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公开(公告)号:CA2211534A1
公开(公告)日:1996-08-29
申请号:CA2211534
申请日:1996-02-13
Applicant: BASF AG
Inventor: HILL REGINA LUISE , VOSSEN MARCUS , RANG HARALD , HARREUS ALBRECHT , KARDORFF UWE , PLATH PETER , WALTER HELMUT , MISSLITZ ULF , OTTEN MARTINA , ENGEL STEFAN , R HL FRANZ , WESTPHALEN KARL-OTTO , VON DEYN WOLFGANG
IPC: A01N43/80 , C07D261/08 , C07D413/10 , C07D417/10 , A01N43/72 , C07D261/18
Abstract: The invention concerns isoxazol-4-yl-benzoyl derivatives of formula (I) in which the substituents have the following meanings: L and M represent hydrogen, C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkinyl, C1-C4 alkoxy (these groups being optionally substituted by one to five halogen atoms or C1-C4 alkoxy), halogen, cyano, nitro, a -(Y)n-S(O)mR7 or (Y)n-CO-R8 group; Z represents a five to six-membered heterocyclic saturated or unsaturated group which contains one to three heteroatoms selected from the group comprising oxygen, sulphur or nitrogen and can optionally be substituted by halogen, cyano, nitro, an -CO-R8 group, C1-C4 alkyl, C1-C4 alkyl halide, C3-C8 cycloalkyl, C1-C4 alkoxy, C1-C4 alkoxy halide, C1-C4 alkyl thio, C1-C4 alkyl thio halide, di-C1-C4 alkyl amino, phenyl optionally substituted by halogen, cyano, nitro, C1-C4 alkyl or C1-C4 alkyl halide, or an oxo group which can be present in the tautomeric form as a hydroxy group, is substituted or, together with a condensation-bound phenyl ring which is optionally substituted by halogen, cyano, nitro, C1-C4 alkyl or C1-C4 alkyl halide, with a condensation-bound carbocycle or with a condensation-bound second heterocycle which can optionally be substituted by halogen, cyano, nitro, C1-C4 alkyl, diC1-C4 alkyl amino, C1-C4 alkoxy, C1-C4 alkoxy halide, or a C1-C4 alkyl halide, form a bicyclic system; Y represents O or NR9; n is 0 or 1; m is 0, 1 or 2; R7 represents C1-C4 alkyl, C1-C4 alkyl halide or NR9R10; R8 represents C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy or NR9R10; R9 represents hydrogen or C1-C4 alkyl; R10 represents C1-C4 alkyl; Q represents an isoxazole ring connected at position 4 and of formula (II) in which R1 represents hydrogen or -C02R3, R2 represents hydrogen, C1-C4 alkyl or C3-C6 cycloalkyl which can optionally be substituted by one or more halogen atoms or C1-C4 alkyl, R3 representing a C1-C4 alkyl; J represents a carbonyl group CO or a -CHR4 group, R4 representing an OH group, a hydroxyl group optionally acylated with C2-C4 acyl, or a chlorine atom. The invention also concerns salts of compounds of formula (I) usually utilized in agriculture.
