公开(公告)号：DK1135387T3

公开(公告)日：2002-11-25

申请号：DK99961051

申请日：1999-12-02

Applicant: BASF AG

Inventor： NEIDLEIN ULF ,  GOETZ NORBERT ,  MISSLITZ ULF ,  GOETZ ROLAND ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  KUDIS STEFFEN ,  LANGEMANN KLAUS ,  MAYER GUIDO ,  WITSCHEL MATTHIAS ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: A01N43/50 ,  A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  C07B61/00 ,  C07D231/20 ,  C07D413/10 ,  C07D413/12 ,  C07D413/00

Abstract: 3-(Heterocyclyl)benzoylpyrazole derivatives of the formula Iwhere:X is O, NH or N-alkyl;R1 is nitro, halogen, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfonyl or haloalkylsulfonyl;R2,R3,R4,R5 are hydrogen, alkyl or haloalkyl;R6 is halogen, nitro, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfonyl or haloalkylsulfonyl;R7 is hydroxyl, alkoxy, alkenyloxy, alkylsulfonyloxy, alkylcarbonyloxy, (alkylthio)carbonyloxy, phenylsulfonyloxy or phenylcarbonyloxy, where the phenyl radical may be substituted;R8,R9 are alkyl;R10 is hydrogen or alkyl;R11 is hydrogen or alkyl;and their agriculturally useful salts,compounds for their preparation, and the use of these compounds or of compositions comprising them for controlling undesirable plants are described.

公开(公告)号：HU221475B

公开(公告)日：2002-10-28

申请号：HU9503040

申请日：1994-04-13

Applicant: BASF AG

Inventor： BAUMANN ERNST ,  BRATZ MATTHIAS ,  GERBER MATTHIAS ,  RADEMACHER WILHELM ,  RHEINHEIMER JOACHIM ,  THEOBALD HANS ,  VOGELBACHER UWE JOSEF ,  WALTER HELMUT ,  WESTPHALEN KARL-OTTO

IPC: A01N43/54 ,  C07D251/22 ,  A01N43/64 ,  A01N43/66 ,  A01N43/72 ,  A01P13/00 ,  A01P21/00 ,  C07C45/58 ,  C07C47/198 ,  C07C47/277 ,  C07C59/125 ,  C07C67/31 ,  C07C69/708 ,  C07C69/734 ,  C07C205/28 ,  C07C323/22 ,  C07C323/50 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/38 ,  C07D239/60 ,  C07D251/24 ,  C07D251/30 ,  C07D251/34 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D411/12 ,  C07D413/12 ,  C07D477/12 ,  C07D491/048

Abstract: PCT No. PCT/EP94/01141 Sec. 371 Date Oct. 19, 1995 Sec. 102(e) Date Oct. 19, 1995 PCT Filed Apr. 13, 1994 PCT Pub. No. WO94/25442 PCT Pub. Date Nov. 10, 19943-(Het)arylcarboxylic acid derivatives of the formula I I where R is formyl, CO2H or a radical hydrolyzable to COOH and the other substituents have the following meanings: R2 and R3 are each halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; X is nitrogen or CR14, where R14 is hydrogen or, together with R3, forms an alkylene or alkenylene chain, in each of which a methylene group is replaced by oxygen; R4 is phenyl or naphthyl, each of which is unsubstituted or substituted or an unsubstituted or substituted five-membered or six-membered heteroaromatic structure containing one to three nitrogen atoms or one sulfur or oxygen atom; R5 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl or phenyl; R6 is C1-C8-alkyl, C3-C6-alkenyl, C3-C6-alkynyl or C3-C4-cyclo-alkyl, each of which may be mono- or polysubstituted; Y is sulfur, oxygen or a single bond; and Z is sulfur or oxygen; with the proviso that R6 is not unsubstituted C1-C4-alkyl when R4 is unsubstituted phenyl, Z is oxygen and simultaneously R5 is methyl or hydrogen.

