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    Method for manufacturing aryl carboxamides
    76.
    发明专利
    Method for manufacturing aryl carboxamides 未知

    公开(公告)号：AU2009245791A1

    公开(公告)日：2009-11-12

    申请号：AU2009245791

    申请日：2009-05-06

    Applicant: BASF SE

    Inventor： KORADIN CHRISTOPHER ,  REICHERT WOLFGANG ,  KEIL MICHAEL ,  ZIERKE THOMAS ,  WOLF BERND ,  SMIDT SEBASTIAN PEER ,  MAYWALD VOLKER ,  RACK MICHAEL

    IPC: C07D213/82 ,  C07C231/02 ,  C07C233/57 ,  C07C233/64 ,  C07D231/14 ,  C07D231/16

    Abstract: A process for preparing arylcarboxamides of the formula (I) where Ar=a mono- to trisubstituted phenyl, pyridyl or pyrazolyl ring, where the substituents are selected from halogen, C1-C4-alkyl and C1-C4-haloalkyl; M=thienyl or phenyl, which may bear a halogen substituent; Q=direct bond, cyclopropylene, fused bicyclo[2.2.1]heptane or bicyclo[2.2.1]heptene ring; R1=hydrogen, halogen, C1-C6-alkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, mono- to trisubstituted phenyl, where the substituents are selected from halogen and trifluoromethylthio, or cyclopropyl; by reacting an acid chloride of the formula (II) with an arylamine (III) in a suitable nonaqueous solvent, wherein, in the absence of an auxiliary base, a) the acid chloride (II) is initially charged, b) a pressure of from 0 to 700 mbar is established, c) the arylamine (III) is metered in an approximately stoichiometric amount and d) the product of value is isolated.

    Method for preparing 1,3,4-substituted pyrazol compounds
    77.
    发明专利
    Method for preparing 1,3,4-substituted pyrazol compounds 未知

    公开(公告)号：AU2009243550A1

    公开(公告)日：2009-11-12

    申请号：AU2009243550

    申请日：2009-05-04

    Applicant: BASF SE

    Inventor： MAYWALD VOLKER ,  WOLF BERND ,  SUKOPP MARTIN ,  KORADIN CHRISTOPHER ,  ZIERKE THOMAS ,  RACK MICHAEL ,  KEIL MICHAEL

    IPC: C07D231/14

    Abstract: The present invention relates to a process for preparing 1,3-substituted pyrazole compounds of the formula I in which X is especially a CX1X2X3 group in which X1, X2 and X3 are each independently especially hydrogen, fluorine or chlorine, R1 is C1-C4-alkyl or cyclopropyl, and R2 is hydrogen, CN or a CO2R2a group in which R2a is especially C1-C6-alkyl, comprising the following steps: i) reacting a compound of the formula II with a hydrazone of the formula III where the variables X and R2 in formula II are each as defined for formula I, Y is oxygen, an NRy1 group or an [NRy2Ry3]+Z- group, R3 is OR3a or an NR3bR3c group, and where the variable R1 in formula III is as defined for formula I, R4 and R5 are each independently hydrogen, C1-C6-alkyl, optionally substituted phenyl, where at least one of the R4 and R5 radicals is different from hydrogen, and where R4 and R5 together with the carbon atom to which they are bonded may also be a 5- to 10-membered saturated carbocycle; ii) treating the reaction product obtained with an acid in the presence of water.

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