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公开(公告)号:CA2233258A1
公开(公告)日:1997-05-09
申请号:CA2233258
申请日:1996-10-24
Applicant: BASF AG
Inventor: AMMERMANN EBERHARD , SAUTER HUBERT , HARRIES VOLKER , GRAMMENOS WASSILIOS , MUELLER RUTH , BAYER HERBERT , OBERDORF KLAUS , R HL FRANZ , HARREUS ALBRECHT , LORENZ GISELA , MUELLER BERND , KIRSTGEN REINHARD , GROTE THOMAS , G TZ NORBERT , STRATHMANN SIEGFRIED
IPC: C07D521/00 , A01N35/10 , A01N37/36 , A01N37/50 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/76 , A01N43/78 , A01N43/80 , A01N47/20 , C07C49/76 , C07C251/40 , C07C251/48 , C07C251/60 , C07C255/17 , C07C271/28 , A01N43/00 , C07D275/02 , C07D249/08 , C07D261/08 , C07D271/10 , C07C323/12 , C07D231/12 , C07C317/16 , C07D333/24 , C07D333/28 , C07D239/30 , C07D277/30 , C07D263/32 , C07C233/33 , C07D207/337 , C07C327/38 , C07D307/54 , C07D213/56 , C07D307/56 , C07D317/60 , C07D213/61 , C07C255/62 , C07C255/64
Abstract: The invention concerns phenylacetic acid derivatives of formula (I), in which the variables have the following meanings: X = NOCH3, CHOCH3 or CHCH3; Y = O or NZ, Z standing for hydrogen or alkyl; R1 = H or alkyl; R2 = cyano, nitro, trifluoromethyl, halogen, alkyl or alkoxy; m = 0, 1 or 2, wherein the group R2 can be different when m = 2; R3 = H, cyano, alkyl, alkyl halide, alkoxy or cyclopropyl; R4 = alkylenedioxy, the alkylene groups being partially or completely halogenated, or one of the groups: -(C=O)-Ra, -C(=NORa)-Ap-Rb, -NRc- (C=O)-Ap-Ra, -O-(C=O)-NRaRb or -N(Rc)-ORd, Ra, Rb, independently of each other, being H or optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, heterocyclyl, aryl or heteroaryl; Rc, Rd, independently of each other, being H or optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, cycloalkyl, cycloalkylcarbonyl, cycloalkyloxycarbonyl, arylcarbonyl or heteroarylcarbonyl; p = 0 or 1; A = O, S or N, the N-atom carrying H or alkyl; n = 1 or 2, wherein the group R4 can be different when n = 2; and R5 = H, alkylsulphonyl or optionally substituted alkyl, alkenyl, alkinyl or cycloalkyl. The invention further concerns salts of these substances, a process and intermediate products for their preparation, and their use as fungicides and pesticides.
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公开(公告)号:CA2218897A1
公开(公告)日:1996-11-28
申请号:CA2218897
申请日:1996-05-13
Applicant: BASF AG
Inventor: AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , MUELLER BERND , K NIG HARTMANN , HARRIES VOLKER , OBERDORF KLAUS , SAUTER HUBERT , R HL FRANZ , KIRSTGEN REINHARD , RACK MICHAEL , LORENZ GISELA
IPC: A01N43/56 , A01N43/653 , C07D231/18 , C07D231/20 , C07D231/22 , C07D249/12 , C07D401/04 , C07D401/12 , C07D403/04 , C07D403/12 , C07D403/02 , C07D405/04 , C07D409/04 , C07D413/04 , C07D417/04 , C07D231/14 , A01N43/48 , A01N43/64 , A01N43/713 , A01N43/72
Abstract: Compounds of the general formula (I) in which n is 0, 1, 2, 3 or 4; R is nitro, cyano, halogen, possibly substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy or, if n is greater than 1, additionally a possibly substituted bridge bonded to two adjacent ring atoms; R1, R2 is alkyl; R3 is a substituted pyrazole or triazole radical of the formulae (A.1) to (A.3), in which the bond marked . is the bond to oxygen, process for their production and their use.