公开(公告)号：SK8682001A3

公开(公告)日：2002-08-06

申请号：SK8682001

申请日：1999-12-09

Applicant: BASF AG

Inventor： AMBERG WILHELM ,  JANSEN ROLF ,  KETTSCHAU GEORG ,  RIECHERS HARTMUT ,  BAUMANN ERNST ,  HERGENRODER STEFAN ,  RASCHACK MANFRED ,  UNGER LILIANE

IPC: C07D251/24 ,  A61K31/505 ,  A61K31/506 ,  A61K31/53 ,  A61P9/04 ,  A61P9/10 ,  A61P9/12 ,  A61P13/08 ,  A61P13/12 ,  A61P15/10 ,  A61P35/00 ,  A61P43/00 ,  C07C229/34 ,  C07C233/87 ,  C07C235/52 ,  C07D239/34 ,  C07D251/22 ,  C07D401/12 ,  C07D491/048 ,  C07D239/60

Abstract: The invention relates to carboxylic acid derivatives of formula (I), in which the substituents have the following meanings: R is tetrazol or a group (a); W and Z, can be identical or different and are nitrogen or methine, provided that if W and Z are methine, then Q is nitrogen; X is nitrogen or CR ; Y is nitrogen or CR ; Q is nitrogen or CR , provided that if Q is nitrogen then X is CR and Y is CR ; R and R are identical or different and are possibly substituted phenyl or naphthyl or phenyl or naphthyl which are linked in an ortho position via a direct bond, a methlyene, ethylene or ethenylene group, an oxygen or sulfur atom or a SO2-, NH- or N-alkyl group or possibly substituted C5-C6-cycloalkyl; R is a rest (b) or (c); and R is hydrogen, C1-C4-alkyl. The invention further relates to their preparation and their use as endothelin receptor antagonists. The invention also relates to compounds of formula (II) and a structural fragment of formula (d) in which the rests R , R , R , R and R have the meanings given in claim no. 1 and to their use as structural elements in an endothelin receptor antagonist.

公开(公告)号：CA2431267A1

公开(公告)日：2002-06-20

申请号：CA2431267

申请日：2001-12-10

Applicant: BASF AG

Inventor： MAYER GUIDO ,  VOLK THORSTEN ,  ZAGAR CYRILL ,  WITSCHEL MATTHIAS ,  MISSLITZ ULF ,  BAUMANN ERNST ,  LANDES ANDREAS ,  VON DEYN WOLFGANG ,  KUDIS STEFFEN ,  LANGEMANN KLAUS ,  HOFMANN MICHAEL

IPC: A01N43/74 ,  A01N43/76 ,  A01N43/78 ,  C07D263/58 ,  C07D277/68 ,  C07D417/06 ,  C07D521/00

Abstract: The invention relates to cyclohexenone derivatives of benzazolons of general formula (I), wherein the variables R1, R2, R3, A and Hex have the meaning as cited in claim 1, and the salts thereof, and the use thereof for controlling harmful plants.

公开(公告)号：BR0012280A

公开(公告)日：2002-06-04

申请号：BR0012280

申请日：2000-06-23

Applicant: BASF AG

Inventor： NEIDLEIN ULF ,  GOETZ NORBERT ,  BAUMANN ERNST ,  DEYN WOLFGANG VON ,  KUDIS STEFFEN ,  GOETZ ROLAND ,  LANGEMANN KLAUS ,  MAYER GUIDO ,  MISSLITZ ULF ,  WITSCHEL MATTHIAS ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: A01N43/56 ,  C07D231/20 ,  C07D231/00

Abstract: Cycloalkyl-substituted benzoylpyrazoles of the formula Iwhere the variables have, for example, the following meanings:R1 is hydrogen, nitro, halogen, cyano, thiocyanato, or an unsubstituted or substituted aliphatic radical;R2 is an unsubstituted or substituted aliphatic radical, halogen, nitro, or substituted sulfonyl or amino groups,R3 is hydrogen, halogen, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C2-C6-alkenyl or C2-C6-alkynyl;R4, R5 are hydrogen, nitro, halogen, cyano, thiocyanato, an unsubstituted or substituted aliphatic radical or substituted sulfonyl or amino groups;R6 is hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C3-C8-cycloalkyl;R7 is a cyclic ring system having 3-14 ring atoms;R16 is hydroxyl or a substituted hydroxyl group;and their tautomers or agriculturally useful salts are described.Moreover, the invention describes processes for preparing compounds of the formula I, compositions comprising them, and the use of the compounds of the formula I and of the compositions comprising them for controlling harmful plants.

