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公开(公告)号:CY1107815T1
公开(公告)日:2013-06-19
申请号:CY071101525
申请日:2007-11-29
Applicant: ABBOTT LAB
Inventor: BENNANI YOUSSEF L , FAGHIH RAMIN , DWIGHT WESLEY J , VASUDEVAN ANIL , CONNER SCOTT E
IPC: C07D207/12 , C07D295/08 , A61K31/40 , A61K31/4025 , A61K31/4178 , A61K31/427 , A61K31/443 , A61K31/4439 , A61K31/455 , A61K31/4709 , A61K31/4725 , A61K31/496 , A61K31/506 , A61K31/5377 , A61P3/04 , A61P9/10 , A61P11/06 , A61P25/06 , A61P25/08 , A61P25/16 , A61P25/18 , A61P25/24 , A61P25/28 , A61P29/00 , A61P31/04 , A61P35/00 , A61P43/00 , C07D207/06 , C07D207/14 , C07D207/16 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/12 , C07D405/12 , C07D409/12 , C07D417/12 , C07D417/14
Abstract: Ενώσειτουτύπου (Ι) είναιχρήσιμοιειςνοσήλειαννόσωνή καταστάσεωνπαρεμποδιζομένωνυπόβελτιουμένωνδιασυνδεσμικώνμέσωνυποδοχέωςισταμίνης-3. Επίσηςαποκαλύπτονταισυνθέσειςσυνδεσμικούμέσουυποδοχέωςισταμίνης-3 καιμέθοδοιανταγωνισμούή συναγωνισμούυποδοχέωνισταμίνης-3.
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公开(公告)号:CA2566896C
公开(公告)日:2012-10-30
申请号:CA2566896
申请日:2005-04-29
Applicant: ABBOTT LAB
Inventor: ALTENBACH ROBERT J , BLACK LAWRENCE A , CHANG SOU-JEN , COWART MARLON D , FAGHIH RAMIN , GFESSER GREGORY A , KU YI-YIN , LIU HUAQING , LUKIN KIRILL A , NERSESIAN DIANA L , PU YU-MING , CURTIS MICHAEL P
IPC: C07D417/14 , A61K31/4709 , A61P25/00 , A61P25/28 , C07D215/12 , C07D401/04 , C07D401/08 , C07D401/14 , C07D409/14 , C07D413/04 , C07D413/14 , C07D417/04
Abstract: Compounds of formula (I) wherein R1 or R2 is an aromatic or non-aromatic ring directly joined or joined by a linker, as represented by L2and L3, to a heteroaromatic core, and X, X', Y, Y', Z, Z', R1, R2, R3, R3a, R3b, R4, R5, L, L2, and L3 are as defined herein, are useful in treating conditions or disorders prevented by or ameliorated by histamine-3 receptor ligands. Also disclosed are pharmaceutical compositions comprising the histamine-3 receptor ligands, methods for using such compounds and compositions, and a process for preparing compounds within the scope of formula (I).
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公开(公告)号:BRPI0712667A2
公开(公告)日:2012-09-04
申请号:BRPI0712667
申请日:2007-06-27
Applicant: ABBOTT LAB
Inventor: FAGHIH RAMIN , GFESSER GREGORY A , LYNCH CHRISTOPHER L , GOPALAKRISHNAN MURALI , GOPALAKRISHNAN SUJATHA , MALYSZ JOHN , GUBBINS EARL J , EL KOUHEN RACHID , LI JINHE
IPC: C07D207/34 , A61K31/402 , A61P25/00 , C07D401/10 , C07D403/10 , C07D405/10 , C07D409/10
Abstract: The invention relates to a series of substituted pyrrole derivatives, compositions comprising the same, and methods of treating conditions and disorders using such compounds and compositions.
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公开(公告)号:CA2440238C
公开(公告)日:2011-09-13
申请号:CA2440238
申请日:2002-03-11
Applicant: ABBOTT LAB
Inventor: COWART MARLON D , BENNANI YOUSSEF L , FAGHIH RAMIN , GFESSER GREGORY A , BLACK LAWRENCE A
IPC: C07D307/79 , A61K31/343 , A61K31/4025 , A61K31/4245 , A61K31/427 , A61K31/437 , A61K31/4427 , A61K31/4439 , A61K31/5377 , A61K31/55 , A61P1/00 , A61P1/08 , A61P3/04 , A61P7/08 , A61P9/00 , A61P9/10 , A61P11/02 , A61P11/06 , A61P25/00 , A61P25/04 , A61P25/06 , A61P25/08 , A61P25/14 , A61P25/16 , A61P25/18 , A61P25/20 , A61P25/22 , A61P25/24 , A61P25/28 , A61P25/30 , A61P29/00 , A61P31/04 , A61P35/00 , A61P43/00 , C07D307/81 , C07D311/18 , C07D333/54 , C07D405/04 , C07D405/06 , C07D405/14 , C07D407/04 , C07D409/04 , C07D409/10 , C07D409/14 , C07D413/04 , C07D413/14 , C07D417/04 , C07D417/14 , C07D471/04 , C07D491/08 , C07D491/10 , C07D521/00
Abstract: Compounds of formula (I), or a pharmaceutically acceptable salt, ester, amide, or prodrug thereof, which are useful for the modulation of the histamine-3 receptors in mammals and which are useful for the treatment of disorders ameliorated by histamine-3 receptor ligands.