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公开(公告)号:CA2217773A1
公开(公告)日:1996-11-14
申请号:CA2217773
申请日:1996-04-26
Applicant: BASF AG
Inventor: K NIG HARTMANN , KIRSTGEN REINHARD , MUELLER BERND , AMMERMANN EBERHARD , GROTE THOMAS , HARREUS ALBRECHT , STRATHMANN SIEGFRIED , SAUTER HUBERT , LORENZ GISELA , R HL FRANZ
IPC: C07D253/06 , A01N37/10 , A01N37/36 , A01N37/44 , A01N39/02 , A01N43/08 , A01N43/10 , A01N43/20 , A01N43/40 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/707 , A01N43/76 , A01N43/80 , A01N43/84 , C07C69/618 , C07C69/734 , C07C69/736 , C07C69/738 , C07C227/18 , C07C229/36 , C07C235/28 , C07C251/48 , C07C251/52 , C07D213/55 , C07D213/64 , C07D215/14 , C07D215/22 , C07D215/38 , C07D215/46 , C07D215/48 , C07D215/50 , C07D239/26 , C07D239/30 , C07D239/34 , C07D241/42 , C07D261/08 , C07D261/10 , C07D261/20 , C07D263/32 , C07D263/56 , C07D271/06 , C07D271/10 , C07D275/02 , C07D277/20 , C07D277/22 , C07D277/24 , C07D277/28 , C07D277/30 , C07D285/08 , C07D307/42 , C07D333/12 , C07D333/16 , C07D333/28 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , A01N43/00 , C07C237/16 , C07D303/16 , C07C327/22 , C07D333/24 , C07C229/30 , A01N37/38 , C07C323/54 , C07D307/54
Abstract: Described are (het)aryloxy-, -thio-, aminocrotonates of formula (I) in which the substituents are defined as follows: U is oxygen, sulphur or amino; V is oxygen, sulphur, amino or alkylamino; X, Y, Z, independently of each other, are =N- or =CR3; R1, R2, independently of each other, are alkyl; R3 is hydrogen, cyano, nitro, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio or alkylthio halide; R4 is an organic group bound directly to the main chain or bound via an oxy, mercapto, amino, carboxy or carbonylamino group. The invention also concerns methods of preparing such compounds and their use.
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公开(公告)号:CA2215514A1
公开(公告)日:1996-10-17
申请号:CA2215514
申请日:1996-03-25
Applicant: BASF AG
Inventor: BAYER HERBERT , R HL FRANZ , WAGNER OLIVER , AMMERMANN EBERHARD , K HLE HARALD
IPC: A01N25/00 , A01N37/50 , A01N43/22 , A01N43/42 , A01N47/18 , A01N61/00 , A01N43/48 , A01N43/64 , A01N43/72 , A01N47/20
Abstract: A process for controlling harmful fungi is characterised in that the fungi, their biotope or materials, plants, seeds, ground, surfaces or rooms to be protected against fungi are treated separately or together, simultaneously or successively with an active substance (I) that inhibits the respiration of cytochrom complex III and with an active substance of formula (II), in which the indices and substituents have the following meanings: m is an integer from 1 to 6, whereas the rests R may differ from each other when m is larger than 1; R stands for hydrogen, cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, sulfo, aminosulphonyl, halogen, alkyl, haydroxyalkyl, alkoxyalkyl, alkoxy, alkoxyalkoxy, alkylthio, alkylamino, dialkylamino, alkylsuphonyl, alkylsulphoxyl, alkylsulphonyloxy, alkylcarbonyl, alkylcarbonyloxy, alkylcarbonylamino, alkoxycarbonyl, alkoxycarbonylamino, alkylaminocarbonyl, dialkylaminocarbonyl, alkylaminothiocarbonyl, dialkylaminothiocarbonyl, alkylaminosulphonyl, dialkylaminosulphonyl, alkenyl, alkenyloxy, alkenylcarbonyloxy, alkinyl