公开(公告)号：CA2557781C

公开(公告)日：2012-01-10

申请号：CA2557781

申请日：2005-03-08

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90 ,  C07D239/00 ,  C07D249/00

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl or alkoxyalkyl, whereby the aliphatic groups can be substituted according to the description; R2 represents CHR3CH3, cyclopropyl, CH=CH2 or CH2CH=CH2 and R3 represents hydrogen, CH3 or CH2CH3. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

公开(公告)号：CA2467683C

公开(公告)日：2011-09-27

申请号：CA2467683

申请日：2002-11-15

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  SCHWOEGLER ANJA ,  RHEINHEIMER JOACHIM ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  ROSE INGO ,  SCHAEFER PETER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: C07D239/46 ,  A01N43/54 ,  C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D401/06 ,  C07D401/14 ,  C07D403/12

Abstract: 5-Phenylpyrimidines of formula (I), where the substituents and the indices have the following meanings: R1, R2 = H, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkinyl or haloalkinyl, where R1 and R2 together with the nitrogen atom to which they are bonded may form a saturated or unsaturated ring, interrupted by an ether, thio, sulphoxy or sulphonyl group and which can be substituted by one to four groups Ra and/or Rb, R3 = H, halo, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy, R4 = H, halo, cyano, hydroxy, mercapto, azido, alkyl, alkenyl, alkinyl, haloalkyl, alkoxy, alkenyloxy, alkinyloxy, haloalkoxy, alkylthio, alkenylthio, alkinylthio, haloalkylthio, -ON=CRaRb, -CRc=NORa, -NRcN=CRaRb, -NRaRb, -NRcNRaRb, -NORa, -NRcC (=NRc') NRaRb, -NRcC (=0) NRaRb, -NRaC (=0) Rc, -NRaC (=NORc)Rc', -OC (=0) Rc, -C (=NORc) NRaRb, -CRc (=NNRaRb), -C (=0) NRaRb or -C (=0) Rc, where Ra,Rb,Rc are as defined in the description, X = halo, alkyl, alkoxy or haloalkyl and m = a whole number from 1 to 5. The invention further relates to methods for production of the above compounds, agents containing the same and use thereof for the treatment of noxious mycoses.

公开(公告)号：CU23683B7

公开(公告)日：2011-07-11

申请号：CU20060172

申请日：2006-09-06

Applicant: BASF AG

Inventor： STIERL REINHARD ,  SCOEFL ULRICH ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  NIEDENBRUECK MATTHIAS ,  WAGNER OLIVER ,  SCHWOEGLER ANJA ,  SCHIEWECK FRANK ,  RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  GEWEHR MARKUS ,  MUELLER BERND ,  BLETTNER CARSTEN ,  JORDI TORMO I BLASCO

IPC: A01N43/90 ,  C07D249/00 ,  C07D487/04

Abstract: 5,6-Dialquil-7-amino-triazolopirimidinas de la fórmula I ESPACIO PARA FÓRMULA en la que los sustituyentes tienen los significados siguientes: R1 significa alquilo C5-C12 o alcoxialquilo C5-C14, pudiendo los grupos alifáticos estar sustituidos por uno o tres de los grupos siguientes: ciano, nitro, hidroxi, cicloalquilo C3-C6, alquiltio C1-C6 y NRaRb; Ra, Rb significan hidrógeno o alquilo C1-C6; R2 significa CHR3CH3, ciclopropilo, CH=CH2 o CH2CH=CH2; R3 es hidrógeno o CH3, CH2CH3; procedimiento para la preparación de estos compuestos, productos que los contienen, así como el uso de los mismos para combatir hongos nocivos fitopatógenos.

公开(公告)号：NZ560916A

公开(公告)日：2010-12-24

申请号：NZ56091606

申请日：2006-03-15

Applicant: BASF AG

Inventor： GRAMMENOS WASSILIOS ,  RHEINHEIMER JOACHIM ,  LOHMANN JAN KLAAS ,  GROTE THOMAS ,  PUHL MICHAEL ,  KORADIN CHRISTOPHER ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  LANGEWALD JURGEN ,  GOTZ NORBERT ,  CULBERTSON DEBORAH L ,  ANSPAUGH DOUGLAS D ,  OLOUMI-SADEGHI HASSAN ,  COTTER HENRY VAN TUYL ,  KUHN DAVID G

IPC: A01N43/40 ,  C07D213/42

Abstract: Disclosed are biphenylsulfonamides of formula I wherein the substituents are disclosed within the specification. Also disclosed are processes for preparing the compounds of formula I. Also disclosed is the use of the compound of formula I for the treatment of phytopathogenic harmful fungi and for combating harmful anthropodes.

