-
公开(公告)号:HRP20241695T1
公开(公告)日:2025-02-14
申请号:HRP20241695
申请日:2020-12-04
Applicant: VERTEX PHARMA
Inventor: DURRANT STEVEN JOHN , AHMAD NADIA , BECK ELIZABETH MARY , CARVALHO MEIRELES LIDIO , CHUDYK EWA IWONA , ETXEBARRIA JARDI GORKA , GALAN BHAIRAVI , HADIDA RUAH SARA S , HURLEY DENNIS JAMES , KNEGTEL RONALD MARCELLUS , NEUBERT TIMOTHY DONALD , PINDER JOANNE LOUISE , PONTILLO JOSEPH , PULLIN ROBERT , SCHMIDT YVONNE , SHAW DAVID MATTHEW , SKERRATT SARAH , STAMOS DEAN , THOMSON STEPHEN ANDREW , VIRANI ANISA NIZARALI , WRAY CHRISTOPHER
IPC: C07D405/12 , A61K31/443 , A61P29/00 , C07D405/14
-
公开(公告)号:AU2019211485B2
公开(公告)日:2025-01-23
申请号:AU2019211485
申请日:2019-01-28
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: BAYLY ANDREW , BLEICH MATTHEW , CHARRIER JEAN-DAMIEN , DODD JAMES , DURRANT STEVEN , ENO MEREDITH SUZANNE , ETXEBARRIA I JARDI GORKA , EVERITT SIMON , FRAYSSE DAMIEN , KELLY SHAZIA , KNEGTEL RONALD , MOCHALKIN IGOR , MORTIMORE MICHAEL , NORTH KIRI , PORICHIS FILIPPOS , PULLIN ROBERT , RUTHERFORD ALISTAIR , STORCK PIERRE-HENRI , TWIN HEATHER CLARE , XIAO YUFANG
IPC: A61K31/495 , A61K31/505 , A61K31/519 , C07D487/00 , C07D487/02 , C07D487/04
Abstract: The present invention provides compounds, compositions thereof, and methods of using the same.
-
公开(公告)号:SI4069691T1
公开(公告)日:2025-02-28
申请号:SI202030535
申请日:2020-12-04
Applicant: VERTEX PHARMA
Inventor: DURRANT STEVEN JOHN , AHMAD NADIA , BECK ELIZABETH MARY , CARVALHO MEIRELES LIDIO , CHUDYK EWA IWONA , ETXEBARRIA JARDI GORKA , GALAN BHAIRAVI , HADIDA RUAH SARA S , HURLEY DENNIS JAMES , KNEGTEL RONALD MARCELLUS , NEUBERT TIMOTHY DONALD , PINDER JOANNE LOUISE , PONTILLO JOSEPH , PULLIN ROBERT , SCHMIDT YVONNE , SHAW DAVID MATTHEW , SKERRATT SARAH , STAMOS DEAN , THOMSON STEPHEN ANDREW , VIRANI ANISA NIZARALI , WRAY CHRISTOPHER
IPC: C07D405/12 , A61K31/443 , A61P29/00 , C07D405/14
-
公开(公告)号:HUE069128T2
公开(公告)日:2025-02-28
申请号:HUE20825397
申请日:2020-12-04
Applicant: VERTEX PHARMA
Inventor: DURRANT STEVEN , AHMAD NADIA , BECK ELIZABETH , CARVALHO MEIRELES LIDIO , CHUDYK EWA , ETXEBARRIA JARDI GORKA , GALAN BHAIRAVI , HADIDA RUAH SARA , HURLEY DENNIS , KNEGTEL RONALD , NEUBERT TIMOTHY , PINDER JOANNE , PONTILLO JOSEPH , PULLIN ROBERT , SCHMIDT YVONNE , SHAW DAVID , SKERRATT SARAH , STAMOS DEAN , THOMSON STEPHEN , VIRANI ANISA , WRAY CHRISTOPHER
IPC: C07D405/12 , A61P29/00 , C07D405/14
-
公开(公告)号:LT4069691T
公开(公告)日:2024-12-10
申请号:LTUS2020063290
申请日:2020-12-04
Applicant: VERTEX PHARMA
Inventor: DURRANT STEVEN , AHMAD NADIA , BECK ELIZABETH , CARVALHO MEIRELES LIDIO , CHUDYK EWA , ETXEBARRIA JARDI GORKA , GALAN BHAIRAVI , HADIDA RUAH SARA , HURLEY DENNIS , KNEGTEL RONALD , NEUBERT TIMOTHY , PINDER JOANNE , PONTILLO JOSEPH , PULLIN ROBERT , SCHMIDT YVONNE , SHAW DAVID , SKERRATT SARAH , STAMOS DEAN , THOMSON STEPHEN , VIRANI ANISA , WRAY CHRISTOPHER
IPC: C07D405/12 , A61K31/443 , A61P29/00 , C07D405/14
-
公开(公告)号:ES2998396T3
公开(公告)日:2025-02-20
申请号:ES20825397
申请日:2020-12-04
Applicant: VERTEX PHARMA
Inventor: DURRANT STEVEN , AHMAD NADIA , BECK ELIZABETH , CARVALHO MEIRELES LIDIO , CHUDYK EWA , ETXEBARRIA JARDI GORKA , GALAN BHAIRAVI , HADIDA RUAH SARA , HURLEY DENNIS , KNEGTEL RONALD , NEUBERT TIMOTHY , PINDER JOANNE , PONTILLO JOSEPH , PULLIN ROBERT , SCHMIDT YVONNE , SHAW DAVID , SKERRATT SARAH , STAMOS DEAN , THOMSON STEPHEN , VIRANI ANISA , WRAY CHRISTOPHER