and alkinyloxy, whereas these groups may be partially or completely halogenated; cycloalkyl, aryl arylalkyl, arylalkoxy, aryloxy, arylthio, arylcarbonyl, arylcarbonyloxy, heteroaryl, heteroarylalkyl, heteroarylalkoxy, heteroaryloxy, heteroarylthio, heteroarylcarbonyl and heteroarylcarbonyloxy, whereas these groups may be partially or completely halogenated and/or bear one to three of the following rests; cyano, nitro, hydroxy, alkyl, alkyl halide, alkoxy, alkoxy halide or alkylthio; R1 stands for hydrogen, cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbornyl, sulfo, aminosulphonyl, halogen, alkyl, hydroxyalkyl, alkoxyalkyl, alkoxy, alkoxyalkoxy, alkylthio, alkylamino, dialkylamino, alkylsulphonyl, alkylsulphoxyl, alkylsulphonyloxy, alkylcarbonyl, alkylcarbonyloxy, alkylcarbonylamino, alkoxycarbonyl, alkoxycarbonylamino, alkylaminocarbonyl, dialkylaminocarbonyl, alkylaminothiocarbonyl, dialkylaminothiocarbonyl, alkylaminosulphonyl, dialkylaminosulphonyl, alkenyl, alkenyloxy, alkenylcarbonyloxy, alkinyl and alkinyloxy, whereas these groups may be partially or completely halogenated; cycloalkyl, aryl, arylalkyl, arylalkoxy, arylthio, arylcarbonyl, arylcarbonyloxy, heteroaryl, heteroarylalkyl, heteroarylalkoxy, heteroaryloxy, heteroarylthio, heteroarylcarbonyl and heteroarylcarbonyloxy, whereas these groups may be partially or completely halogenated and/or bear one to three of the following rests: cyano, nitro, hydroxy, alkyl, alkyl halide, alkoxy, alkoxy halide or alkylthio. Also disclosed are appropriate mixtures therefor.
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公开(公告)号:CA2206270A1
公开(公告)日:1996-05-30
申请号:CA2206270
申请日:1995-11-10
Applicant: BASF AG
Inventor: MUELLER BERND , LORENZ GISELA , G TZ NORBERT , AMMERMANN EBERHARD , SAUTER HUBERT , R HL FRANZ
IPC: A01N47/24 , A01N47/30 , C07C271/60 , C07D209/48 , C07D239/30 , C07D239/34 , C07D401/04 , C07D403/04 , C07D405/04 , C07D239/26 , A01N43/00 , C07D209/04 , C07D213/56 , C07D213/60 , C07D215/00 , C07D217/00 , C07D237/06 , C07D241/10 , C07D251/14 , C07D253/06 , C07D401/00 , C07D403/00 , C07D405/00 , C07D409/00 , C07D413/00 , C07D417/00 , C07D473/00
Abstract: Iminooxymethylene anilides have the formula (I), in which the indices and substituents have the following meanings: n equals 0, 1, 2, 3 or 4; R stands for nitro, cyano, halogen, optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy or an optionally substituted bridge bound to two adjacent ring atoms; X stands for a direct bond, CH2, O or NRa; Ra stands for hydrogen, alkyl, alkenyl, alkinyl, cycloalkyl or cycloalkenyl; R1 stands for hydrogen, optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, alkylcarbonyl or alkoxycarbonyl; R2 stands for alkyl, alkenyl, alkinyl, cycloalkyl or cycloalkenyl and when X stands for NRa it may also stand for hydrogen; R3 stands for hydrogen, cyano, halogen, alkyl, alkylhalide, alkoxy, alkoxyhalide, alkylthio, alkylthiohalide or cycloalkyl; R4 stands for a substituted 6 to 10-membered monocyclic or bicyclic heteroaromatic ring system. Also disclosed are a process and intermediate products for preparing these compounds and their use.