公开(公告)号：SK287476B6

公开(公告)日：2010-11-08

申请号：SK16872000

申请日：1999-05-04

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  VON DEYN WOLFGANG ,  GEBHARDT JOACHIM ,  RACK MICHAEL ,  LOCHTMAN RENE ,  GOTZ NORBERT ,  KEIL MICHAEL ,  WITSCHEL MATTHIAS ,  HAGEN HELMUT ,  MISSLITZ ULF ,  BAUMANN ERNST

IPC: C07C205/00 ,  C07C20060101 ,  C07C201/00 ,  C07C201/12 ,  C07C205/44 ,  C07C249/00 ,  C07C249/06 ,  C07C251/48 ,  C07C251/52 ,  C07C253/00 ,  C07C255/50 ,  C07C317/00 ,  C07C317/32 ,  C07C319/00 ,  C07C319/14 ,  C07C323/09 ,  C07D20060101 ,  C07D261/02 ,  C07D261/04 ,  C07D261/08 ,  C07D413/00 ,  C07D413/02 ,  C07D413/10

Abstract: A method for producing isoxazolene of the formula (I), where R1 is hydrogen, C1-C6 alkyl, R2 is C1-C6 alkyl, R3, R4, R5 are hydrogen, C1-C6 alkyl or R4 and R5 together form a bond, R6 is a heterocyclic ring, and n is 0, 1 or 2. Said method comprises the production of an intermediate compound of the formula (VI), where R1, R3, R4 and R5 have the meanings given above. This step is followed by halogenation, thiomethylation, oxidation and acylation to yield compounds of formula (I). The invention also relates to new intermediate products for producing compounds of formula (I).

公开(公告)号：CU20060172A7

公开(公告)日：2010-10-30

申请号：CU20060172

申请日：2006-09-06

Applicant: BASF AG

Inventor： STIERL REINHARD ,  SCOEFL ULRICH ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  NIEDENBRUECK MATTHIAS ,  WAGNER OLIVER ,  SCHWOEGLER ANJA ,  SCHIEWECK FRANK ,  RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  GEWEHR MARKUS ,  MUELLER BERND ,  BLETTNER CARSTEN ,  JORDI TORMO I BLASCO

IPC: A01N43/90 ,  C07D249/00 ,  C07D487/04

Abstract: 5,6-Dialquil-7-amino-triazolopirimidinas de la fórmula I ESPACIO PARA FÓRMULA en la que los sustituyentes tienen los significados siguientes: R1 significa alquilo C5-C12 o alcoxialquilo C5-C14, pudiendo los grupos alifáticos estar sustituidos por uno o tres de los grupos siguientes: ciano, nitro, hidroxi, cicloalquilo C3-C6, alquiltio C1-C6 y NRaRb; Ra, Rb significan hidrógeno o alquilo C1-C6; R2 significa CHR3CH3, ciclopropilo, CH=CH2 o CH2CH=CH2; R3 es hidrógeno o CH3, CH2CH3; procedimiento para la preparación de estos compuestos, productos que los contienen, así como el uso de los mismos para combatir hongos nocivos fitopatógenos.

公开(公告)号：EA014240B1

公开(公告)日：2010-10-29

申请号：EA200702350

申请日：2006-05-16

Applicant: BASF AG

Inventor： DIETZ JOCHEN ,  GEWEHR MARCUS ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  HUNGER UDO ,  MULLER BERND ,  SCHIEWECK ANJA ,  SCHWOGLER ANJA ,  LOHMANN JAN KLAUS ,  RHEINHEIMER JOACHIM ,  RENNER JENS ,  SCHAFER PETER

IPC: C07D277/20 ,  A01N43/78

Abstract: Анилидытиазолкарбоновойкислотыформулы Iвкоторойпеременныеимеютследующеезначение:X - галоген; R- C-Салкилили C-Сгалогеналкил; R- метил; W - кислород; способполученияэтихсоединений, содержащееихсредствои посевнойматериал, атакжеспособборьбыс патогеннымигрибами.

