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81.
公开(公告)号:MX2012006391A
公开(公告)日:2012-06-19
申请号:MX2012006391
申请日:2010-06-01
Applicant: ABBOTT LAB
Inventor: WANG GARY T , HEXAMER LAURA , SULLIVAN GERARD M , WANG LE , TAO ZHI-FU , BRUNCKO MILAN , WENDT MICHAEL D , DAI YUJIA , DING HONG , ELMORE STEVEN W , MCCELLAN WILLIAM J , HANSEN TODD M , SOUERS ANDREW J , SONG XIAOHONG , PARK CHEOL-MIN , MANTEI ROBERT A , DOHERTY GEORGE A , HASVOLD LISA , PARK CHANG H , PETROS ANDREW M , KUNZER AARON
IPC: C07D209/08 , C07D211/58 , C07D213/74 , C07D213/84 , C07D231/56 , C07D235/06 , C07D277/24 , C07D309/04 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D413/12 , C07D417/12 , C07D471/04
Abstract: Se describen los compuestos que inhiben la actividad de las proteínas anti-apoptóticas BcI-2, las composiciones que contienen los compuestos, y los métodos para tratar las enfermedades durante las cuales se expresa la proteína anti-apoptótica Bcl-2.
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82.
公开(公告)号:ECSP11011554A
公开(公告)日:2012-01-31
申请号:ECSP11011554
申请日:2011-12-26
Applicant: ABBOTT LAB
Inventor: DOHERTY GEORGE ANDREW , HASVOLD LISA A , SULLIVAN GERARD M , WANG XILU , MANTEI ROBERT A , ELMORE STEVEN W , SOUERS ANDREW J , BRUNCKO MILAN , SONG XIAOHONG , WANG LE , KUNZER AARON R , WENDT MICHAEL D , TAO ZHI-FU , DING HONG , HEXAMER LAURA , HANSEN TODD M
IPC: C07D471/04 , A61K31/437 , A61P35/00
Abstract: Compuestos que inhiben la actividad de proteínas anti-apoptóticas Bcl-2, composiciones que contienen a dichos compuestos y métodos de tratamiento de enfermedades durante cuyo transcurso hay expresión de la proteína anti-apoptótica Bcl-2.
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83.
公开(公告)号:MX2011012257A
公开(公告)日:2011-12-16
申请号:MX2011012257
申请日:2010-05-26
Applicant: ABBOTT LAB
Inventor: SOUERS ANDREW J , BRUNCKO MILAN , DING HONG , DOHERTY GEORGE , ELMORE STEVEN , HASVOLD LISA , HEXAMER LAURA , KUNZER AARON R , SONG XIAOHONG , SULLIVAN GERARD , TAO ZHI-FU , WANG GARY T , WANG LE , WENDT MICHAEL , WANG XILU , MANTEI ROBERT , HANSEN TODD M
IPC: C07D471/04 , A61K31/437 , A61P35/00
Abstract: Compuestos que inhiben la actividad de proteínas anti-apoptóticas Bcl-2, composiciones que contienen a dichos compuestos y métodos de tratamiento de enfermedades durante cuyo transcurso hay expresión de la proteína anti-apoptótica Bcl-2.
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84.
公开(公告)号:SG175253A1
公开(公告)日:2011-11-28
申请号:SG2011075843
申请日:2010-05-26
Applicant: ABBOTT LAB
Inventor: BRUNCKO MILAN , DING HONG , DOHERTY GEORGE , ELMORE STEVEN , HASVOLD LISA , HEXAMER LAURA , KUNZER AARON R , SONG XIAOHONG , SOUERS ANDREW J , SULLIVAN GERARD , TAO ZHI-FU , WANG GARY T , WANG LE , WANG XILU , WENDT MICHAEL , MANTEI ROBERT , HANSEN TODD M
Abstract: Disclosed are compounds which inhibit the activity of anti-apoptotic Bcl-2 proteins, compositions containing the compounds and methods of treating diseases during which is expressed anti-apoptotic Bcl-2 protein.
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85.
公开(公告)号:ECSP11011173A
公开(公告)日:2011-08-31
申请号:ECSP11011173
申请日:2011-07-04
Applicant: ABBOTT LAB
Inventor: DOHERTY GEORGE ANDREW , HASVOLD LISA A , SULLIVAN GERARD M , WANG GARY , WANG XILU , MANTEI ROBERT A , ELMORE STEVEN W , SOUERS ANDREW J , BRUNCKO MILAN , SONG XIAOHONG , WANG LE , KUNZER AARON R , PARK CHEOL-MIN , WENDT MICHAEL D , TAO ZHI-FU , DAI YUJIA , DING HONG , HEXAMER LAURA , MCCLELLAN WILLIAM J , PARK CHANG H , PETROS ANDREW M
IPC: A61P35/00 , A61K31/496 , C07D403/12
Abstract: Compuestos que inhiben la actividad de proteínas anti-apoptóticas Bcl-2, composiciones que contienen a dichos compuestos y métodos de tratamiento de enfermedades durante cuyo transcurso hay expresión de la proteína anti-apoptótica Bcl-2.
