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公开(公告)号:AT177420T
公开(公告)日:1999-03-15
申请号:AT94931987
申请日:1994-10-20
Applicant: ABBOTT LAB
Inventor: BAKER WILLIAM R , ROCKWAY TODD W , DONNER B GREGORY , SHEN WANG , ROSENBERG SAUL H , FAKHOURY STEPHEN A , O'CONNOR STEPHEN J , STOUT DAVID M , FUNG ANTHONY K L , GARVEY DAVID S , PRASAD RAJNANDAN , SULLIVAN GERARD M
IPC: C12N9/99 , A61K31/195 , A61K31/215 , A61K31/34 , A61K31/341 , A61K31/357 , A61K31/36 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/41 , A61K31/42 , A61K31/421 , A61K31/4245 , A61K31/44 , A61K31/4409 , A61K31/4418 , A61P3/06 , A61P7/00 , A61P9/10 , A61P31/04 , A61P43/00 , C07C69/52 , C07C69/74 , C07C231/02 , C07C233/19 , C07C233/58 , C07C233/59 , C07C233/60 , C07C233/61 , C07C233/62 , C07C233/63 , C07C235/36 , C07C235/40 , C07C237/24 , C07C245/14 , C07C251/42 , C07C259/08 , C07C275/26 , C07C311/51 , C07C323/40 , C07C323/46 , C07C327/20 , C07C327/36 , C07C327/38 , C07D207/325 , C07D213/40 , C07D257/04 , C07D257/06 , C07D263/24 , C07D271/06 , C07D271/10 , C07D277/20 , C07D277/34 , C07D285/16 , C07D285/18 , C07D307/42 , C07D307/52 , C07D309/32 , C07D317/60 , C07D319/06 , C07D333/08 , C07D333/58 , A61K31/16
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公开(公告)号:DK0677039T3
公开(公告)日:1999-09-27
申请号:DK94931987
申请日:1994-10-20
Applicant: ABBOTT LAB
Inventor: BAKER WILLIAM R , DONNER B GREGORY , FAKHOURY STEPHEN A , FUNG ANTHONY K L , GARVEY DAVID S , O'CONNOR STEPHEN J , PRASAD RAJNANDAN , ROCKWAY TODD W , ROSENBERG SAUL H , SHEN WANG , STOUT DAVID M , SULLIVAN GERARD M
IPC: C12N9/99 , A61K31/195 , A61K31/215 , A61K31/34 , A61K31/341 , A61K31/357 , A61K31/36 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/41 , A61K31/42 , A61K31/421 , A61K31/4245 , A61K31/44 , A61K31/4409 , A61K31/4418 , A61P3/06 , A61P7/00 , A61P9/10 , A61P31/04 , A61P43/00 , C07C69/52 , C07C69/74 , C07C231/02 , C07C233/19 , C07C233/58 , C07C233/59 , C07C233/60 , C07C233/61 , C07C233/62 , C07C233/63 , C07C235/36 , C07C235/40 , C07C237/24 , C07C245/14 , C07C251/42 , C07C259/08 , C07C275/26 , C07C311/51 , C07C323/40 , C07C323/46 , C07C327/20 , C07C327/36 , C07C327/38 , C07D207/325 , C07D213/40 , C07D257/04 , C07D257/06 , C07D263/24 , C07D271/06 , C07D271/10 , C07D277/20 , C07D277/34 , C07D285/16 , C07D285/18 , C07D307/42 , C07D307/52 , C07D309/32 , C07D317/60 , C07D319/06 , C07D333/08 , C07D333/58 , A61K31/16
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公开(公告)号:AU5673196A
公开(公告)日:1996-11-21
申请号:AU5673196
申请日:1996-05-02
Applicant: ABBOTT LAB
Inventor: BAKER WILLIAM R , ROSENBERG SAUL H , FUNG K L ANTHONY , ROCKWAY TODD W , FAKHOURY STEPHEN A , GARVEY DAVID S , DONNER B GREGORY , O'CONNOR STEPHEN J , PRASAD RAJNANDAN N , SHEN WANG , STOUT DAVID M , SULLIVAN GERARD M