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公开(公告)号:CA2241219A1
公开(公告)日:1997-07-10
申请号:CA2241219
申请日:1996-12-16
Applicant: BASF AG
Inventor: OBERDORF KLAUS , HARRIES VOLKER , MUELLER BERND , LORENZ GISELA , G TZ NORBERT , RACK MICHAEL , GRAMMENOS WASSILIOS , STRATHMANN SIEGFRIED , AMMERMANN EBERHARD , HARREUS ALBRECHT , GROTE THOMAS , R HL FRANZ , SAUTER HUBERT , KIRSTGEN REINHARD , MUELLER RUTH , BAYER HERBERT
IPC: C07C249/04 , A01N37/50 , A01N43/40 , A01P3/00 , A01P7/00 , C07C251/50 , C07C251/56 , C07C251/58 , C07C251/60 , C07C255/40 , A01N37/36 , A01N43/00 , A01N43/04 , A01N43/48 , A01N43/80 , C07C255/62 , C07C255/64 , C07C323/47 , C07D213/61 , C07D213/63 , C07D231/12 , C07D241/16 , C07D261/08 , C07D309/28 , C07D333/24 , C07D335/02
Abstract: The invention relates to 2-imino oxyphenyl acetic acid derivatives of formula (I) in which the substituents and the index have the following meanings: R1 is C(CO2CH3)=NOCH3 (Ia), C(CONHCH3)=NOCH3 (Ib), C(CONH2)=NOCH3 (Ic), C(CO2CH3)=CHOCH3 (Id), or C(CO2CH3)=CHCH3 (Ie); R2 is cyano, nitro, halogen, alkyl, alkyl halide or alkoxy; m is 0,1 or 2; R3 is hydrogen, cyano, hydroxy, halogen, alkyl, alkyl halide, alkoxy alkyl, alkoxy, alkoxy halide, alkylthio, cyclopropyl, alkenyl, optionally substituted aryloxy alkyl, benzyl or benzyloxy; R4 is hydrogen, cyano, optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, heterocyclyl, aryl and hetaryl, optionally substituted alkoxy, alkenyloxy, alkinyloxy, cycloalkoxy, heterocyclyloxy, aryloxy and hetaryloxy, optionally substituted arylthio and hetarylthio; -Q-C(R5)=N-Y1-R6 or -Q-O-N=CR7R8; R3 and R4 together with the carbon atom to which they are bound, are an optionally substituted four to eight-membered ring which can contain in addition to carbon atoms one or two oxygen atoms and/or sulphur atoms and/or NH- and/or N(C1-C4-alkyl)groups; wherein R3 and R4 are not simultaneously bound via heteroatoms to the carbon atom. The invention also relates to the salts of said derivatives, methods and intermediates for their preparation and use thereof.
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8.
公开(公告)号:CA2225361A1
公开(公告)日:1997-02-20
申请号:CA2225361
申请日:1996-07-22
Applicant: BASF AG
Inventor: SAUTER HUBERT , STRATHMANN SIEGFRIED , AMMERMANN EBERHARD , R HL FRANZ , MUELLER RUTH , BAYER HERBERT , HARREUS ALBRECHT , LORENZ GISELA , HARRIES VOLKER
IPC: C07D261/12 , A01N37/36 , A01N37/50 , A01N37/52 , C07C259/06 , C07C327/58 , C07D261/08 , C07D271/02 , C07D285/04 , C07D261/06 , A01N43/06 , C07D249/08 , C07D231/10 , C07C323/12 , C07C259/14 , C07C317/18 , C07D277/20 , C07D239/24 , C07D333/24 , C07D333/28 , C07D207/30 , C07D263/30 , C07D307/34 , A01N43/34 , C07D303/38 , A01N43/48 , C07D213/54 , C07D233/54 , C07D213/61 , C07D213/63 , A01N43/64 , A01N43/72
Abstract: Hydroximic acid derivatives have the formula (I), in which the substituents have the following meanings: X stands for CH, CHO or NO; Y stands for O or NH; Z stands for O, S or NRa; Ra stands for hydrogen, alkyl, alkenyl or alkinyl; R1 stands for hydrogen, alkyl or halogen alkyl; R2 stands for optionally substituted alkyl, alkenyl, alkinyl or cycloalkyl; R3 stands for optionally substituted alkyl, alkenyl or alkinyl. Also disclosed are a process for preparing these compounds and agents containing the same for controlling animal pests and harmful fungi.
