-
61.
公开(公告)号:AU2007220889A1
公开(公告)日:2007-09-07
申请号:AU2007220889
申请日:2007-02-16
Applicant: ABBOTT LAB
Inventor: FICKES MICHAEL G , SUN MINGHUA , ZHAO CHEN , SHEIKH AHMAD Y , HENRY RODGER F , BARNES DAVID M , GREGG ROBERT J , HAIGHT ANTHONY R , KOLACZKOWSKI LAWRENCE , WITTENBERGER STEVEN J , ZHANG GEOFF G Z , COWART MARLON D , LOU XIAOCHUN , ZHENG GUO ZHU , BLACK LAWRENCE A , CHANG SOU-JEN
IPC: C07D487/04 , A61K31/407
Abstract: Octahydro-pyrrolo[3,4-b]pyrrole derivatives are useful in treating conditions or disorders prevented by or ameliorated by histamine-3 receptor ligands. Octahydro-pyrrolo[3,4-b]pyrrole compounds, methods for using such compounds, compositions for making them, and processes for preparing such compounds are disclosed herein.
-
公开(公告)号:MX2007000948A
公开(公告)日:2007-04-16
申请号:MX2007000948
申请日:2005-07-08
Applicant: ABBOTT LAB
Inventor: BUCKLEY MICHAEL J , JI JIANGUO , ROBBINS TIMOTHY A , WITTENBERGER STEVEN J , HENRY RODGER F , WAYNE GREG S , ZHANG GEOFF G , WANG WEILI W , LI WENKE , TOWNE TIMOTHY B , HANNICK STEVEN M , KOTECKI BRIAN J , MARCI BRYAN S
IPC: A61K31/4439 , C07D487/04
Abstract: La presente invencion describe (1s, 5s)-3-(5, 6-dicloro-3 -piridinil)-3, 6-diazabiciclo [3.2.0] heptano, sales del mismo, y su uso en tratar dolor y otros trastornos con el receptor de la aceticolina nicotinica.
-
63.
公开(公告)号:CZ296660B6
公开(公告)日:2006-05-17
申请号:CZ253798
申请日:1997-02-12
Applicant: ABBOTT LAB
Inventor: WINN MARTIN , BOYD STEVEN A , HUTCHINS CHARLES W , JAE HWAN-SOO , TASKER ANDREW S , VON GELDERN THOMAS W , KESTER JEFFREY A , SORENSEN BRYAN K , SZCZEPANKIEWICZ BRUCE G , HENRY KENNETH J , LIU GANG , WITTENBERGER STEVEN J , KING STEVEN A
IPC: C07D405/04 , A61K31/34 , A61K31/395 , A61K31/40 , A61K31/4015 , A61K31/4025 , A61K31/4035 , A61K31/41 , A61K31/415 , A61K31/4164 , A61K31/4166 , A61K31/421 , A61K31/425 , A61K31/435 , A61K31/4439 , A61K31/454 , A61K31/495 , A61K31/506 , A61K31/675 , A61P1/00 , A61P1/04 , A61P7/02 , A61P9/00 , A61P9/04 , A61P9/10 , A61P9/12 , A61P11/00 , A61P11/06 , A61P13/12 , A61P25/06 , A61P35/00 , A61P43/00 , C07D207/16 , C07D211/60 , C07D401/04 , C07D403/04 , C07D405/12 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14 , C07D419/14 , C07D453/02 , C07D471/04 , C07D491/04 , C07F9/572
Abstract: Benzo-1,3-dioxolyl- a benzofuranyl-substituované pyrrolidinové deriváty vzorce I nebo jejich farmaceuticky prijatelné soli, farmaceutický prostredek a jejich pouzití k výrobe léciva pro antagonizaci endothelinu a lécbe hypertenze, mestnavého selhánísrdce, aterosklerózy, rakoviny prostaty, atd. Resení se také týká meziproduktu vzorce II.
-
公开(公告)号:CA2573688A1
公开(公告)日:2006-02-23
申请号:CA2573688
申请日:2005-07-08
Applicant: ABBOTT LAB
Inventor: HANNICK STEVEN M , HENRY RODGER F , ROBBINS TIMOTHY A , WAYNE GREG S , WITTENBERGER STEVEN J , WANG WEILI W , LI WENKE , TOWNE TIMOTHY B , MARCI BRYAN S , BUCKLEY MICHAEL J , KOTECKI BRIAN J , ZHANG GEOFF G , JI JIANGUO
IPC: C07D487/04 , A61K31/4439
Abstract: The present invention discloses (1S,5S)-3-(5,6-dichloro-3-pyridinyl)-3,6-diazabicyclo[3.2.0]heptane, salts thereof, and its use to treat pain and other disorders associated with the nicotinic acetylcholine receptor.