IPC: C07C65/24 , C07C65/28 , C07C65/40 , C07C69/94 , C07C229/38 , C07C233/22 , C07C233/65 , C07C233/69 , C07C233/73 , C07C233/87 , C07C235/16 , C07C235/34 , C07C235/42 , C07C235/48 , C07C235/60 , C07C235/84 , C07C237/08 , C07C237/20 , C07C237/32 , C07C251/48 , C07C255/57 , C07C259/10 , C07C271/48 , C07C275/42 , C07C311/08 , C07C311/29 , C07C311/51 , C07C323/59 , C07C327/48 , C07C333/04 , C07D209/16 , C07D213/40 , C07D231/12 , C07D271/10 , C07D271/113 , C07D307/88 , C07D307/89 , C07D309/32 , C07D311/68 , C07D319/06 , C07D333/20 , C07C235/38 , C07D257/04 , C07C335/22 , C07C233/12
Abstract: The present invention provides a compound of the formula which inhibit squalene synthetase and cholesterol biosynthesis and are useful in the treatment of e.g., hyperlipidaemia, atherosclerosis, or fungal infections, processes for the preparation of the compounds of the invention, intermediates useful in these processes, and pharmaceutical compositions containing the compounds.
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公开(公告)号:AU2044495A
公开(公告)日:1996-08-01
申请号:AU2044495
申请日:1995-06-01
Applicant: ABBOTT LAB
Inventor: STEIN HERMAN H , BAKER WILLIAM R , FUNG ANTHONY K L , ROSENBERG SAUL H , ROCKWAY TODD W , FAKHOURY STEPHEN A , GARVEY DAVID S , DONNER B GREGORY , MCCLELLAN WILLIAM J , O'CONNOR STEPHEN J , PRASAD RAJNANDAN , SHEN WANG , SULLIVAN GERARD M
IPC: A61K31/19 , C07C20060101 , C07C69/74 , C07C233/58 , C07C233/59 , C07C233/60 , C07C233/62 , C07C233/63 , C07C323/40 , C07D207/32 , C07D211/16 , C07D211/70 , C07D217/16 , C07D277/34 , C07D307/58 , C07D307/91 , C07D317/64 , C07D333/32
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5.
公开(公告)号:GR3030342T3
公开(公告)日:1999-09-30
申请号:GR990401431
申请日:1999-05-27
Applicant: ABBOTT LAB
Inventor: BAKER WILLIAM R , ROCKWAY TODD W , DONNER B GREGORY , SHEN WANG , ROSENBERG SAUL H , FAKHOURY STEPHEN A , O'CONNOR STEPHEN J , STOUT DAVID M , FUNG ANTHONY K L , GARVEY DAVID S , PRASAD RAJNANDAN , SULLIVAN GERARD M
IPC: C12N9/99 , A61K31/195 , A61K31/215 , A61K31/34 , A61K31/341 , A61K31/357 , A61K31/36 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/41 , A61K31/42 , A61K31/421 , A61K31/4245 , A61K31/44 , A61K31/4409 , A61K31/4418 , A61P3/06 , A61P7/00 , A61P9/10 , A61P31/04 , A61P43/00 , C07C69/52 , C07C69/74 , C07C231/02 , C07C233/19 , C07C233/58 , C07C233/59 , C07C233/60 , C07C233/61 , C07C233/62 , C07C233/63 , C07C235/36 , C07C235/40 , C07C237/24 , C07C245/14 , C07C251/42 , C07C259/08 , C07C275/26 , C07C311/51 , C07C323/40 , C07C323/46 , C07C327/20 , C07C327/36 , C07C327/38 , C07D207/325 , C07D213/40 , C07D257/04 , C07D257/06 , C07D263/24 , C07D271/06 , C07D271/10 , C07D277/20 , C07D277/34 , C07D285/16 , C07D285/18 , C07D307/42 , C07D307/52 , C07D309/32 , C07D317/60 , C07D319/06 , C07D333/08 , C07D333/58 , A61K31/16