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公开(公告)号:CA2207381A1
公开(公告)日:1996-06-06
申请号:CA2207381
申请日:1995-11-20
Applicant: BASF AG
Inventor: LORENZ GISELA , R HL FRANZ , AMMERMANN EBERHARD , MUELLER BERND , GRAMMENOS WASSILIOS , SAUTER HUBERT , G TZ NORBERT
IPC: C07D237/08 , A01N43/38 , A01N43/40 , A01N43/42 , A01N43/50 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/647 , A01N43/84 , A01N43/90 , C07D213/53 , C07D213/61 , C07D213/63 , C07D213/78 , C07D213/84 , C07D215/12 , C07D215/18 , C07D215/22 , C07D215/42 , C07D215/50 , C07D217/02 , C07D217/22 , C07D217/24 , C07D217/26 , C07D237/10 , C07D239/26 , C07D239/28 , C07D239/34 , C07D241/12 , C07D241/14 , C07D401/04 , C07D401/06 , C07D401/12 , C07D403/04 , C07D403/06 , C07D405/12 , C07D413/04 , C07D473/00 , C07D473/04 , C07D473/28 , C07D473/32 , C07D473/40 , C07D239/24 , C07D217/00 , C07D401/00 , C07D403/00 , C07D405/00 , C07D409/00 , C07D413/00 , C07D417/00 , A01N43/00 , C07D209/04 , C07D237/06 , C07D253/065 , C07D241/10 , C07D251/12 , C07D207/33 , C07D213/55 , C07D213/60
Abstract: The invention concerns iminooxybenzylcrotonic acid esters of formula (I) in which the index and the substituents have the following meanings: n is 0, 1, 2, 3 or 4; R is nitro, cyano, halogen, optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy or, if n stands for 2, additionally an optionally substituted bridge bonded to two adjacent ring atoms; R1 is a C1 to C4 alkyl; R2 is hydrogen or alkyl; R3 is hydrogen, cyano, halogen, alkyl, alkylhalide, alkoxy, alkoxyhalide, alkylthio, alkylthiohalide or cycloalkyl; and R4 is a 5 to 10-member mono or bicyclic substituted heteroaromatic cyclic system. The invention further concerns a process for their preparation and the use thereof.
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公开(公告)号:CA2255555A1
公开(公告)日:1997-11-27
申请号:CA2255555
申请日:1997-05-09
Applicant: BASF AG
Inventor: R HL FRANZ , KIRSTGEN REINHARD , GROTE THOMAS , AMMERMANN EBERHARD , GRAMMENOS WASSILIOS , HARRIES VOLKER , SAUTER HUBERT , MUELLER RUTH , RACK MICHAEL , MUELLER BERND , BAYER HERBERT , OBERDORF KLAUS , STRATHMANN SIEGFRIED , LORENZ GISELA
IPC: C07D239/28 , A01N43/54 , C07D239/34 , C07D239/36 , C07D239/46 , C07D239/52 , A01N43/48 , A01N43/64 , A01N43/713 , A01N43/72 , A01N55/10 , C07D239/47 , C07D239/56 , C07D401/04 , C07D403/04 , C07D405/04 , C07D409/04 , C07D413/04 , C07D417/04 , C07F7/10
Abstract: 2-(O-¢pyrimidin-4-yl! methylene oxy)phenyl acetic acid derivatives of general formula (I) and their salts and N oxides, in which R1 is halogen, alkyl or alkyl halide; R2 is hydrogen, amino, hydroxy, mercapto, halogen, possibly phenyl-substituted alkyl, alkyl halide, alkoxy alkyl, alkoxy, monoalkyl amino, dialkyl amino, alkylthio, alkyl sulphoxyl, alkylsulphonyl, cycloalkyl, trialkyl silyloxy or phenyl, phenoxy, phenoxy methyl, benzyloxy or heteroaryl possibly substituted in the aromatic ring, R2 being different from R1; R3 is hydrogen, cyano, halogen, C1-C4 alkyl, C1-C4 alkyl halide or C1-C4 alkoxy, and Q is C(=CHCH3)-COOCH3 or C(=CHOCH3)-COOCH3, and their use in combatting noxious fungi and animal pests.
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