IPC: C07D405/12 , A61K31/443 , A61P29/00 , C07D405/14
Abstract: Se proporcionan compuestos y sales farmacéuticamente aceptables de los mismos, útiles como inhibidores de los canales de sodio. También se proporcionan composiciones farmacéuticas que comprenden los compuestos o sales farmacéuticamente aceptables y métodos de uso de los compuestos, sales farmacéuticamente aceptables y composiciones farmacéuticas en el tratamiento de diversos trastornos, incluido el dolor. (Traducción automática con Google Translate, sin valor legal)
-
公开(公告)号:PL4069691T3
公开(公告)日:2025-01-27
申请号:PL20825397
申请日:2020-12-04
Applicant: VERTEX PHARMA
Inventor: DURRANT STEVEN JOHN , AHMAD NADIA , BECK ELIZABETH MARY , CARVALHO MEIRELES LIDIO , CHUDYK EWA IWONA , ETXEBARRIA JARDI GORKA , GALAN BHAIRAVI , HADIDA RUAH SARA S , HURLEY DENNIS JAMES , KNEGTEL RONALD MARCELLUS , NEUBERT TIMOTHY DONALD , PINDER JOANNE LOUISE , PONTILLO JOSEPH , PULLIN ROBERT , SCHMIDT YVONNE , SHAW DAVID MATTHEW , SKERRATT SARAH , STAMOS DEAN , THOMSON STEPHEN ANDREW , VIRANI ANISA NIZARALI , WRAY CHRISTOPHER
IPC: C07D405/12 , A61K31/443 , A61P29/00 , C07D405/14
-
公开(公告)号:SG11202006832YA
公开(公告)日:2020-08-28
申请号:SG11202006832Y
申请日:2019-01-28
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: BLEICH MATTHEW , CHARRIER JEAN-DAMIEN , DONG HUIJUN , DURRANT STEVEN , ENO MEREDITH SUZANNE , ETXEBARRIA I JARDI GORKA , EVERITT SIMON , FRAYSSE DAMIEN , KNEGTEL RONALD , MOCHALKIN IGOR , NORTH KIRI , PORICHIS FILIPPOS , PULLIN ROBERT , QIU HUI , STORCK PIERRE-HENRI , TWIN HEATHER CLARE , XIAO YUFANG
IPC: A61K31/395 , A61K31/437 , A61K31/4375 , C07D231/02 , C07D471/04 , C07D487/04
Abstract: The present invention provides compounds, compositions thereof, and methods of using the same.
-
公开(公告)号:MD4069691T2
公开(公告)日:2025-03-31
申请号:MDE20221109
申请日:2020-12-04
Applicant: VERTEX PHARMA
Inventor: DURRANT STEVEN JOHN , AHMAD NADIA , BECK ELIZABETH MARY , CARVALHO MEIRELES LIDIO , CHUDYK EWA IWONA , ETXEBARRIA JARDI GORKA , GALAN BHAIRAVI , HADIDA RUAH SARA S , HURLEY DENNIS JAMES , KNEGTEL RONALD MARCELLUS , NEUBERT TIMOTHY DONALD , PINDER JOANNE LOUISE , PONTILLO JOSEPH , PULLIN ROBERT , SCHMIDT YVONNE , SHAW DAVID MATTHEW , SKERRATT SARAH , STAMOS DEAN , THOMSON STEPHEN ANDREW , VIRANI ANISA NIZARALI , WRAY CHRISTOPHER
IPC: C07D405/12 , A61K31/443 , A61P29/00 , C07D405/14
Abstract: Sunt furnizaţi compuşi şi săruri acceptabile farmaceutic ale acestora, utile ca inhibitori ai canalelor de sodiu. Sunt de asemenea furnizate compoziţii farmaceutice care cuprind compuşii sau sărurile acceptabile farmaceutic şi metode de utilizare a compuşilor, sărurilor acceptabile farmaceutic şi compoziţiilor farmaceutice ȋn tratarea a diferite tulburări, incluzând durere.
-
公开(公告)号:RS66307B1
公开(公告)日:2025-01-31
申请号:RSP20241330
申请日:2020-12-04
Applicant: VERTEX PHARMA
Inventor: DURRANT STEVEN JOHN , AHMAD NADIA , BECK ELIZABETH MARY , CARVALHO MEIRELES LIDIO , CHUDYK EWA IWONA , ETXEBARRIA JARDI GORKA , GALAN BHAIRAVI , HADIDA RUAH SARA S , HURLEY DENNIS JAMES , KNEGTEL RONALD MARCELLUS , NEUBERT TIMOTHY DONALD , PINDER JOANNE LOUISE , PONTILLO JOSEPH , PULLIN ROBERT , SCHMIDT YVONNE , SHAW DAVID MATTHEW , SKERRATT SARAH , STAMOS DEAN , THOMSON STEPHEN ANDREW , VIRANI ANISA NIZARALI , WRAY CHRISTOPHER
IPC: C07D405/12 , A61K31/443 , A61P29/00 , C07D405/14
-
-
-
-
-
-
-
-
-