公开(公告)号：DE59410073D1

公开(公告)日：2002-04-11

申请号：DE59410073

申请日：1994-04-14

Applicant: BASF AG

Inventor： BAUMANN ERNST ,  RHEINHEIMER JOACHIM ,  VOGELBACHER JOSEF ,  BRATZ MATTHIAS ,  MEYER NORBERT ,  GERBER MATTHIAS ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT ,  RADEMACHER WILHELM

IPC: C07D251/34 ,  A01N43/54 ,  A01N43/60 ,  A01N43/66 ,  A01P13/00 ,  C07C69/22 ,  C07C69/712 ,  C07C69/734 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/38 ,  C07D239/52 ,  C07D239/60 ,  C07D251/30 ,  C07D307/46 ,  C07D307/54 ,  C07D333/24 ,  C07D405/12 ,  C07D409/12 ,  C07D491/048

Abstract: PCT No. PCT/EP94/01156 Sec. 371 Date Oct. 19, 1995 Sec. 102(e) Date Oct. 19, 1995 PCT Filed Apr. 14, 1994 PCT Pub. No. WO94/25443 PCT Pub. Date Nov. 10, 19943-(Het)aryloxy(thio)carboxylic acid derivatives of the formula I I where R1 is hydrogen, COOH or a radical which can be hydrolyzed to give COOH; R2 and R3 are each halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; X is nitrogen or CR14, where R14 is hydrogen or, together with R3, forms a 3-membered or 4-membered alkylene or alkenylene chain, in each of which a methylene group is replaced by oxygen; R4 is alkyl, cycloalkyl, cycloalkenyl, alkenyl or alkynyl, each of which is unsubstituted or substituted; an unsubstituted or substituted five-membered or six-membered heteroaromatic structure containing one to three nitrogen atoms or one sulfur or oxygen atom; unsubstituted or substituted phenyl or naphthyl; R4 and R5, together with the neighboring carbon atom, form a 3-membered to 8-membered ring which may contain an oxygen or sulfur atom and which is unsubstituted or substituted; R5 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl or phenyl, each of which is unsubstituted or substituted; R6 is unsubstituted or substituted phenyl or naphthyl or an unsubstituted or substituted five-membered or six-membered heteroaromatic structure containing one to three nitrogen atoms or one sulfur or oxygen atom; Y is sulfur or oxygen or a single bond; and Z is sulfur or oxygen.

公开(公告)号：BR0012285A

公开(公告)日：2002-03-26

申请号：BR0012285

申请日：2000-06-23

Applicant: BASF AG

Inventor： NEIDLEIN ULF ,  GOETZE NORBERT ,  BAUMANN ERNST ,  DEYN WOLFGANG VON ,  KUDIS STEFFEN ,  GOETZ ROLAND ,  LANGEMANN KLAUS ,  MAYER GUIDO ,  MISSLITZ ULF ,  WITSCHEL MATTHIAS ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: C07D231/20 ,  A01N43/48 ,  A01N43/56 ,  C07D231/24 ,  C07D231/00

Abstract: Pyrazoles of the formula Iwhere:R1 is hydrogen, nitro, halogen, cyano, thiocyanato or an aliphatic radical;R2 is a substituted sulfur, nitrogen or phosphorus atom;R3 is hydrogen, halogen or an aliphatic radical;R4, R5 are hydrogen, nitro, halogen, cyano, thiocyanato, or an aliphatic radical;R6 is hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C3-C8-cycloalkyl;R7, R8, R9 are hydrogen, C1-C6-alkyl, but at most one of the radicals R7, R8 and R9 is hydrogen;and their tautomers and agriculturally useful salts are described.Moreover, the invention relates to processes for preparing compounds of the formula I, to compositions comprising them and to the use of the compounds of the formula I and of the compositions comprising them for controlling harmful plants.