公开(公告)号：UA91537C2

公开(公告)日：2010-08-10

申请号：UAA200710262

申请日：2006-02-15

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  DIETZ JOCHEN ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GRAMMENOS WASSILIOS ,  HUENGER UDO ,  MUELLER BERND ,  SCHWOEGLER ANJA ,  LOHMANN JAN KLAAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  STRATHMANN SIEGFRIED ,  STIERL REINHARD

IPC: C07D231/14 ,  A01C1/06 ,  A01N43/56 ,  A01P3/00 ,  C07C211/46

公开(公告)号：NZ552589A

公开(公告)日：2010-07-30

申请号：NZ55258905

申请日：2005-07-22

Applicant: BASF AG

Inventor： GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  HUNGER UDO ,  MULLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  SCHOFL ULRICH ,  KOHLE HARALD ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  STIERL REINHARD ,  RETHER JAN

IPC: A01N43/54 ,  C07D401/04

Abstract: Disclosed are compounds of formula (I), wherein k is 1-3, R3 is C1-C4 alkyl, n is 1-5 and the remaining substituents are as defined in the specification, and agriculturally acceptable salts thereof. The compounds are useful for controlling phytopathogenic fungi and as plant protection products.

公开(公告)号：BRPI0607108A2

公开(公告)日：2010-03-09

申请号：BRPI0607108

申请日：2006-01-30

Applicant: BASF AG

Inventor： SCHIEWECK FRANK ,  GROTE THOMAS ,  NAVE BARBARA ,  SCHWIGLER ANJA ,  JABS THORSTEN ,  BLETTNER CARSTEN ,  RHEINHEIMER JOACHIM ,  MUELLER BERND

IPC: A61K31/506 ,  A61K31/505 ,  C07D239/42 ,  C07D239/48 ,  C07D401/04 ,  C07D403/04 ,  C07D417/04

Abstract: The present invention relates to substituted 5-phenyl pyrimidines I, which carry a radical X in the 4-position of the pyrimidine ring, a radical Y in the 6-position of the pyrimidine ring, the radical X denoting a group of the formula NR 1 R 2 , OR 1a or SR 1a , in which R 1 , R 2 , independently of each other, denote hydrogen, C 1 -C 10 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 1 -C 10 -haloalkyl, C 3 -C 8 -cycloalkyl, C 3 -C 8 -halocycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which radicals may be unsubstituted or may carry 1, 2, 3 or 4 radicals R a1 ; or the radical NR 1 R 2 may also form a 5- or 6-membered optionally substituted heterocyclic ring, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which are non-adjacent to the nitrogen of NR 1 R 2 , in which two adjacent C atoms or one N atom and one adjacent C atom can be linked by a C 1 -C 4 -alkylene chain and wherein the heterocyclic ring may be unsubstituted or may carry 1, 2, 3 or 4 radicals R a1 as defined in claim 1 , R 1a has one of the meanings given for R 1 except for hydrogen; the radical Y being selected from the group consisting of halogen, cyano, C 1 -C 4 -alkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 4 -alkoxy, C 3 -C 4 -alkenyloxy, C 3 -C 4 -alkynyloxy, C 1 -C 6 -alkylthio, di-(C 1 -C 6 -alkyl)amino or C 1 -C 6 -alkylamino, where the alkyl, alkenyl and alkynyl radicals of Y may be substituted by halogen, cyano, nitro, C 1 -C 2 -alkoxy or C 1 -C 4 -alkoxycarbonyl; and wherein the pyrimidine radical may also carry a radical different from hydrogen in the 2-position and wherein the phenyl ring in the 5-position of the pyrimidine ring may be unsubstituted or carry 1, 2, 3, 4 or 5 radicals L which are different from hydrogen, and the pharmaceutically acceptable salts substituted 5-phenyl pyrimidines for use in therapy, in particular in therapy or treatment of cancerous diseases.