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公开(公告)号:MX2011003435A
公开(公告)日:2011-05-02
申请号:MX2011003435
申请日:2009-09-28
Applicant: ABBOTT LAB
Inventor: BUNNELLE WILLIAM H , FAGHIH RAMIN , GFESSER GREGORY A , NERSESIAN DIANA L , SHI LEI , LEE CHIH-HUNG , MORTELL KATHLEEN H , SCHRIMPF MICHAEL R , LI TAO , SIPPY KEVIN B , GOPALAKRISHNAN MURALI , SCANIO MARC , DONNELLY-ROBERTS DIANA , HU MIN
IPC: C07D487/18 , A61K31/33 , A61P25/00
Abstract: La presente solicitud se refiere a derivados de indol e indolina de las fórmulas (I), (II), (III), (IV), (y), o (VI), en las cuales R1, R2, R3, R4, R5, U, V, W, X, Y, y Z son como se definen en la descripción. La presente solicitud también se refiere a composiciones que comprenden dichos compuestos, y a métodos para tratar condiciones patológicas utilizando dichos compuestos y composiciones, y a métodos para identificar dichos compuestos.
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公开(公告)号:ZA200808757B
公开(公告)日:2010-03-31
申请号:ZA200808757
申请日:2008-10-14
Applicant: ABBOTT LAB
Inventor: FAGHIH RAMIN , GFESSER GREGORY A , LYNCH CHRISTOPHER L , GOPALAKRISHNAN MURALI , GOPALAKRISHNAN SUJATHA , MALYSZ JOHN , GUBBINS EARL J , EL KOUHEN RACHID , LI JINHE
IPC: A61K20100101 , A61P20100101 , C07D20100101
Abstract: The invention relates to a series of substituted pyrrole derivatives, compositions comprising the same, and methods of treating conditions and disorders using such compounds and compositions.
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公开(公告)号:CA2709676A1
公开(公告)日:2009-07-09
申请号:CA2709676
申请日:2008-12-19
Applicant: ABBOTT LAB
Inventor: FAGHIH RAMIN , GFESSER GREGORY A , MORTELL KATHLEEN H , GOPALAKRISHNAN MURALI
IPC: C07D277/02 , A61P25/00 , C07D277/50
Abstract: The invention relates to novel thiazolylidine urea and amide derivatives that are PAMs of neuronal nicotinic receptors, compositions comprising the same, processes for preparing such compounds, and methods for using such compounds and compositions.
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公开(公告)号:DK1301480T3
公开(公告)日:2008-01-21
申请号:DK01952653
申请日:2001-07-11
Applicant: ABBOTT LAB
Inventor: BENNANI YOUSSEF L , FAGHIH RAMIN , DWIGHT WESLEY J , VASUDEVAN ANIL , CONNER SCOTT E
IPC: C07D207/12 , C07D295/08 , A61K31/40 , A61K31/4025 , A61K31/4178 , A61K31/427 , A61K31/443 , A61K31/4439 , A61K31/455 , A61K31/4709 , A61K31/4725 , A61K31/496 , A61K31/506 , A61K31/5377 , A61P3/04 , A61P9/10 , A61P11/06 , A61P25/06 , A61P25/08 , A61P25/16 , A61P25/18 , A61P25/24 , A61P25/28 , A61P29/00 , A61P31/04 , A61P35/00 , A61P43/00 , C07D207/06 , C07D207/14 , C07D207/16 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/12 , C07D405/12 , C07D409/12 , C07D417/12 , C07D417/14
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公开(公告)号:PT1301480E
公开(公告)日:2007-11-29
申请号:PT01952653
申请日:2001-07-11
Applicant: ABBOTT LAB
Inventor: FAGHIH RAMIN , BENNANI YOUSSEF L , DWIGHT WESLEY J , VASUDEVAN ANIL , CONNER SCOTT E
IPC: C07D207/12 , C07D295/08 , A61K31/40 , A61K31/4025 , A61K31/4178 , A61K31/427 , A61K31/443 , A61K31/4439 , A61K31/455 , A61K31/4709 , A61K31/4725 , A61K31/496 , A61K31/506 , A61K31/5377 , A61P3/04 , A61P9/10 , A61P11/06 , A61P25/06 , A61P25/08 , A61P25/16 , A61P25/18 , A61P25/24 , A61P25/28 , A61P29/00 , A61P31/04 , A61P35/00 , A61P43/00 , C07D207/06 , C07D207/14 , C07D207/16 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/12 , C07D405/12 , C07D409/12 , C07D417/12 , C07D417/14
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公开(公告)号:DE60130460D1
公开(公告)日:2007-10-25
申请号:DE60130460
申请日:2001-07-11
Applicant: ABBOTT LAB
Inventor: BENNANI YOUSSEF L , FAGHIH RAMIN , DWIGHT WESLEY J , VASUDEVAN ANIL , CONNER SCOTT E
IPC: C07D207/12 , C07D295/08 , A61K31/40 , A61K31/4025 , A61K31/4178 , A61K31/427 , A61K31/443 , A61K31/4439 , A61K31/455 , A61K31/4709 , A61K31/4725 , A61K31/496 , A61K31/506 , A61K31/5377 , A61P3/04 , A61P9/10 , A61P11/06 , A61P25/06 , A61P25/08 , A61P25/16 , A61P25/18 , A61P25/24 , A61P25/28 , A61P29/00 , A61P31/04 , A61P35/00 , A61P43/00 , C07D207/06 , C07D207/14 , C07D207/16 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/12 , C07D405/12 , C07D409/12 , C07D417/12 , C07D417/14
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