公开(公告)号：GR3036931T3

公开(公告)日：2002-01-31

申请号：GR20010401798

申请日：2001-10-18

Applicant: BASF AG

Inventor： RIECHERS HARTMUT ,  KLINGE DAGMAR ,  AMBERG WILHELM ,  KLING ANDREAS ,  MUELLER STEFAN ,  BAUMANN ERNST ,  RHEINHEIMER JOACHIM ,  VOGELBACHER UWE JOSEF ,  WERNET WOLFGANG ,  UNGER LILIANE ,  RASCHACK MANFRED

IPC: C07D251/30 ,  A61K31/505 ,  A61P9/00 ,  A61P9/08 ,  A61P9/10 ,  A61P9/12 ,  A61P11/08 ,  A61P13/02 ,  A61P15/00 ,  A61P25/04 ,  C07D239/00 ,  C07D239/26 ,  C07D239/28 ,  C07D239/34 ,  C07D239/38 ,  C07D239/60 ,  C07D239/70 ,  C07D239/96 ,  C07D251/12 ,  C07D251/52 ,  C07D257/02 ,  C07D309/00 ,  C07D403/06 ,  C07D403/12 ,  C07D405/12 ,  C07D417/12 ,  C07D487/04 ,  C07D491/04 ,  C07D491/044 ,  C07D491/048

Abstract: Heterocyclyl-substd. propanoic acids and their derivs., of formula (I), are new. R = formyl, tetrazolyl, nitrile, COOH or a gp. that can be hydrolysed to COOH; X = N or CR14; R2 = H, OH, NH2, alkylamino, dialkylamino, halo, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; R14 = H or 1-5 C alkyl; R3 = R2 or alkoxyimino; or CR3 + CR14 = 5 or 6 membered alkylene or alkenyl ring (opt. substd. by 1-2 alkyl) in which a methylene can be replaced by O, S, NH or alkylamino; R4, R5 = phenyl or naphthyl (both opt. substd. by one or more halo, NO2, CN, OH, alkyl, haloalkyl, alkoxy, haloalkyloxy, phenoxy, alkylthio, NH2, alkylamine or dialkylamino) or 3-7 C cycloalkyl; or the phenyl or naphthyl gps. are opt. bonded at the O- position (by a bond, CH2, O, S, SO2, ethylene, ethenylene or opt. alkylated amino); R6 = H, 1-8 C alkyl, 2-6 C alkenyl, 3-6 C alkynyl, 3-8 C cycloalkyl (all opt. substd. by 1 or more halo, NO2, CN, alkoxy 3-6 C alkenyloxy, 3-6 C alkynyloxy, alkylthio, haloalkoxy, alkylcarbonyl, alkoxycarbonyl, 3-8 C alkylcarbonylalkyl, alkylamino, dialkylamino, phenyl, Ph or OPh), Ar or Het; Y = S, O or bond; Q = S, O, SO, SO2 or bond; Ph = substd. phenyl, where substits. are halo, NO2, CN, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; Ar = phenyl or naphthyl (both opt. substd. by 1 or more halo, NO2, CN, OH, NH2, alkylamino, dialkylamino or OCH2CH2O); Het = 5 or 6 membered heteroaromatic with 1-3 N atoms and/or one S or O (opt. substd. by 1-4 halo and/or 1 or 2 alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, phenyl, phenoxy or phenyl carbonyl (where the phenyl is opt. substd. by 1-5 halo and/or 1-3 alkyl, haloalkyl, alkoxy, haloalkoxy and/or alkylthio)); alkyl and alkoxy have 1-4 C unless otherwise stated; provided that R6 is not H when Q = bond.

公开(公告)号：ES2162942T3

公开(公告)日：2002-01-16

申请号：ES95935916

申请日：1995-10-07

Applicant: BASF AG

Inventor： RIECHERS HARTMUT ,  KLINGE DAGMAR ,  AMBERG WILHELM ,  KLING ANDREAS ,  MULLER STEFAN ,  BAUMANN ERNST

IPC: C07D251/30 ,  A61K31/505 ,  A61P9/00 ,  A61P9/08 ,  A61P9/10 ,  A61P9/12 ,  A61P11/08 ,  A61P13/02 ,  A61P15/00 ,  A61P25/04 ,  C07D239/00 ,  C07D239/26 ,  C07D239/28 ,  C07D239/34 ,  C07D239/38 ,  C07D239/60 ,  C07D239/70 ,  C07D239/96 ,  C07D251/12 ,  C07D251/52 ,  C07D257/02 ,  C07D309/00 ,  C07D403/06 ,  C07D403/12 ,  C07D405/12 ,  C07D417/12 ,  C07D487/04 ,  C07D491/04 ,  C07D491/044 ,  C07D491/048