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86.
公开(公告)号:CA2759182A1
公开(公告)日:2010-12-02
申请号:CA2759182
申请日:2010-05-26
Applicant: ABBOTT LAB
Inventor: BRUNCKO MILAN , DING HONG , DOHERTY GEORGE , ELMORE STEVEN , HASVOLD LISA , HEXAMER LAURA , KUNZER AARON R , SONG XIAOHONG , SOUERS ANDREW J , SULLIVAN GERARD , TAO ZHI-FU , WANG GARY T , WANG LE , WANG XILU , WENDT MICHAEL , MANTEI ROBERT , HANSEN TODD M
IPC: C07D471/04 , A61K31/437 , A61P35/00
Abstract: Disclosed are compounds which inhibit the activity of anti-apoptotic Bcl-2 proteins, compositions containing the compounds and methods of treating diseases during which is expressed anti-apoptotic Bcl-2 protein.
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公开(公告)号:DE60118955T2
公开(公告)日:2007-01-04
申请号:DE60118955
申请日:2001-11-30
Applicant: ABBOTT LAB
Inventor: CLAIBORNE K , GWALTNEY L , HASVOLD A , LI QUN , LI TOMGMEI , LIN NAN-HORNG , MANTEI A , ROCKWAY W , SHAM L , SULLIVAN M , TONG YUNSONG , WANG T , WANG LE , WANG XILU , WANG WEIBO
IPC: C07D233/64 , A61K31/4164 , A61K31/4178 , A61K31/426 , A61K31/4439 , A61K31/4709 , A61P35/00 , A61P43/00 , C07D233/54 , C07D277/20 , C07D277/30 , C07D401/12 , C07D405/12 , C07D409/12
Abstract: Substituted imidazoles and thiazoles having the formula are useful for inhibiting farnesyltransferase. Also disclosed are farnesyltransferase-inhibiting compositions and methods of inhibiting farnesyltransferase in a patient.
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公开(公告)号:PT1339695E
公开(公告)日:2006-08-31
申请号:PT01273519
申请日:2001-11-30
Applicant: ABBOTT LAB
Inventor: CLAIBORNE AKIYO K , GWALTNEY STEPHEN L II , HASVOLD LISA A , LI QUN , LI TOMGMEI , LIN NAN-HORNG , MANTEI ROBERT A , ROCKWAY TODD W , SHAM HING L , SULLIVAN GERARD M , TONG YUNSONG , WANG GARY T , WANG LE , WANG XILU
IPC: A61K31/4164 , A61K31/4178 , A61K31/426 , A61K31/4439 , A61K31/4709 , A61P35/00 , A61P43/00 , C07D233/54 , C07D233/64 , C07D277/20 , C07D277/30 , C07D401/12 , C07D405/12 , C07D409/12 , C07D233/00 , C07D401/00 , C07D405/00 , C07D409/00
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公开(公告)号:ZA200506760B
公开(公告)日:2006-06-28
申请号:ZA200506760
申请日:2005-08-23
Applicant: ABBOTT LAB
Inventor: HASVOLD LISA A , LI GAOQUAN , SHAM HING , SULLIVAN GERARD M , XIA PING , HEXAMER LAURA , LIN NAN-HORNG , SOWIN TOM , WANG LE
IPC: A61K20060101 , A61P20060101 , C07D20060101
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公开(公告)号:DE60118955D1
公开(公告)日:2006-05-24
申请号:DE60118955
申请日:2001-11-30
Applicant: ABBOTT LAB
Inventor: CLAIBORNE K , GWALTNEY L , HASVOLD A , LI QUN , LI TOMGMEI , LIN NAN-HORNG , MANTEI A , ROCKWAY W , SHAM L , SULLIVAN M , TONG YUNSONG , WANG T , WANG LE , WANG XILU , WANG WEIBO
IPC: C07D233/64 , A61K31/4164 , A61K31/4178 , A61K31/426 , A61K31/4439 , A61K31/4709 , A61P35/00 , A61P43/00 , C07D233/54 , C07D277/20 , C07D277/30 , C07D401/12 , C07D405/12 , C07D409/12
Abstract: Substituted imidazoles and thiazoles having the formula are useful for inhibiting farnesyltransferase. Also disclosed are farnesyltransferase-inhibiting compositions and methods of inhibiting farnesyltransferase in a patient.
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