-
公开(公告)号:TR200501137T2
公开(公告)日:2005-12-21
申请号:TR200501137
申请日:1998-07-27
Applicant: ABBOTT LAB
Inventor: WINN MARTIN , BOYD STEVEN A , HUTCHINS CHARLES W , JAE HWAN-SOO , TASKER ANDREW S , GELDERN THOMAS W VON , KESTER JEFFREY A , SORENSEN BRYAN K , SZCZEPANKIEWICZ BRUCE G , HENRY KENNETH J , LIU GANG , WITTENBERGER STEVEN J , KING STEVEN A
IPC: C07D491/048 , A61K31/40 , A61K31/41 , A61K31/423 , A61K31/435 , A61K31/4355 , A61K31/495 , A61K31/506 , A61K31/535 , A61K31/55 , A61P1/00 , A61P1/04 , A61P7/02 , A61P9/08 , A61P9/10 , A61P9/12 , A61P9/14 , A61P13/08 , A61P13/12 , A61P21/00 , A61P21/04 , A61P25/06 , A61P35/00 , A61P43/00 , C07D207/16 , C07D207/26 , C07D207/27 , C07D403/04 , C07D405/00 , C07D405/04 , C07D405/14 , C07D413/14 , C07D417/14 , C07D491/056
-
公开(公告)号:PT1272500E
公开(公告)日:2005-09-30
申请号:PT00942860
申请日:2000-06-15
Applicant: ABBOTT LAB
Inventor: COOPER ARTHUR J , HAIGHT ANTHONY R , KU YI-YIN , MORTON HOWARD E , PLATA DANIEL J , STONER ERIC J , PETERSON MATTHEW J , CINK RUSSELL D , DESHPANDE MAHENDRA N , TIM GRIEME , HILL DAVID R , CHI-PING HSU MARGARET , KING STEVEN A , LEANNA MARVIN R , LEE ELAINE C , MCLAUGHLIN MAUREEN A , NAPIER JAMES J , RAJE PRASAD S , MICHAEL RASMUSSEN , DAVID RILEY , TIEN JIEN-HEH J , WITTENBERGER STEVEN J
-
公开(公告)号:PL360183A1
公开(公告)日:2004-09-06
申请号:PL36018301
申请日:2001-03-30
Applicant: ABBOTT LAB
Inventor: HILL DAVID R , HSIAO CHI-NUNG , KURUKULASURIYA RAVI , WITTENBERGER STEVEN J
IPC: C07D233/74 , C07C239/10 , C07C259/06 , C07D277/34 , C07D317/28 , C07C231/02 , C07D233/66 , C07D317/14
Abstract: The instant invention provides a process for the selective N-formylation of N-hydroxylamines.
-
公开(公告)号:BR0108622A
公开(公告)日:2004-06-15
申请号:BR0108622
申请日:2001-03-30
Applicant: ABBOTT LAB
Inventor: HILL DAVID R , HSIAO CHI-NUNG , KURUKULASURIYA RAVI , WITTENBERGER STEVEN J
IPC: C07D233/74 , C07C239/10 , C07C259/06 , C07D277/34 , C07D317/28 , C07C231/02
Abstract: The instant invention provides a process for the selective N-formylation of N-hydroxylamines.
-
公开(公告)号:HU0302004A2
公开(公告)日:2003-09-29
申请号:HU0302004
申请日:2001-03-30
Applicant: ABBOTT LAB
Inventor: HILL DAVID R , HSIAO CHI-NUNG , KURUKULA-SURIYA RAVI , WITTENBERGER STEVEN J
IPC: C07D233/74 , C07C239/10 , C07C259/06 , C07D277/34 , C07D317/28 , C07C231/02
Abstract: The instant invention provides a process for the selective N-formylation of N-hydroxylamines.
-
公开(公告)号:NO20024678L
公开(公告)日:2002-09-30
申请号:NO20024678
申请日:2002-09-30
Applicant: ABBOTT LAB
Inventor: HILL DAVID R , HSIAO CHI-NUNG , KURUKULA-SURIYA RAVI , WITTENBERGER STEVEN J
IPC: C07D233/74 , C07C239/10 , C07C259/06 , C07D277/34 , C07D317/28 , C07C231/02
Abstract: The instant invention provides a process for the selective N-formylation of N-hydroxylamines.
-
-
-
-
-
-
-
-
-