Abstract: Heterocyclyl-substd. propanoic acids and their derivs., of formula (I), are new. R = formyl, tetrazolyl, nitrile, COOH or a gp. that can be hydrolysed to COOH; X = N or CR14; R2 = H, OH, NH2, alkylamino, dialkylamino, halo, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; R14 = H or 1-5 C alkyl; R3 = R2 or alkoxyimino; or CR3 + CR14 = 5 or 6 membered alkylene or alkenyl ring (opt. substd. by 1-2 alkyl) in which a methylene can be replaced by O, S, NH or alkylamino; R4, R5 = phenyl or naphthyl (both opt. substd. by one or more halo, NO2, CN, OH, alkyl, haloalkyl, alkoxy, haloalkyloxy, phenoxy, alkylthio, NH2, alkylamine or dialkylamino) or 3-7 C cycloalkyl; or the phenyl or naphthyl gps. are opt. bonded at the O- position (by a bond, CH2, O, S, SO2, ethylene, ethenylene or opt. alkylated amino); R6 = H, 1-8 C alkyl, 2-6 C alkenyl, 3-6 C alkynyl, 3-8 C cycloalkyl (all opt. substd. by 1 or more halo, NO2, CN, alkoxy 3-6 C alkenyloxy, 3-6 C alkynyloxy, alkylthio, haloalkoxy, alkylcarbonyl, alkoxycarbonyl, 3-8 C alkylcarbonylalkyl, alkylamino, dialkylamino, phenyl, Ph or OPh), Ar or Het; Y = S, O or bond; Q = S, O, SO, SO2 or bond; Ph = substd. phenyl, where substits. are halo, NO2, CN, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; Ar = phenyl or naphthyl (both opt. substd. by 1 or more halo, NO2, CN, OH, NH2, alkylamino, dialkylamino or OCH2CH2O); Het = 5 or 6 membered heteroaromatic with 1-3 N atoms and/or one S or O (opt. substd. by 1-4 halo and/or 1 or 2 alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, phenyl, phenoxy or phenyl carbonyl (where the phenyl is opt. substd. by 1-5 halo and/or 1-3 alkyl, haloalkyl, alkoxy, haloalkoxy and/or alkylthio)); alkyl and alkoxy have 1-4 C unless otherwise stated; provided that R6 is not H when Q = bond.

公开(公告)号：AU9139501A

公开(公告)日：2002-01-10

申请号：AU9139501

申请日：2001-11-16

Applicant: BASF AG

Inventor： DEYN WOLFGANG VON ,  HILL REGINA LUISE ,  KARDORFF UWE ,  BAUMANN ERNST ,  ENGEL STEFAN ,  MAYER GUIDO ,  WITSCHEL MATTHIAS ,  RACK MICHAEL ,  GOTZ NORBERT ,  GEBHARDT JOACHIM ,  MISSLITZ ULF ,  WALTER HELMUT ,  WESTPHALEN KARL-OTTO ,  OTTEN MARTINA ,  RHEINHEIMER JOACHIM

IPC: C07D277/10 ,  A01N43/72 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  C07D231/20 ,  C07D237/00 ,  C07D261/00 ,  C07D261/04 ,  C07D261/20 ,  C07D263/10 ,  C07D273/00 ,  C07D277/20 ,  C07D277/34 ,  C07D291/04 ,  C07D311/00 ,  C07D403/10 ,  C07D413/10 ,  C07D417/10 ,  C07D419/10 ,  C07D498/10

Abstract: Benzoyl derivatives of the formula I where the variables have the following meanings: R1, R2 are hydrogen, nitro, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl or C1-C6-haloalkylsulfonyl; R3 is hydrogen, halogen or alkyl; R4, R5 are hydrogen, halogen, cyano, nitro, alkyl, alkoxy, alkylthio, dialkylamino, phenyl or carbonyl, it being possible for the 6 last-mentioned radicals to be substituted; X is O, S, NR9, CO or CR10R11; Y is O, S, NR12, CO or CR13R14; R15 is pyrazole which is unsubstituted or substituted, linked in the 4-position and has attached to it in the 5-position a hydroxyl or sulfonyloxy radical; and the agriculturally useful salts thereof; processes and intermediates for the preparation of the 3-heterocyclyl-substituted benzoyl derivatives; compositions comprising them; and the use of these derivatives or compositions comprising them for controlling undesirable plants.