hydrogen; V is oxygen (-O-), sulphur (-S-) or an amino group which can carry one of the following radicals: alkyl, alkenyl, alkinyl or cycloalkyl; X is cyano, nitro, halogen, optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy, or where n > 1, an optionally substituted bridge bound to two adjacent C-atoms of the pyridyl ring and containing 3 to 4 members from the group of 3 or 4 carbon atoms, 2 to 3 carbon atoms and one or two nitrogen, oxygen and/or sulphur atoms, said bridge being able to form a partially unsaturated or aromatic radical together with the ring to which it is bound; n is 0, 1, 2 or 3, and the radicals X may be different when n > 1; R is halogen, hydroxy, mercapto, amino, formyl, carboxyl, carbonylamino or an organic radical which is bound directly or via an oxy group, mercapto group, amino group, carboxyl or carbonylamino group, or along with one group X and the pyridyl ring to which they are bound, an optionally substituted bicyclic, partially or completely unsaturated system which can contain heteroatoms from the group of oxygen, sulphur and nitrogen in addition to carbon ring members. It also relates to a process and intermediates for the preparation of said pyridil carbamates and use thereof.

公开(公告)号：DE19540989A1

公开(公告)日：1997-05-07

申请号：DE19540989

申请日：1995-11-03

Applicant: BASF AG

Inventor： MUELLER BERND DR ,  SAUTER HUBERT DR ,  BAYER HERBERT DR ,  GRAMMENOS WASSILIOS DR ,  GROTE THOMAS DR ,  KIRSTGEN REINHARD DR ,  OBERDORF KLAUS DR ,  ROEHL FRANZ DR ,  GOETZ NORBERT DR ,  RACK MICHAEL DR ,  MUELLER RUTH DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR ,  STRATHMANN SIEGFRIED DR ,  HARRIES VOLKER DR

IPC: C07D213/30 ,  A01N43/40 ,  C07D213/53 ,  C07D213/54 ,  C07D213/55

Abstract: The invention concerns pyridylacetic acid derivatives of formula (I), in which the substituents and the index have the following meanings: X - NOCH3, CHOCH3, CHCH3 and CHCH2CH3; Y - oxygen or NR', R' representing hydrogen or alkyl; R - cyano, nitro, trifluoromethyl, halogen, alkyl and alkoxy; m is 0, 1 or 2; R is hydrogen and alkyl; R - hydrogen, cyano, nitro, hydroxy, amino, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkyl thio, alkylamino or dialkylamino; R - hydrogen, cyano, nitro, hydroxy, amino, halogen; or optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkinyl, alkinyloxy, alkinylthio, alkinylamino, N-alkinyl-N-alkylamino, cycloalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocyclyl-N-alkylamino,aryl, aryloxy, arylthio,arylamino, N-aryl-N-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetarylamino, and N-hetaryl-N-alkylamino; R - hydrogen, optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, alkylsulphonyl, cycloalkyl, aryl, arylcarbonyl, arylsulphonyl, hetaryl, hetarylcarbonyl, or hetarylsulphonyl. Also disclosed are the salts of the above derivatives,and methods and intermediate products for producing them and agents containing them.