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公开(公告)号:ES2130452T3
公开(公告)日:1999-07-01
申请号:ES94931987
申请日:1994-10-20
Applicant: ABBOTT LAB
Inventor: BAKER WILLIAM R , ROCKWAY TODD W , DONNER B GREGORY , SHEN WANG , ROSENBERG SAUL H , FAKHOURY STEPHEN A
IPC: C12N9/99 , A61K31/195 , A61K31/215 , A61K31/34 , A61K31/341 , A61K31/357 , A61K31/36 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/41 , A61K31/42 , A61K31/421 , A61K31/4245 , A61K31/44 , A61K31/4409 , A61K31/4418 , A61P3/06 , A61P7/00 , A61P9/10 , A61P31/04 , A61P43/00 , C07C69/52 , C07C69/74 , C07C231/02 , C07C233/19 , C07C233/58 , C07C233/59 , C07C233/60 , C07C233/61 , C07C233/62 , C07C233/63 , C07C235/36 , C07C235/40 , C07C237/24 , C07C245/14 , C07C251/42 , C07C259/08 , C07C275/26 , C07C311/51 , C07C323/40 , C07C323/46 , C07C327/20 , C07C327/36 , C07C327/38 , C07D207/325 , C07D213/40 , C07D257/04 , C07D257/06 , C07D263/24 , C07D271/06 , C07D271/10 , C07D277/20 , C07D277/34 , C07D285/16 , C07D285/18 , C07D307/42 , C07D307/52 , C07D309/32 , C07D317/60 , C07D319/06 , C07D333/08 , C07D333/58 , A61K31/16
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7.
公开(公告)号:CA2152822A1
公开(公告)日:1995-05-11
申请号:CA2152822
申请日:1994-10-20
Applicant: ABBOTT LAB
Inventor: BAKER WILLIAM R , ROCKWAY TODD W , DONNER B GREGORY , SHEN WANG , ROSENBERG SAUL H , FAKHOURY STEPHEN A , O'CONNOR STEPHEN J , STOUT DAVID M , FUNG ANTHONY K L , GARVEY DAVID S , PRASAD RAJNANDAN , SULLIVAN GERARD M
IPC: C12N9/99 , A61K31/195 , A61K31/215 , A61K31/34 , A61K31/341 , A61K31/357 , A61K31/36 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/41 , A61K31/42 , A61K31/421 , A61K31/4245 , A61K31/44 , A61K31/4409 , A61K31/4418 , A61P3/06 , A61P7/00 , A61P9/10 , A61P31/04 , A61P43/00 , C07C69/52 , C07C69/74 , C07C231/02 , C07C233/19 , C07C233/58 , C07C233/59 , C07C233/60 , C07C233/61 , C07C233/62 , C07C233/63 , C07C235/36 , C07C235/40 , C07C237/24 , C07C245/14 , C07C251/42 , C07C259/08 , C07C275/26 , C07C311/51 , C07C323/40 , C07C323/46 , C07C327/20 , C07C327/36 , C07C327/38 , C07D207/325 , C07D213/40 , C07D257/04 , C07D257/06 , C07D263/24 , C07D271/06 , C07D271/10 , C07D277/20 , C07D277/34 , C07D285/16 , C07D285/18 , C07D307/42 , C07D307/52 , C07D309/32 , C07D317/60 , C07D319/06 , C07D333/08 , C07D333/58 , C07C235/82 , A61K31/33 , C07D207/337 , C07D249/02 , C07D285/06 , C07D307/54 , C07D333/24
Abstract: The present invention provides a compound of formula (I) processes for the preparation of the compounds of the invention in addition to intermediates useful in these processes, a pharmaceutical composition, and a method of treating disorders resulting from an excess of cholesterol or cancer or a fungal infection.
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