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公开(公告)号:HRP20190660T1
公开(公告)日:2019-05-31
申请号:HRP20190660
申请日:2010-02-18
Applicant: VERTEX PHARMA
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公开(公告)号:PL2328618T3
公开(公告)日:2018-06-29
申请号:PL09789125
申请日:2009-08-13
Applicant: VERTEX PHARMA
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公开(公告)号:HRP20180328T1
公开(公告)日:2018-04-20
申请号:HRP20180328
申请日:2018-02-22
Applicant: VERTEX PHARMA
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64.
公开(公告)号:AU2016219571B2
公开(公告)日:2018-03-15
申请号:AU2016219571
申请日:2016-08-23
Applicant: VERTEX PHARMA
Inventor: HURTER PATRICIA , CONNELLY PATRICK , ROWE WILLIAM , YOUNG CHRISTOPHER R , COSTACHE ADRIANA , KRAWIEC MARIUSZ , GONG YUCHUAN , FENG YUSHI , TRUDEAU MARTIN
IPC: A61K31/445
Abstract: The present invention relates to solid state forms of N-[2,4-bis(1,1 -dimethylethyl)-5 hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide (Compound 1), pharmaceutical compositions thereof and methods therewith.
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65.
公开(公告)号:RS55940B1
公开(公告)日:2017-09-29
申请号:RSP20170454
申请日:2006-12-28
Applicant: VERTEX PHARMA
Inventor: HURTER PATRICIA , GONG YUCHUAN , YOUNG CHRISTOPHER R , CONNELLY PATRICK , ROWE WILLIAM , COSTACHE ADRIANA , KRAWIEC MARIUSZ , FENG YUSHI , TRUDEAU MARTIN
IPC: C07D215/56 , A61K31/445
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66.
公开(公告)号:LT1993360T
公开(公告)日:2017-06-12
申请号:LT06848237
申请日:2006-12-28
Applicant: VERTEX PHARMA
Inventor: HURTER PATRICIA , GONG YUCHUAN , YOUNG CHRISTOPHER R , CONNELLY PATRICK , ROWE WILLIAM , COSTACHE ADRIANA , KRAWIEC MARIUSZ , FENG YUSHI , TRUDEAU MARTIN
IPC: C07D215/56 , A61K31/445
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公开(公告)号:CA2733908C
公开(公告)日:2017-05-30
申请号:CA2733908
申请日:2009-08-13
Applicant: VERTEX PHARMA
Inventor: ROWE WILLIAM , HURTER PATRICIA , YOUNG CHRISTOPHER , DINEHART KIRK , VERWIJS MARINUS JACOBUS , OVERHOFF KIRK , GROOTENHUIS PETER D J , BOTFIELD MARTYN , GROSSI ALFREDO
IPC: A61K47/32
Abstract: The present invention relates to pharmaceutical compositions comprising a solid dispersion of N- [2,4-Bis( 1, 1-dimethylethyl)-5 -hydroxyphenyl]- 1,4-dihydro-4-oxoquinoline-3-carboxamide, and a polymer, wherein Compound 1 is present in an amount of about 80% by weight of the solid dispersion.
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68.
公开(公告)号:CA2635581C
公开(公告)日:2017-02-28
申请号:CA2635581
申请日:2006-12-28
Applicant: VERTEX PHARMA
Inventor: HURTER PATRICIA , YOUNG CHRISTOPHER R , COSTACHE ADRIANA , CONNELLY PATRICK , KRAWIEC MARIUSZ , GONG YUCHUAN , ROWE WILLIAM , FENG YUSHI , TRUDEAU MARTIN
IPC: C07D215/56 , A61K31/47 , A61P11/00
Abstract: The present invention relates to solid state forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide (Compound I ), and pharmaceutical compositions thereof.
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69.
公开(公告)号:AU2013201426B2
公开(公告)日:2016-06-02
申请号:AU2013201426
申请日:2013-03-12
Applicant: VERTEX PHARMA
Inventor: HURTER PATRICIA , ROWE WILLIAM , YOUNG CHRISTOPHER R , COSTACHE ADRIANA , CONNELLY PATRICK , KRAWIEC MARIUSZ , GONG YUCHUAN , TRUDEAU MARTIN , FENG YUSHI
IPC: A61K31/445
Abstract: The present invention relates to solid state forms of N-[2,4-bis(1 ,1-dimethylethyl)-5 hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide (Compound 1), pharmaceutical compositions thereof and methods therewith.
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公开(公告)号:BRPI0916877A2
公开(公告)日:2016-02-10
申请号:BRPI0916877
申请日:2009-08-13
Applicant: VERTEX PHARMA
Inventor: GROSSI ALFREDO , YOUNG CHRISTOPHER , OVERHOFF KIRK , DINEHART KRIK , VERWIJS MARINUS JACOBUS , BOTFIELD MARTYN , HURTER PATRICIA , GROOTENHUIS PETER D J , ROWE WILLIAM
IPC: A61K47/32
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