New amino-pyridinoazine derivatives, useful as fungicides for protection of plants and materials, also new intermediates in their synthesis

    公开(公告)号:DE102005051514A1

    公开(公告)日:2007-05-03

    申请号:DE102005051514

    申请日:2005-10-26

    Applicant: BASF AG

    Abstract: Amino-substituted pyridinoazines (I) are new. Amino-substituted pyridinoazines of formula (I) are new. R1>1-14C alkyl, 1-12C alkoxy(1-12C)alkyl, 1-6C alkoxy(2-12C)-alkenyl or -alkynyl, 5-8C cycloalkyl, phenyl, phenyl(1-4C)alkyl, 2-12C alkenyl or alkynyl, where the carbon chain may be substituted by 1-3, same or different, Ra> and/or Rb>; Ra>halo, cyano, nitro, hydroxy, 1-6C alkylthio, 3-12C alkenyloxy or alkynyloxy, NR11>R12>, or phenyl or 3-6C cycloalkyl optionally substituted by 1-4, same or different, Rb>, and carbon chains in Ra> may themselves be halogenated; Rb>halo, cyano, hydroxy, mercapto, 1-6C (halo)alkyl, 3-8C cycloalkyl, 2-10C alkenyl or alkynyl, 1-6C alkoxy or alkylthio, 1-6C alkoxy(1-6C)alkyl or NR11>R12>; R11> and R12>hydrogen or 1-6C alkyl; R2>1-12C alkyl, or 2-12C alkenyl or alkynyl, optionally substituted by 1-3 Rc>; Rc>cyano, nitro, hydroxy, NR11>R12> or 3-6C cycloalkyl (optionally substituted by 1-4 of, same or different, 1-4C alkyl, halo, cyano, nitro, hydroxy, 1-6C alkoxy or alkylthio, 3-6C alkenyloxy or alkynyloxy, or NR11>R12>; W1 and X1, W1 and Y1, W1 and Z1, X1 and Y1, X1 and Z1, or Y1 and Z1 each : N and the others CR3>, or W1, Z1 and one of X1 and Y1 = N and the other CR3>; each R3>hydrogen, halo, or 1-4C alkyl or alkoxy . Independent claims are included for the following: (1) several methods for preparing (I); (2) intermediates of formulae (V), (VI), (VII) and (IX); and (3) seeds treated with (I) at 1-1000 g per 100 kg. in (VI) and (VII) X on the pyrido ring : halo; R22>hydrogen or 1-11C alkyl; R : 1-4C alkyl . [Image] [Image] ACTIVITY : Plant Antifungal. No details of tests for antifungal activity are given. MECHANISM OF ACTION : None given.

    85.
    发明专利
    未知

    公开(公告)号:BRPI0417765A

    公开(公告)日:2007-04-17

    申请号:BRPI0417765

    申请日:2004-12-17

    Applicant: BASF AG

    Abstract: Triazolopyrimidines of the formula I in which the substituents are as defined below: R 1 , R 2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R 1 and R 2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and may be substituted as defined in the description; L is halogen, cyano, alkyl, haloalkyl, alkoxy, alkenyloxy or alkoxycarbonyl; m is 1, 2, 3 or 4, where the groups L may be different if m is greater than 1; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi

    87.
    发明专利
    未知

    公开(公告)号:BRPI0417628A

    公开(公告)日:2007-03-27

    申请号:BRPI0417628

    申请日:2004-12-14

    Applicant: BASF AG

    Abstract: The present invention relates to 6-(2,4,6-trihalophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R 1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-member saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R 2 is hydrogen or one of the groups mentioned under R 1 , R 1 and R 2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R 1 and/or R 2 may be substituted as defined in the description; L 1 , L 2 , L 3 are chlorine or fluorine, where at least one group is chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

    89.
    发明专利
    未知

    公开(公告)号:BRPI0416849A

    公开(公告)日:2007-02-27

    申请号:BRPI0416849

    申请日:2004-11-18

    Applicant: BASF AG

    Abstract: 6-(2,4,6-Trifluorophenyl)triazolopyrimidines of the formula I in which the substituents have the following meanings: R 1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl, cycloalkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R 2 is hydrogen or one of the groups mentioned in R 1 , R 1 and R 2 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered ring which is interrupted by an atom from the group consisting of O, N and S, and/or R 1 and/or R 2 can be substituted according to the description; X is cyano, C 1 -C 4 -alkoxy, C 3 -C 4 -alkenyloxy, C 1 -C 2 -haloalkoxy or C 3 -C 4 -halo-alkenyloxy; process for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.

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